T13674 |
Elacestrant
|
722533-56-4
|
98%
|
|
Elacestrant with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is an orally available selective estrogen receptor degrader .
|
T3645 |
Endoxifen E-isomer hydrochloride
|
1197194-61-8
|
98%
|
|
Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
|
T11237 |
Camizestrant
|
2222844-89-3
|
98%
|
|
Camizestrant is an antagonist of the estrogen receptor and can be used in studies about ER+ HER2-advanced breast cancer[1].
|
T6404 |
Bazedoxifene hydrochloride
|
198480-56-7
|
98%
|
|
Bazedoxifene HCl is a novel, non-steroidal, indole-based estrogen receptor modulator (SERM) binding to both ERα and ERβ with IC50 of 23 nM and 89 nM, respectivel...
|
T11237L |
Camizestrant TFA
|
T11237L
|
98%
|
|
Camizestrant TFA is a potent and orally active antagonist of estrogen receptor (ER).
|
T20419 |
Raloxifene
|
84449-90-1
|
98%
|
|
Raloxifene is a selective oestrogen receptor modulator. It has effects on bone and breast cancer and cardiovascular disease risk.
|
T6827 |
Endoxifen Z-isomer hydrochloride
|
1032008-74-4
|
98%
|
|
Endoxifen HCl is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.
|
T11098 |
Droloxifene
|
82413-20-5
|
98%
|
|
Droloxifene, a tamoxifen derivative, is an oral active and selective estrogen receptor modulator.Droloxifene induced p53 expression and apoptosis in McF-7 cells....
|
T10239 |
Acolbifene
|
182167-02-8
|
98%
|
|
Acolbifene is a selective antagonist of estrogen receptors with IC50s of 2 nM and 0.4 nM for estradiol-induced transcriptional activity of ERα and ERβ. Acolbifen...
|
TN1052 |
Lindleyin
|
59282-56-3
|
98%
|
|
Lindleyin is a novel phytoestrogen and might trigger many of the biological responses evoked by the physiological estrogens.
|
T36857L |
Premarin
|
481-97-0
|
98%
|
|
Premarin is an an estrogen sulfate with neuroprotective actions during traumatic brain injury.
|
T21897L |
MPP hydrochloride
|
|
98%
|
|
MPP hydrochloride is a selective estrogen receptor (ERR) modulator.
|
T12654 |
(Rac)-Acolbifene
|
151533-34-5
|
98%
|
|
(Rac)-Acolbifene is a racemic form of EM652 with anti-estrogenic and estrogenic activities.
|
T20625 |
Prochloraz
|
67747-09-5
|
98%
|
|
Prochloraz, a broad-spectrum contact imidazole fungicide, is used against several diseases in wheat, barley, and oleaginous plants but also for the treatment of ...
|
T7389 |
G15
|
1161002-05-6
|
|
|
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
|
T6533 |
Hexestrol
|
84-16-2
|
100%
|
|
Hexestrol binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.
|
T1579 |
Mestranol
|
72-33-3
|
100%
|
|
Mestranol, a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.
|
T39710 |
ARV-471
|
2229711-68-4
|
97.15%
|
|
ARV-471 is a orally active Cereblon -based estrogen receptor ( ER ) PROTAC degrader. ARV-471 is developed for the research of breast cancer.
|
T2882 |
Genistin
|
529-59-9
|
97.65%
|
|
Genistin is the major isoflavonoid of soybeans and soy products.It has been reported to possess various therapeutic effects, including anti-inflammatory and anti...
|
T15788 |
LSZ-102
|
2135600-76-7
|
97.84%
|
|
LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.
|