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Search Results for "carboxypeptidase"

Targets

Compounds

Cat No. Product Name
T10678 Carboxypeptidase G2 (CPG2) Inhibitor Carboxypeptidase G2 Inhibitor,CPG2 Inhibitor Carboxypeptidase
Carboxypeptidase G2 (CPG2) Inhibitor 是新型的羧肽酶 G2(CPG2)抑制剂,显示出抗癌活性。
T76167 Carboxypeptidase A
Carboxypeptidase A(EC 3.4.2.1) 是一种含锌的金属蛋白酶,常用于生化研究。Carboxypeptidase A 催化与多肽链 C 端相邻的肽键的水解。Carboxypeptidase A 是典型的金属蛋白酶,在生...
T10876 CPA inhibitor Carboxypeptidase inhibitor Carboxypeptidase
CPA inhibitor 是一种有效的羧肽酶 A (CPA) 抑制剂,Ki 值为 0.32 μM。
T76102 Carboxypeptidase B
Carboxypeptidase B 是一种肽链外切酶,可专一性地降解肽链。Carboxypeptidase B 从 C 端逐个降解,释放出游离氨基酸。Carboxypeptidase B 只水解以碱性氨基酸(如精氨酸和赖氨酸)为 C 末端...
T76168 Carboxypeptidase C
CarboxypeptidaseC 是一种羧肽酶,常用于生化研究。CarboxypeptidaseC 去除多肽链羧基末端赖氨酸、精氨酸和脯氨酸,以及所有中性、脂肪族、芳香族和肽链的酸性蛋白质氨基酸。
T3440 2-PMPA 2-(Phosphonomethyl)pentanedioic acid Carboxypeptidase
2-PMPA 是谷氨酸羧肽酶II 的选择性抑制剂(IC50:300 pM)。
T16116 MLN-4760 RAAS
MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μ...
T8093 2-Benzylsuccinic acid 2-苄基丁二酸,DL-Benzylsuccinic acid Carboxypeptidase
DL-Benzylsuccinic acid 是羧肽酶 A (CPA) 抑制剂。
T71126 Allixin
Allixin is a phytoallexin found in garlic (Allium sativum) bulbs. Allixin has weak antimicrobial activity and exerts an ...
T22497 2-MPPA Others
glutamate carboxypeptidase II (GCP II) inhibitor
T26725 AZD-9684 AZD 9684,AZD9684
AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.
T28466 PSMA-11 Psma-hbed-CC,HBED-CC-PSMA
PSMA-11通过与前列腺特异性膜抗原(PSMA)的细胞外结构域结合来检测前列腺癌的复发和转移。PSMA-11常被用作正电子发射断层扫描(PET)中用作表达PSMA 的肿瘤的示踪剂,通过静脉注射镓Ga 68标记的PSMA-11,Glu-ur...
T69327 E2072
E2072 is a potent and selective thiol-based Glutamate Carboxypeptidase II (GCP-II) inhibitor.
T25968 PMPA sodium PMPA sodium salt,PMPA Na,PMPA tetrasodium salt
PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) ...
T28842 SQ-24,798 SQ 24,798,SQ24,798
SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).
T62423 GCPII-IN-1 TFA
GCPII-IN-1 TFA 是一种谷氨酸羧肽酶 II (GCPII; PSMA) 抑制剂支架 (Ki: 44.3 nM)。
TP2076 [Phe8Ψ(CH-NH)-Arg9]-Bradykinin
Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage. 5-fold more potent and exhibits...
T38420 GCPII-IN-1
GCPII-IN-1 is a potent inhibitor scaffold targeting glutamate carboxypeptidase II (GCPII), also known as prostate-specif...
TP1747 Bradykinin (1-6)
Bradykinin (1-6) is an amino-truncated Bradykinin peptide. Bradykinin (1-6) is a stable metabolite of Bradykinin, cleave...
T75118 AN15368
AN15368 是一种具有口服活性的小分子前药,可以被寄生虫羧肽酶激活,产生一种靶向 T. cruzi.中信使 RNA 加工途径的化合物 cruzi. AN15368 具有预防和研究南美锥虫病的潜力。
Carboxypeptidase G2 (CPG2) Inhibitor
T10678
synonym: Carboxypeptidase G2 Inhibitor,CPG2 Inhibitor
Target:
Carboxypeptidase A
T76167
synonym:
Target:
CPA inhibitor
T10876
synonym: Carboxypeptidase inhibitor
Target:
Carboxypeptidase B
T76102
synonym:
Target:
Carboxypeptidase C
T76168
synonym:
Target:
2-PMPA
T3440
synonym: 2-(Phosphonomethyl)pentanedioic acid
Target:
MLN-4760
T16116
synonym:
Target:
2-Benzylsuccinic acid
T8093
synonym: 2-苄基丁二酸,DL-Benzylsuccinic acid
Target:
Allixin
T71126
synonym:
Target:
2-MPPA
T22497
synonym:
Target:
AZD-9684
T26725
synonym: AZD 9684,AZD9684
Target:
PSMA-11
T28466
synonym: Psma-hbed-CC,HBED-CC-PSMA
Target:
E2072
T69327
synonym:
Target:
PMPA sodium
T25968
synonym: PMPA sodium salt,PMPA Na,PMPA tetrasodium salt
Target:
SQ-24,798
T28842
synonym: SQ 24,798,SQ24,798
Target:
GCPII-IN-1 TFA
T62423
synonym:
Target:
[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
TP2076
synonym:
Target:
GCPII-IN-1
T38420
synonym:
Target:
Bradykinin (1-6)
TP1747
synonym:
Target:
AN15368
T75118
synonym:
Target: