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Search Results for "��-synuclein"

Compounds

Cat No. Product Name
T61404 α-Synuclein inhibitor 3
α-Synuclein inhibitor 3 (Compound 7g) is a potent inhibitor of α-synuclein (α -Syn) aggregation. It has potential applic...
T61611 α-Synuclein inhibitor 4
α-Synuclein inhibitor 4 (compound 3gh) is a highly effective and blood-brain barrier-permeable inhibitor of α-Synuclein ...
T61644 α-Synuclein inhibitor 6
α-Synuclein inhibitor 6 (compound 3ge) is a highly effective and blood-brain barrier-permeable inhibitor that targets th...
TMPY-06318 Human alpha-Synuclein Protein (H50Q)
T40541 α-Synuclein (61-75)
α-Synuclein (61-75) is a peptide fragment derived from the larger protein α-Synuclein. α-Synuclein is predominantly foun...
T61920 α-Synuclein inhibitor 7
α-Synuclein inhibitor 7 (化合物 3gf) 是有效的α-Synuclein (α-Syn)聚集的抑制剂,IC50为 1.95 μM,30 μM 处的抑制率为 85.8%。α-Synuclein inhibitor 7...
T62131 α-Synuclein inhibitor 5
α-Synuclein inhibitor 5 是一种有效的、能够透过血脑屏障的 α-Synuclein (α-Syn) 聚集的抑制剂 (IC50: 1.22 μM),在 30 μM 时的抑制率为 94.3%。
TMPY-02512 Alpha-Synuclein Protein, Human, Recombinant
T62226 Dyrk1A/α-synuclein-IN-2
Dyrk1A/α-synuclein-IN-2 (Compound b20) 是一种双重的 Dyrk1A 和α-synuclein aggregation 的抑制剂,能够作用于α-synuclein (IC50: 7.8 μM)。Dyrk1...
T76199 α-Synuclein (61-75) (TFA)
α-Synuclein(61-75) TFA 是α-Synuclein 的 61-75 片段。α-Synuclein 是一种丰富的神经元蛋白,在突触前神经末梢高度丰富。α-Synuclein 是一种帕金森氏病 (PD) 的生物标志物。
T62096 Dyrk1A/α-synuclein-IN-1
Dyrk1A/α-synuclein-IN-1 (Compound b1) 是一种双重的 Dyrk1A (IC50: 177 nM) 和 α-synuclein aggregation (IC50: 10.5 μM) 抑制剂。Dyrk1A/...
TMP-00579 Human Alpha-synuclein, Fc Tag
TMP-00580 Human Alpha-synuclein, His Tag
TMPY-06460 Alpha-Synuclein Protein, Mouse, Recombinant (His Tag), HPLC-verified
T9722 YTX-465 Stearoyl-CoA Desaturase (SCD)
YTX-465 是有效的硬脂酰辅酶 A 去饱和酶 (Ole1/SCD) 抑制剂,抑制 Ole1 和 SCD1的IC50=分别为 0.039 μM 和 30.4 μM。YTX-465在帕金森病和其他突触核蛋白病领域有研究的价值。
T5S0658 Corynoxine 柯诺辛,柯诺辛碱 Autophagy
Corynoxine 是从大叶钩藤中分离出的一种四环羟吲哚生物碱。它是一种自噬增强剂,可通过Akt/mTOR 途径促进 α-突触核蛋白的清除。
T4659 ELN484228 Others
ELN484228 是一种 α-突触核蛋白的阻断剂。α-突触核蛋白是帕金森病中的关键蛋白质。
T22026 AGK7 Others , Sirtuin
AGK7 是 sirtuin 2 (SIRT2) 抑制剂。它在体外和帕金森病果蝇模型中均能抑制多巴胺能细胞的凋亡。在帕金森病细胞模型中,它改善了 α-突触核蛋白毒性和修饰的包涵体形态
T7441 Cuminaldehyde Cuminal,Cuminic aldehyde,4-异丙基苯甲醛 Endogenous Metabolite
Cuminaldehyde 是一种具有抑制 α-突触核蛋白纤颤和细胞毒性作用的天然醛,是一种 Cuminum cyminum 的主要成分。它显示抗癌特性。
T13048 SynuClean-D SC-D Others
SynuClean-D 是一种 α-突触核蛋白聚集的抑制剂,能够破坏成熟的淀粉样蛋白原纤维,抑制原纤维繁殖,防止帕金森氏病动物模型中多巴胺能神经元的变性。
α-Synuclein inhibitor 3
T61404
synonym:
Target:
α-Synuclein inhibitor 4
T61611
synonym:
Target:
α-Synuclein inhibitor 6
T61644
synonym:
Target:
Human alpha-Synuclein Protein (H50Q)
TMPY-06318
synonym:
Target:
α-Synuclein (61-75)
T40541
synonym:
Target:
α-Synuclein inhibitor 7
T61920
synonym:
Target:
α-Synuclein inhibitor 5
T62131
synonym:
Target:
alpha-Synuclein Protein, Human, Recombinant
TMPY-02512
synonym:
Target:
Dyrk1A/α-synuclein-IN-2
T62226
synonym:
Target:
α-Synuclein (61-75) (TFA)
T76199
synonym:
Target:
Dyrk1A/α-synuclein-IN-1
T62096
synonym:
Target:
Human Alpha-synuclein, Fc Tag
TMP-00579
synonym:
Target:
Human Alpha-synuclein, His Tag
TMP-00580
synonym:
Target:
alpha-Synuclein Protein, Mouse, Recombinant (His Tag), HPLC-verified
TMPY-06460
synonym:
Target:
YTX-465
T9722
synonym:
Target:
Corynoxine
T5S0658
synonym: 柯诺辛,柯诺辛碱
Target:
ELN484228
T4659
synonym:
Target:
AGK7
T22026
synonym:
Target:
Cuminaldehyde
T7441
synonym: Cuminal,Cuminic aldehyde,4-异丙基苯甲醛
Target:
SynuClean-D
T13048
synonym: SC-D
Target:
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