T10678 |
Carboxypeptidase G2 (CPG2) Inhibitor
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Carboxypeptidase G2 Inhibitor,CPG2 Inhibitor |
Carboxypeptidase
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Carboxypeptidase G2 (CPG2) Inhibitor 是新型的羧肽酶 G2(CPG2)抑制剂,显示出抗癌活性。 |
T76167 |
Carboxypeptidase A
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Carboxypeptidase A(EC 3.4.2.1) 是一种含锌的金属蛋白酶,常用于生化研究。Carboxypeptidase A 催化与多肽链 C 端相邻的肽键的水解。Carboxypeptidase A 是典型的金属蛋白酶,在生... |
T10876 |
CPA inhibitor
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Carboxypeptidase inhibitor |
Carboxypeptidase
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CPA inhibitor 是一种有效的羧肽酶 A (CPA) 抑制剂,Ki 值为 0.32 μM。 |
T76102 |
Carboxypeptidase B
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Carboxypeptidase B 是一种肽链外切酶,可专一性地降解肽链。Carboxypeptidase B 从 C 端逐个降解,释放出游离氨基酸。Carboxypeptidase B 只水解以碱性氨基酸(如精氨酸和赖氨酸)为 C 末端... |
T76168 |
Carboxypeptidase C
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CarboxypeptidaseC 是一种羧肽酶,常用于生化研究。CarboxypeptidaseC 去除多肽链羧基末端赖氨酸、精氨酸和脯氨酸,以及所有中性、脂肪族、芳香族和肽链的酸性蛋白质氨基酸。 |
T3440 |
2-PMPA
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2-(Phosphonomethyl)pentanedioic acid |
Carboxypeptidase
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2-PMPA 是谷氨酸羧肽酶II 的选择性抑制剂(IC50:300 pM)。 |
T16116 |
MLN-4760
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RAAS
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MLN-4760 是选择性的人ACE2抑制剂,IC50=0.44 nM,对人ACE2的选择性是其他相关蛋白的 5000 多倍,包括人睾丸 ACE (IC50,>100 μM) 和牛 carboxypeptidase A (IC50,27 μ... |
T8093 |
2-Benzylsuccinic acid
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2-苄基丁二酸,DL-Benzylsuccinic acid |
Carboxypeptidase
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DL-Benzylsuccinic acid 是羧肽酶 A (CPA) 抑制剂。 |
T71126 |
Allixin
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Allixin is a phytoallexin found in garlic (Allium sativum) bulbs. Allixin has weak antimicrobial activity and exerts an ... |
T22497 |
2-MPPA
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Others
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glutamate carboxypeptidase II (GCP II) inhibitor |
T26725 |
AZD-9684
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AZD 9684,AZD9684 |
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AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis. |
T28466 |
PSMA-11
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Psma-hbed-CC,HBED-CC-PSMA |
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PSMA-11通过与前列腺特异性膜抗原(PSMA)的细胞外结构域结合来检测前列腺癌的复发和转移。PSMA-11常被用作正电子发射断层扫描(PET)中用作表达PSMA 的肿瘤的示踪剂,通过静脉注射镓Ga 68标记的PSMA-11,Glu-ur... |
T69327 |
E2072
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E2072 is a potent and selective thiol-based Glutamate Carboxypeptidase II (GCP-II) inhibitor. |
T25968 |
PMPA sodium
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PMPA sodium salt,PMPA Na,PMPA tetrasodium salt |
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PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) ... |
T28842 |
SQ-24,798
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SQ 24,798,SQ24,798 |
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SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN). |
T62423 |
GCPII-IN-1 TFA
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GCPII-IN-1 TFA 是一种谷氨酸羧肽酶 II (GCPII; PSMA) 抑制剂支架 (Ki: 44.3 nM)。 |
TP2076 |
[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
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Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage. 5-fold more potent and exhibits... |
T38420 |
GCPII-IN-1
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GCPII-IN-1 is a potent inhibitor scaffold targeting glutamate carboxypeptidase II (GCPII), also known as prostate-specif... |
TP1747 |
Bradykinin (1-6)
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Bradykinin (1-6) is an amino-truncated Bradykinin peptide. Bradykinin (1-6) is a stable metabolite of Bradykinin, cleave... |
T75118 |
AN15368
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AN15368 是一种具有口服活性的小分子前药,可以被寄生虫羧肽酶激活,产生一种靶向 T. cruzi.中信使 RNA 加工途径的化合物 cruzi. AN15368 具有预防和研究南美锥虫病的潜力。 |