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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T76288 | GPR | ||
GPR, a tripeptide, shows promise in Alzheimer's disease (AD) research by protecting cultured rat hippocampal neurons from amyloid-beta (Aβ)-induced death through the inhibition of caspase-3/p53-dependent apoptosis. | |||
T36951 | N-(p-Tosyl)-GPR-pNA acetate | Others | |
N-(p-Tosyl)-GPR-pNA acetate is a colorimetric substrate for thrombin that can act as a measure of thrombin activity. | |||
TP1026 | Tos-Gly-Pro-Arg-ANBA-IPA | tos-GPR-ANBA-IPA | |
Tos-Gly-Pro-Arg-ANBA-IPA is a chromogenic peptide substrate. Tos-Gly-Pro-Arg-ANBA-IPA is used for the rapid and specific photometric assay of recombinant hirudin (r-hirudin). | |||
TP1025 | Tos-Gly-Pro-Arg-ANBA-IPA acetate | tos-GPR-ANBA-IPA acetate | |
Tos-Gly-Pro-Arg-ANBA-IPA (acetate) is a peptide substrate for luminescence measurement. | |||
T11458 | GPR40/FFAR1 modulator 1 | GPR | |
GPR40/FFAR1 modulator 1 is a Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1) agonist and allosteric modulator. | |||
T9975 | GPR183 | 3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide | Others |
GPR183 (3-(3,4-difluorophenyl)-N-[3-fluoro-5-(morpholin-4-yl)phenyl]propanamide) is a chemotactic receptor known for its role in the maturation of B cells, and the endogenous ligand is the oxysterol 7α,25-dihydroxycholes... | |||
T23434 | GPR35 agonist 2 | TC-G 1001 | GPR , Arrestin |
GPR35 agonist 2 (TC-G 1001) is a potent GPR35 agonist.The EC50 values of GPR35 agonist 2 in the β-arrestin and Ca2+ release assays were 26 and 3.2 nM, respectively. | |||
T15413 | GPR120 Agonist 3 | GPR120-IN-1 | GPR |
GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62). | |||
T4312 | GPR120 Agonist 2 | GPR120 receptor agonist | GPR |
GPR120 Agonist 2 is a potent and selective GPR120 receptor agonist. | |||
T11455 | GPR35 agonist 1 | Others | |
GPR35 agonist 1 is a highly effective and specific GPR35/CXCR8 agonist (EC50: 5.8 nM). | |||
T15267 | GPR40 agonist 4 | Others | |
GPR40 agonist 4 is a potent free fatty acid agonist of receptor 1 (pEC50: 7.54). | |||
T11453 | GPR120 modulator 1 | Others | |
GPR120 modulator 1 is useful for modulating GPR120. | |||
T11452 | GPR120 Agonist 1 | GPR | |
GPR120 Agonist 1 is a selective GPR120 agonist. In GPR120 transfected HEK293 cells, GPR120 Agonist 1 displays good EC50 of 42 nM and 77 nM for human and mouse GPR120 (the calcium flux assay), respectively. | |||
T11460 | GPR4 antagonist 1 | GPR | |
GPR4 antagonist 1 is a GPR4 antagonist (IC50: 189 nM). | |||
T11456 | GPR40 Activator 1 | Others | |
GPR40 Activator 1 is a potent GPR40 activator for treatment of type 2 diabetes. | |||
T11457 | GPR40 Activator 2 | Others | |
GPR40 Activator 2 is a highly effective activator of the GPR40 receptor. | |||
T11462 | GPR84 antagonist 8 | GPR | |
GPR84 antagonist 8 is a selective GPR84 antagonist. | |||
T10507 | GPR40 Agonist 2 | GPR | |
GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of diabetes. | |||
T11459 | GPR40 agonist 1 | Others | |
GPR40 agonist 1 is an effective new GPR40 agonist (EC50s: 17 nM and 2 nM for rGPR40 and hGPR40). | |||
T11454 | GPR120 modulator 2 | Others | |
GPR120 modulator 2 is useful for modulating GPR120. |