Powder: -20°C for 3 years | In solvent: -80°C for 1 year
A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the research of chronic heart diseases [1].
Pack Size | Availability | Price/USD | Quantity |
---|---|---|---|
25 mg | 8-10 weeks | $ 1,820.00 | |
50 mg | 8-10 weeks | $ 2,380.00 | |
100 mg | 8-10 weeks | $ 3,100.00 |
Description | A1/A3 AR Antagonist 3 is a dual A1R/A3R antagonist that demonstrates high affinity within the low-micromolar to nanomolar range, and is potentially useful in the research of chronic heart diseases [1]. |
In vitro | Compound A1/A3 AR antagonist 3 (A17) exhibits binding affinity towards both A1R and A3R, with pKd values of 8.25 and 7.87, respectively [1]. Additionally, this antagonist has demonstrated binding affinity for A1R and A3R with pKi values of 8.36 and 8.01, respectively [1]. |
Molecular Weight | 401.42 |
Formula | C22H19N5O3 |
CAS No. | 2665804-57-7 |
Powder: -20°C for 3 years | In solvent: -80°C for 1 year
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A1/A3 AR antagonist 3 2665804-57-7 GPCR/G Protein Neuroscience Adenosine Receptor inhibitor inhibit