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Results for "

adrenoceptor antagonist

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    118
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    2
    TargetMol | Peptide_Products
  • Dye Reagents
    1
    TargetMol | Dye_Reagents
  • Natural Products
    4
    TargetMol | Natural_Products
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    2
    TargetMol | Isotope_Products
5-HT2 antagonist 1
T12597191592-09-3In house
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist with weak α1 adrenoceptor blocking activity.
  • Inquiry Price
6-8 weeks
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QTY
TargetMol | Inhibitor Hot
Cicloprolol hydrochloride
T1081263686-79-3In house
Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.
  • Inquiry Price
6-8 weeks
Size
QTY
Midaglizole hydrochloride
(±)-DG5128 hydrochloride, DG5128 hydrochloride
T1101579689-25-1In house
Midaglizole hydrochloride ((±)-DG5128) (DG5128) is a preferred α2-adrenoceptor antagonist. Midazolazole hydrochloride (DG5128) has an affinity for α2-adrenoceptor (pKi = 6.28) 7.4 times higher than that of α1-adrenoceptor.
  • Inquiry Price
6-8 weeks
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QTY
TargetMol | Inhibitor Sale
Fiduxosin
ABT 980, A 185980.1
T11286208993-54-8In house
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with Ki values of 0.160 nM, 24.9 nM and 0.920 nM, respectively. Fiduxosin can be used for the treatment of benign prostatic hyperplasia.
  • Inquiry Price
8-10 weeks
Size
QTY
L-771688
SNAP 6383
T15688200050-59-5In house
L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benign prostatic hyperplasia.
  • Inquiry Price
6-8 weeks
Size
QTY
Pamatolol
T1643159110-35-9In house
Pamatolol is a selective and potent beta-adrenoceptor antagonist that has not shown sympathomimetic activity in ex vivo experiments.
  • Inquiry Price
6-8 weeks
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QTY
RS 17053 hydrochloride
RS-17053
T16798169505-93-5In house
RS 17053 hydrochloride is a potent and selective antagonist of the α1A adrenoceptor, with a pKi value of 9.1 in native cell membranes and a pA2 value of 9.8 in functional assays.
  • Inquiry Price
6-8 weeks
Size
QTY
jp1302
T2288280259-18-3In house
JP1302 is a selective α2C adrenoceptor antagonist with a Kb value of 16 nM and a Ki of 28 nM for human α2C receptors.JP1302 has antidepressant activity, disrupts the FACT complex and degrades histone H1.JP1302 has been used in the study of neuropsychiatric disorders, acute renal failure, and renal injury.
  • Inquiry Price
6-8 weeks
Size
QTY
Monatepil maleate
AJ2615 maleate, AJ-2615 maleate, AJ 2615 maleate
T25828103379-03-9In house
Monatepil maleate (AJ-2615 maleate) is an orally active Ca2+-channel and α1-adrenoceptor antagonist and non-competitive heparanoyl-coenzyme A:cholesterol acyltransferase (ACAT) inhibitor with antihypertensive activity.Monatepil maleate is used in studies of hyperlipidemia and atherosclerosis. Monatepil maleate is used to study hyperlipidemia and atherosclerosis.
  • Inquiry Price
6-8 weeks
Size
QTY
Bunazosin Hydrochloride
E-643, E643, E-1015, E 643, E 1015
T2692352712-76-2In house
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.
  • Inquiry Price
6-8 weeks
Size
QTY
TargetMol | Inhibitor Sale
orm-10921
ORM10921, ORM 10921
T28267610782-82-6In house
ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.
  • Inquiry Price
6-8weeks
Size
QTY
TargetMol | Inhibitor Sale
Taprizosin
UK-338003, UK338003, UK-338,003, UK 338003, Taprizosin Mesylate
T28922210538-44-6In house
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.
  • Inquiry Price
6-8weeks
Size
QTY
TargetMol | Inhibitor Sale
CGP-20712
UNII-SIO2UEZ19H, CGP 20712
T30846137888-49-4In house
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
  • Inquiry Price
8-10weeks
Size
QTY
Neldazosin
T61535109713-79-3In house
Neldazosin is used as a potent α1-adrenoceptor antagonist.
  • Inquiry Price
6-8weeks
Size
QTY
SM-2470
T6289399899-45-3In house
SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity that decreases anterior ganglionic adrenal nerve activity and aortic descending nerve activity.SM-2470 has hypocholesterolemic activity and inhibits cholesterol absorption.
  • Inquiry Price
6-8 weeks
Size
QTY
Tolnapersine
T6802370312-00-4In house
Tolnapersine is a mixed dopamine agonist and alpha-adrenoceptor antagonist.
  • Inquiry Price
1-2 weeks
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Midaglizole
DG5128 free base, (±)-DG5128 free base
T6809866529-17-7In house
Midaglizole ((±)-DG5128 free base, DG5128 free base) is a potent α2-adrenoceptor antagonist that acts as a hypoglycemic agent by lowering blood glucose levels and increasing blood pressure in vivo.
  • Inquiry Price
1-2 weeks
Size
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Saterinone
T68138102669-89-6In house
Saterinone is a potent and selective phosphodiesterase III inhibitor and a potent antagonist of the vascular α-1-adrenoceptor. Saterinone has vasodilatory properties and can be used in the acute treatment of chronic heart failure. Saterinone inhibited crude cAMP phosphodiesterase (PDE) activity in guinea pig right ventricular homogenates The ic50 value is 2.3 × 10(-5) mol l.
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β2AR/M-receptor agonist-2
T722261017857-38-3In house
β2AR M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA). It demonstrates significant activity towards the β2 adrenoceptor with an EC50 of 3.7 nM and exhibits affinity for the human cloned M3 receptor with a Ki of 0.73 nM. This potent bronchodilator holds potential for research in chronic obstructive pulmonary disease (COPD) treatment.
  • Inquiry Price
7-10 days
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Fluparoxan hydrochloride
T77565105227-44-9In house
Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental disorders and neurodegenerative diseases.
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Urapidil hydrochloride
Urapidil HCl
T008864887-14-5
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
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Naftopidil
KT-611, BM-15275
T069657149-07-2
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-blocker.
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Phenoxybenzamine hydrochloride
NCI-c01661, NSC 37448, Phenoxybenzamine HCl
T115863-92-3
Phenoxybenzamine hydrochloride (NCI-c01661) is the hydrochloride salt form of phenoxybenzamine, a synthetic, dibenzamine alpha-adrenergic antagonist with antihypertensive and vasodilatory properties. Phenoxybenzamine non-selectively and irreversibly blocks the postsynaptic alpha-adrenergic receptor in smooth muscle, thereby preventing vasoconstriction, relieving vasospasms, and decreasing peripheral resistance. Reflex tachycardia may occur and may be enhanced by blockade of alpha-2 receptors which enhances norepinephrine release. Phenoxybenzamine is reasonably anticipated to be a human carcinogen.
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Atipamezole hydrochloride
MPV-1248 hydrochloride, Antisedan
T6765104075-48-1
Atipamezole is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug. Atipamezole hydrochloride (MPV-1248 hydrochloride) is hydrochloride form of atipamezole.
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