TN1663 |
Ganoderic acid DM
|
173075-45-1
|
98%
|
|
Ganoderic acid DM is an antiandrogenic osteoclastogenesis inhibitor, it especially suppresses the expression of c-Fos and nuclear factor of activated T cells c1 ...
|
TN1061 |
Ganoderol B
|
104700-96-1
|
98%
|
|
Ganoderol B is a potent β ±-glucosidase and angiotensin-converting enzyme inhibitor, with an IC(50) of β ±-glucosidase is 119.8 uM. It may be useful in prostate ...
|
T15749 |
LGD-2226
|
328947-93-9
|
98%
|
|
LGD-2226 is a selective and orally active androgen receptor modulator (EC50: 0.2 nM, Ki: 1.5 nM for the human androgen receptor). LGD-2226 can be used for muscle...
|
T15816 |
LY341495
|
201943-63-7
|
98%
|
|
LY341495 is an antagonist of metabotropic glutamate receptor (IC50s: 2.9 nM, 10 nM, 170 nM for mGluR-2, mGluR-3, mGluR-8, respectively).
|
T10946 |
D4-abiraterone
|
154229-21-7
|
98%
|
|
D4-Abiraterone is an inhibitor of CYP17A1, 3b-hydroxysteroid dehydrogenase (3βHSD) and steroid 5a-reductase (SRD5A), the main metabolite of abiraterone. D4-Abira...
|
TN4774 |
Physalin A
|
23027-91-0
|
98%
|
|
Physalin A exerts anti-tumor activity in non-small cell lung cancer cell lines by suppressing JAK/STAT3 signaling, it inhibits androgen-independent prostate canc...
|
T14675 |
BMS-564929
|
627530-84-1
|
98%
|
|
BMS-564929 is an agonist of androgen receptor (AR, Ki of 2.11±0.16 nM).
|
T14843 |
Bifluranol
|
34633-34-6
|
98%
|
|
Bifluranol is an anti-androgen.
|
TMA1012 |
Ganoderiol F
|
114567-47-4
|
98%
|
|
Ganoderiol F has anti-inflammatory, cytotoxic and anti-HIV activity, it inhibits activity of topoisomerases in vitro, and it inhibits human immunodeficiency viru...
|
T19449 |
N-desmethyl Enzalutamide D6
|
T19449
|
98%
|
|
N-desmethyl Enzalutamide D6 is a deuterium labeled N-desmethyl Enzalutamide.
|
T0380 |
Bicalutamide
|
90357-06-5
|
99.97%
|
|
Bicalutamide, a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the receptor bind...
|
T68020 |
Zanoterone
|
107000-34-0
|
99.96%
|
|
Zanoterone is an AR antagonist (androgen receptor).Zanoterone has antitumor activity for the treatment of genitourinary disorders and oncological disorders and m...
|
T0419 |
Testosterone propionate
|
57-85-2
|
99.92%
|
|
Testosterone Propionate is a short acting oil-based injectable formulation of testosterone. Testosterone inhibits gonadotropin secretion from the pituitary gland...
|
T0489 |
Flutamide
|
13311-84-7
|
99.92%
|
|
Flutamide is an antiandrogen with about the same potency as cyproterone in rodent and canine species.
|
T9179 |
CLP-3094
|
312749-73-8
|
99.84%
|
|
CLP-3094 is a potent androgen receptor BF3 (binding function 3) inhibitor. BF3-IN-1 inhibits AR transcriptional activity with IC50 of 4 μM. CLP-3094 is a selecti...
|
TN1370 |
Allura Red AC
|
25956-17-6
|
99.82%
|
|
Allura Red AC is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to ...
|
T2236 |
RU 58841
|
154992-24-2
|
99.77%
|
|
RU 58841 is a specific androgen receptor antagonist or anti-androgen; RU 58841 has a significant effect on hair regrowth.
|
TQ0209 |
Ailanthone
|
981-15-7
|
99.71%
|
|
Ailanthone is an effective inhibitor of both full-length androgen receptor (AR) (IC50: 69 nM) and constitutively active truncated AR splice variants (IC50: 309 n...
|
T13272 |
UT-155
|
2031161-35-8
|
99.63%
|
|
UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM for UT-155 binding to AR-LBD).
|
T0476 |
Spironolactone
|
52-01-7
|
99.63%
|
|
Spironolactone is an Aldosterone Antagonist. The mechanism of action of spironolactone is as an Aldosterone Antagonist.
|