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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T9345 | Aminopeptidase M | Others | |
Aminopeptidase M (AMP) inhibition is of interest for several diseases, such as highly vascularized cancer types. | |||
T61278 | Aminopeptidase-IN-1 | Aminopeptidase | |
Aminopeptidase-IN-1 is a potent inhibitor of insulin-regulated aminopeptidase (IRAP) (Ki: 7.7 μM).Aminopeptidase-IN-1 can be used in studies of cognitive and memory disorders. | |||
T36943 | Aminopeptidase N Inhibitor | ||
Aminopeptidase N (AP-N) inhibitor is a reversible inhibitor of AP-N/CD13 (IC50 = 25 μM). It is selective for AP-N/CD13 over matrix metalloproteinase-9 (MMP-9), angiotensin converting enzyme (ACE), neutral endopeptidase (... | |||
T76568 | Aminopeptidase N Ligand (CD13) NGR peptide | ||
Aminopeptidase N Ligand (CD13) NGR peptide, a polypeptide that targets CD13, functions as a carrier for mediating intracellular transmission and is commonly utilized in cancer research [1] [2]. | |||
TQ0047 | DG051 | Aminopeptidase | |
DG051 is a potent leukotriene A4 hydrolase (LTA4H) inhibitor (IC50: 47 nM). | |||
T1257 | Bestatin | Ubenimex | Others , Aminopeptidase , Antibacterial , Antibiotic , LTR |
Bestatin (Ubenimex) competitively inhibits many aminopeptidases, including B, N and leucine aminopeptidases. Ubenimex is a microbial metabolite and dipeptide with potential immunomodulatory and antitumor activities. Amin... | |||
T11221 | ERAP1-IN-1 | Others | |
ERAP1-IN-1 is an endoplasmic reticulum aminopeptidase 1 (ERAP1) inhibitor. ERAP1-IN-1 allosterically activates ERAP1’s hydrolysis of fluorogenic and chromogenic amino acid substrates but competitively inhibits its activi... | |||
T6301 | Tosedostat | CHR-2797 | Aminopeptidase , AChR |
Tosedostat (CHR-2797) is an orally bioavailable inhibitor of the M1 family of aminopeptidases with potential antineoplastic activity. Tosedostat is converted intracellularly into a poorly membrane-permeable active metabo... | |||
T3715 | Acebilustat | CTX-4430 | Aminopeptidase , LTR |
Acebilustat (CTX-4430) (ZK322) is an effective and specific leukotriene B4 hydrolase inhibitor. | |||
T21859 | ARM1 | Aminopeptidase , Epoxide Hydrolase | |
ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase. | |||
T7958 | Methyl arachidate | Methyl Icosanoate | Others , Aminopeptidase |
Methyl arachidate (Methyl Icosanoate) is an esterified form of arachidic acid | |||
T3529 | Bestatin hydrochloride | Ubenimex hydrochloride | Integrin , Aminopeptidase , Antibacterial , Antibiotic |
Bestatin hydrochloride (Ubenimex hydrochloride) is an inhibitor of aminopeptidase N (APN)/CD13 and aminopeptidase B. | |||
T16684 | Puromycin aminonucleoside | NSC 3056 | Apoptosis , Proteasome , Aminopeptidase , Antibacterial , Antibiotic |
Puromycin aminonucleoside (NSC-3056) increases podocyte permeability by modulating ZO-1 in an oxidative stress-dependent manner. | |||
T21696 | SC-57461A | Aminopeptidase | |
SC 57461A is a potent and specific leukotriene A4 hydrolase (LTA4H) inhibitor. | |||
T28482 | Firibastat | QGC 001,QGC-001,RB-150,RB150,QGC001,RB 150 | Aminopeptidase |
Firibastat (RB150) is a glutamyl aminopeptidase antagonist and an orally active brain penetrating prodrug of EC33. It is a first-in-class brain aminopeptidase A (APA) inhibitor with a Ki of 200 nM. Firibastat selectively... | |||
T5652 | L(+)-Leucinol | Aminopeptidase | |
L(+)-Leucinol is a potent inhibitor of leucine aminopeptidase. | |||
T18997 | GPDA | Glycylproline p-nitroanilide tosylate,GPN | Others |
GPDA (Glycylproline p-nitroanilide tosylate) is a substrate of X-Prolyl dipeptidyl-aminopeptidase in the enzyme assay. | |||
TP1181 | Bradykinin (2-9) | Des-Arg1-bradykinin | Bradykinin Receptor |
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin. It is formed by the cleavage action of Aminopeptidase P. | |||
T60021 | EcMetAP-IN-1 | Others | |
ecMetAP-IN-1 can be used as a QSAR model to study methionine aminopeptidase inhibitor as an anticancer agent using multiple linear regression. | |||
T64341 | H-β-Ala-AMC TFA | Others | |
H-β-Ala-AMC TFA is a substrate for aminopeptidase. Building block for synthesizing the fluorogenic vanin I substrate pantothenate-AMC. |