Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T11762	Kira8 Hydrochloride	2250019-92-0	98%
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
T16281	Nelonicline	1026134-63-3	98%
Nelonicline is a selective agonist of neuronal nicotinic receptors.
T22031	ANR 94	634924-89-3	98%
ANR 94 is a potent and selective antagonist of adenosine A2A receptor (AA2AR) (hAA2AR, Ki= 46 nM).
T13008	ST3932	1246018-21-2	98%
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T27629	ISAM-140	932191-62-3	98%
ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.
T16158	PF-02575799	863491-70-7	98%
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
TQ0136	GR79236	124555-18-6	98%
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T28861	ST-1535	496955-42-1	98%
ST-1535 is a neuroprotective and anti-inflammatory effects of the adenosine A(2A) receptor antagonist.
T21620	2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine	133240-06-9	98%
2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.
T16140	MRS 1754	264622-58-4	98%
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.
T23201	PSB 1115	152529-79-8	98%
human A2B adenosine receptor antagonist
T23016	MRS1220	183721-15-5	98%
MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...
T37793	A2B receptor antagonist 2	784-90-7	98%
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T29112	VPC171	1018830-99-3	98%
VPC171 is a positive allosteric modulator (PAM) of the adenosine A1 receptor (A1R).
T37792	A2A receptor antagonist 1	443103-97-7	98%
A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
T15418	GS-6201	752222-83-6	98%
GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62...
T12163	N6-(2-Phenylethyl)adenosine	20125-39-7	98%
N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.
T8613	1-Ethyl-6-aminouracil	41862-09-3
1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...
T14078	AB928	2239273-34-6	100%
AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].
T9180	LUF6096	1116652-18-6	100%
LUF6096 is a potent allosteric enhancer of the adenosine A3 receptor. LUF6096 is able to allosterically enhance agonist binding. LUF6096 shows low orthosteric af...

Cat. No.

Product name

CAS No.

Purity

Chemical Structure

T11762

Kira8 Hydrochloride

2250019-92-0

98%

Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.

T16281

Nelonicline

1026134-63-3

98%

Nelonicline is a selective agonist of neuronal nicotinic receptors.

T22031

ANR 94

634924-89-3

98%

ANR 94 is a potent and selective antagonist of adenosine A2A receptor (AA2AR) (hAA2AR, Ki= 46 nM).

T13008

ST3932

1246018-21-2

98%

ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).

T27629

ISAM-140

932191-62-3

98%

ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.

T16158

PF-02575799

863491-70-7

98%

PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).

TQ0136

GR79236

124555-18-6

98%

GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.

T28861

ST-1535

496955-42-1

98%

ST-1535 is a neuroprotective and anti-inflammatory effects of the adenosine A(2A) receptor antagonist.

T21620

2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine

133240-06-9

98%

2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine is an adenosine receptor antagonist.

T16140

MRS 1754

264622-58-4

98%

MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.

T23201

PSB 1115

152529-79-8

98%

human A2B adenosine receptor antagonist

T23016

MRS1220

183721-15-5

98%

MRS1220, a highly potent and selective human A3 adenosine receptor (hA3AR) antagonist with a Ki of 0.59 nM, has therapeutic potential for the research of disease...

T37793

A2B receptor antagonist 2

784-90-7

98%

A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).

T29112

VPC171

1018830-99-3

98%

VPC171 is a positive allosteric modulator (PAM) of the adenosine A1 receptor (A1R).

T37792

A2A receptor antagonist 1

443103-97-7

98%

A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

T15418

GS-6201

752222-83-6

98%

GS-6201 is a selective antagonist of adenosine A2B receptor. GS-6201 shows high affinity and selectivity for the human adenosine A2B receptors (Ki: 22 nM). GS-62...

T12163

N6-(2-Phenylethyl)adenosine

20125-39-7

98%

N6-(2-Phenylethyl)adenosine is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for rat and human A1.

T8613

1-Ethyl-6-aminouracil

41862-09-3

1-Ethyl-6-aminouracil is an intermediate in the synthesis of a series of new substituted Xanthines which have high affinity and selectivity for the human adenosi...

T14078

AB928

2239273-34-6

100%

AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].

T9180

LUF6096

1116652-18-6