Search Result

Search Results for " pdgfr "

Targets

Libraries

FDA-Approved Kinase Inhibitor Library Kinase Inhibitor Library

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Compounds

Cat No.	Product Name
T60108	PDGFR Tyrosine Kinase Inhibitor III	PDGF Receptor Tyrosine Kinase Inhibitor III	PDGFR
	PDGFR Tyrosine Kinase Inhibitor III (PDGF Receptor Tyrosine Kinase Inhibitor III) is a multikinase inhibitor that inhibi...		PDGFR
T62872	PDGFR-IN-1
	PDGFR-IN-1 (compound 7m) is an orally active PDGFR (platelet-derived growth factor receptor) inhibitor that acts on PDGF...
T4332	C-Kit-IN-1	PDGFR inhibitor 1,DCC-2618	c-Met/HGFR , c-Kit
	DCC-2618 is an effective inhibitor of c-Met and c-Kit (IC50s<200 nM).		c-Met/HGFR , c-Kit
TQ0003	740 Y-P	PDGFR 740Y-P,740YPDGFR	PI3K , Autophagy
	740 Y-P is a potent and cell-permeable activator of PI3K.		PI3K , Autophagy
TQ0003L1	740 Y-P acetate	PDGFR 740Y-P Acetate,740 Y-P acetate(1236188-16-1 Free base),740YPDGFR acetate	PI3K
	740 Y-P acetate is a potent and cell-permeable PI3K activator.740 Y-P acetate tends to bind to GST fusion proteins conta...		PI3K
T6091	CP-673451		PDGFR , c-Kit , VEGFR
	CP-673451 is a specific inhibitor of PDGFRα/β (IC50: 10/1 nM) with antiangiogenic and antitumor activity and the selecti...		PDGFR , c-Kit , VEGFR
T14137	AG 1295		PDGFR
	AG 1295 is a selective platelet-derived growth factor receptor (PDGFR) tyrosine-kinase inhibitor. AG1295 abolishes autop...		PDGFR
T2734	Sennoside B		PDGFR
	Sennoside B is an anthranoid. Anthranoid derivatives are used all over the world as a treatment for constipation.		PDGFR
TQ0003L	740 Y-P(TFA)(1236188-16-1 free base)	740YPDGFR(TFA),740 Y-P(TFA),PDGFR 740Y-P(TFA)	PI3K
	740 Y-P(TFA) is a potent and cell-permeable activator of PI3K.		PI3K
T5109	Avapritinib	BLU-285	PDGFR , c-Kit
	Avapritinib is a dual inhibitor of the mutant KIT receptor (KIT D816V, IC50: 0.27 nM) and PDGFRα (PDGFRα D842V, IC50: 0....		PDGFR , c-Kit
T16975	TAK-593		PDGFR , VEGFR
	TAK-593 is an effective VEGFR and PDGFR family inhibitor (IC50s: 3.2, 0.95, 1.1, 4.3, and 13 nM for VEGFR1, VEGFR2, VEGF...		PDGFR , VEGFR
T4320	Flumatinib	HHGV678	c-Kit , PDGFR , Bcr-Abl
	Flumatinib is an orally bioavailable tyrosine kinase inhibitor flumatinib, with potential antineoplastic activity.		c-Kit , PDGFR , Bcr-Abl
T3570	SU4312	NSC 86429,SU 4312	PDGFR , VEGFR
	SU-4312, also known as DMBI, is a potent and selective inhibitor of VEGFR and PDGFR tyrosine kinases (IC50 values are 0....		PDGFR , VEGFR
T6932	PD168393		FGFR , EGFR , Autophagy , IGF-1R , PKC , PDGFR , Apoptosis
	PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, FGFR, P...		FGFR , EGFR , Autophagy , IGF-1R , PKC , PDGFR , Apoptosis
T3476	JI-101	JI 101,CGI-1842	PDGFR , Ephrin Receptor , VEGFR
	JI-101 is an oral multi-kinase inhibitor that targets vascular endothelial growth factor receptor type 2 (VEGFR-2), plat...		PDGFR , Ephrin Receptor , VEGFR
TN1969	N-(p-Coumaroyl) serotonin		PDGFR
	N-(p-Coumaroyl) Serotonin is a polyphenol isolated from the seeds of safflower. N-(p-Coumaroyl) serotonin has antioxidan...		PDGFR
T8900	Seralutinib	GB002	PDGFR
	Seralutinib is an inhibitor of inhaled PDGFRα and PDGFRβ. It is used in the study for pulmonary arterial hypertension.		PDGFR
T7945	SU14813		PDGFR , c-Kit , VEGFR
	SU14813 is a multi-receptor tyrosine kinase inhibitor with potent antiangiogenesis and antitumor activity (IC50s of 50, ...		PDGFR , c-Kit , VEGFR
T6996	SU 5402	SU5402	PDGFR , FGFR , VEGFR
	SU5402 is a potent multi-targeted receptor tyrosine kinase inhibitor with IC50 of 20 nM, 30 nM, and 510 nM for VEGFR2, F...		PDGFR , FGFR , VEGFR
T0080	Trapidil	AR-12008,Avantrin,Rocornal,Trapymin,Trapymine	PDGFR , PDE
	Trapidil is a coronary vasodilator agent. It was originally developed as a vasodilator and anti-platelet agent and has b...		PDGFR , PDE