Adenosine Receptor

The adenosine receptors are a class of purinergic G protein-coupled receptors with adenosine as the endogenous ligand. There are four known types of adenosine receptors in humans: A1, A2A, A2B and A3; each is encoded by a different gene.

Cat. No.	Product name	CAS No.	Purity
T31731	Evodenoson	844873-47-8	98%
Evodenoson is a potent and selective adenosine A2a receptor (A2aR) agonist for the treatment of eye diseases, tumors, and immune system disorders, and may be use...
T27439	GS-9667	618380-90-8	98%
GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via low...
T27509	GW-493838	253124-46-8	98%
GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...
T27323	FK-453	121524-18-3	98%
FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.
T28881	Sulmazole	73384-60-8	98%
Sulmazole is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Sulmazole has been ...
T28748	Selodenoson	110299-05-3	98%
Selodenoson is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.
T14506	BAY 60-6583	910487-58-0	98%
BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 recepto...
T27800	LAS38096	851371-22-7	98%
LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .
T10248	Adenosine antagonist-1	431040-19-6	98%
Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
T23535	Xanthine amine congener	96865-92-8	98%
Adenosine receptor antagonist
T37793	A2B receptor antagonist 2	784-90-7	98%
A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).
T11762	Kira8 Hydrochloride	2250019-92-0	98%
Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.
T13008	ST3932	1246018-21-2	98%
ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).
T16281	Nelonicline	1026134-63-3	98%
Nelonicline is a selective agonist of neuronal nicotinic receptors.
TQ0136	GR79236	124555-18-6	98%
GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.
T16158	PF-02575799	863491-70-7	98%
PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).
T8598	CHEMBL241987	109740-09-2	98%
CHEMBL241987 targets the Adenosine receptor A3 (human)
T12161	N6-Ethyladenosine	14357-08-5	98%
N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).
T6745	5-Iodotubercidin	24386-93-4	98%
5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphoryl...
T0480	Doxofylline	69975-86-6	98%
Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown...

Cat. No.

Product name

CAS No.

Purity

Chemical Structure

T31731

Evodenoson

844873-47-8

98%

Evodenoson is a potent and selective adenosine A2a receptor (A2aR) agonist for the treatment of eye diseases, tumors, and immune system disorders, and may be use...

T27439

GS-9667

618380-90-8

98%

GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia via low...

T27509

GW-493838

253124-46-8

98%

GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgia or...

T27323

FK-453

121524-18-3

98%

FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.

T28881

Sulmazole

73384-60-8

98%

Sulmazole is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.Sulmazole has been ...

T28748

Selodenoson

110299-05-3

98%

Selodenoson is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.

T14506

BAY 60-6583

910487-58-0

98%

BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3 recepto...

T27800

LAS38096

851371-22-7

98%

LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .

T10248

Adenosine antagonist-1

431040-19-6

98%

Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.

T23535

Xanthine amine congener

96865-92-8

98%

Adenosine receptor antagonist

T37793

A2B receptor antagonist 2

784-90-7

98%

A2B receptor antagonist 2 is an antagonist of adenosine receptor A2B (Ki = 2.30 μM for rA1, 6.8 μM for rA2A, 3.44 μM for hA2B).

T11762

Kira8 Hydrochloride

2250019-92-0

98%

Kira8 Hydrochloride is a mono-selective IRE1α inhibitor that allosterically attenuates IRE1α RNase activity with an IC50 of 5.9 nM.

T13008

ST3932

1246018-21-2

98%

ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).

T16281

Nelonicline

1026134-63-3

98%

Nelonicline is a selective agonist of neuronal nicotinic receptors.

TQ0136

GR79236

124555-18-6

98%

GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.

T16158

PF-02575799

863491-70-7

98%

PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).

T8598

CHEMBL241987

109740-09-2

98%

CHEMBL241987 targets the Adenosine receptor A3 (human)

T12161

N6-Ethyladenosine

14357-08-5

98%

N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).

T6745

5-Iodotubercidin

24386-93-4

98%

5-Iodotubercidin is a potent adenosine kinase inhibitor with IC50 of 26 nM. It inhibits nucleoside transporter, CK1, insulin receptor tyrosine kinase, phosphoryl...

T0480

Doxofylline

69975-86-6

98%

Doxofylline is a methylxanthine derivative with the presence of a dioxolane group in position 7. As a drug used in the treatment of asthma, doxofylline has shown...