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Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T23535 Xanthine amine congener 96865-92-8 99.7%
Xanthine amine congener
Xanthine amine congener is an Adenosine receptor antagonist.
T37793 A2B receptor antagonist 2 784-90-7 100%
A2B receptor antagonist 2
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T15715 LAS101057 925676-48-8 100%
LAS101057
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
T11762 Kira8 Hydrochloride 2250019-92-0 98%
Kira8 Hydrochloride
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
T78084 PSB 0777 ammonium hydrate 98%
PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for hu...
T79027 A1/A3 AR antagonist 3 2665804-57-7 98%
A1/A3 AR antagonist 3
A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the...
T79372 A3AR agonist 1 98%
A3AR agonist 1
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective conc...
T79373 A3AR agonist 2 98%
A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. Thi...
T13008 ST3932 1246018-21-2 98%
ST3932
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T72626 A2AR-antagonist-1 2922920-71-4 98%
A2AR-antagonist-1
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability...
T16281 Nelonicline 1026134-63-3 98%
Nelonicline
Nelonicline is a selective agonist of neuronal nicotinic receptors.
TQ0136 GR79236 124555-18-6 98%
GR79236
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T16158 PF-02575799 863491-70-7 98%
PF-02575799
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
T8598 CHEMBL241987 109740-09-2 99.98%
CHEMBL241987
CHEMBL241987 targets the Adenosine receptor A3 (human)
T12161 N6-Ethyladenosine 14357-08-5 99.98%
N6-Ethyladenosine
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T0362 Ticlopidine hydrochloride 53885-35-1 99.98%
Ticlopidine hydrochloride
Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.
T6745 5-Iodotubercidin 24386-93-4 99.98%
5-Iodotubercidin
5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinas...
T0480 Doxofylline 69975-86-6 99.98%
Doxofylline
Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
T2205 Acefylline 652-37-9 99.95%
Acefylline
Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhyd...
T23336 SCH442416 316173-57-6 99.95%
SCH442416
SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.0...
Xanthine amine congener
T23535
Xanthine amine congener is an Adenosine receptor antagonist.
A2B receptor antagonist 2
T37793
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
LAS101057
T15715
LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.
Kira8 Hydrochloride
T11762
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
PSB 0777 ammonium hydrate
T78084
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for hu...
A1/A3 AR antagonist 3
T79027
A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the...
A3AR agonist 1
T79372
A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective conc...
A3AR agonist 2
T79373
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM. Thi...
ST3932
T13008
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
A2AR-antagonist-1
T72626
A2AR-antagonist-1 (compound 38), an orally active adenosine A2A receptor antagonist with an IC50 value of 29 nM, demonstrates anti-tumor properties and stability...
Nelonicline
T16281
Nelonicline is a selective agonist of neuronal nicotinic receptors.
GR79236
TQ0136
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
PF-02575799
T16158
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
CHEMBL241987
T8598
CHEMBL241987 targets the Adenosine receptor A3 (human)
N6-Ethyladenosine
T12161
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
Ticlopidine hydrochloride
T0362
Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.
5-Iodotubercidin
T6745
5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinas...
Doxofylline
T0480
Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofy...
Acefylline
T2205
Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist. It is combined with diphenhyd...
SCH442416
T23336
SCH442416 (SCH 442416) is an selective antagonist of adenosine A2A receptor. SCH442416 binds to human and rat A2A receptors with high affinity (Ki values are 0.0...
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TargetMol