Estrogen Receptor/ERR

The ERRs are orphan nuclear receptors, meaning the identity of their endogenous ligand has yet to be unambiguously determined. They are named because of sequence homology with estrogen receptors, but do not appear to bind estrogens or other tested steroid hormones.There are three human estrogen related receptors:ERRα,ERRβand ERRγ .

Cat. No.	Product name	CAS No.	Purity
T6827	Endoxifen Z-isomer hydrochloride	1032008-74-4	98%
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
T6404	Bazedoxifene hydrochloride	198480-56-7	98%
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
T20625	Prochloraz	67747-09-5	98%
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
T3645	Endoxifen E-isomer hydrochloride	1197194-61-8	98%
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
T13542	α-Zearalenol	36455-72-8	98%
α-Zearalenol is a Mycotoxin with a high affinity for the estrogen receptors. Due to xenoestrogen effects, it causes reproductive disorders in animals.
T21897L	MPP hydrochloride		98%
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
T7389	G15	1161002-05-6	98%
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
T1579	Mestranol	72-33-3	98%
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
TN1768	Iriflophenone	52591-10-3	98%
Standard reference
T8370	GSK5182	877387-37-6	98%
GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)
T15788	LSZ-102	2135600-76-7	98%
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
T39710	ARV-471	2229711-68-4	98%
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
T5S0543	Isocurcumenol	24063-71-6	98%
1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).
T0035	Dienestrol	84-17-3	98%
Dienestrol is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the vagina and m...
T2544	Bazedoxifene acetate	198481-33-3	98%
Bazedoxifene acetate is a novel selective estrogen receptor modulator (SERM).
T5835	PROTAC ERRα ligand 2	2306388-57-6	98%
PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)
T5531	GSK-4716	101574-65-6	98%
GSK4716 is an ERRβ/γ agonist (IC50 = 2 µM) that can activate the receptor with similar potency as the protein ligand
T5624	Bisphenol B	77-40-7	98%
Bisphenol B has a binding affinity for estrogen receptors.
T7299	β-Estradiol 17-acetate	1743-60-8	98%
beta-estradiol 17-acetate is a metabolite of estradiol.
T7313	Enclomiphene citrate	7599-79-3	98%
Enclomiphene citrate is a non-steroidal estrogen receptor antagonist,with antioestrogenic property

Cat. No.

Product name

CAS No.

Purity

Chemical Structure

T6827

Endoxifen Z-isomer hydrochloride

1032008-74-4

98%

Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.

T6404

Bazedoxifene hydrochloride

198480-56-7

98%

Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...

T20625

Prochloraz

67747-09-5

98%

Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...

T3645

Endoxifen E-isomer hydrochloride

1197194-61-8

98%

Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).

T13542

α-Zearalenol

36455-72-8

98%

α-Zearalenol is a Mycotoxin with a high affinity for the estrogen receptors. Due to xenoestrogen effects, it causes reproductive disorders in animals.

T21897L

MPP hydrochloride

98%

MPP hydrochloride is a selective estrogen receptor (ERR) modulator.

T7389

G15

1161002-05-6

98%

G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)

T1579

Mestranol

72-33-3

98%

Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.

TN1768

Iriflophenone

52591-10-3

98%

Standard reference

T8370

GSK5182

877387-37-6

98%

GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)

T15788

LSZ-102

2135600-76-7

98%

LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.

T39710

ARV-471

2229711-68-4

98%

ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.

T5S0543

Isocurcumenol

24063-71-6

98%

1. Isocurcumenol inhibits 5α-reductase which converts testosterone to dihydrotestosterone (DHT).

T0035

Dienestrol

84-17-3

98%

Dienestrol is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist. Estrogens can increase a normal clear discharge from the vagina and m...

T2544

Bazedoxifene acetate

198481-33-3

98%