avp — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T30231	AVP-13358		Others
	AVP-13358 is a CD23 antagonist (immunoglobulin ε-Fc receptor antagonist), an immunoglobulin E inhibitor. AVP-13358 has potent activity against IgE, cytokines and CD23 and is used in the treatment of immune system disorde...		Others
TP2082L	D[Cha4]-AVP acetate(500170-27-4 free base)		Vasopressin Receptor
	d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secre...		Vasopressin Receptor
TP2082	D[Cha4]-AVP
	Potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligi...
T9857	Vasopressin	antidiuretic hormone (ADH),argipressin,arginine vasopressin (AVP)	Endogenous Metabolite
	Vasopressin (argipressin), a cyclic nine-peptide synthesized by hypothalamic neurons, is one of the hormones involved in peptide prohormone synthesis. Vasopressin is involved in the regulation process of hypothalamic-pit...		Endogenous Metabolite
T75933	D[Cha4]-AVP TFA
	d[Cha4]-AVP TFA is a potent and selective agonist for the vasopressin (AVP) V1b receptor, displaying a high affinity with a K i of 1.2 nM. It exhibits greater selectivity for the V1b receptor over the V1a receptor, V2 re...
T83487	[Pmp1,Tyr(OEt)2] AVP
	[Pmp1,Tyr(OEt)2] AVP, a linear analog of the cyclic arginine vasopressin (AVP) antagonist, retains the antagonistic properties of its parent compound while featuring modified phenylalanine (Pmp) and diethyltyrosine (Tyr(...
T7434	Argipressin	Arg8-vasopressin,Vasopressin,AVP	Vasopressin Receptor
	Argipressin (Vasopressin) is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values of 1.31 and 1.44 nM in A7r5 rat aortic smooth ...		Vasopressin Receptor
T80137	(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin	d(CH2)5[Tyr(Me)2, Dab5]AVP	Vasopressin Receptor
	(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].		Vasopressin Receptor
T6288	Mozavaptan	OPC31260l,OPC-31260	Vasopressin Receptor
	Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.		Vasopressin Receptor
T4355	Fuscoside	OPC 21268	Vasopressin Receptor
	Fuscoside (OPC 21268) is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.		Vasopressin Receptor
T28257	OPC-51803	SOU-003,SOU 003,SOU003,OPC51803,OPC 51803	Vasopressin Receptor
	OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.		Vasopressin Receptor
T5444	CLP290	CLP-290	Potassium Channel
	CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatric indications.		Potassium Channel
T40884	SKF 100398	d(CH2)5Tyr(Et)VAVP
	SKF 100398, also known as d(CH2)5Tyr(Et)VAVP, is a particular analog of arginine vasopressin (AVP). It acts as a specific antagonist, specifically targeting the antidiuretic effect caused by both exogenous and endogenous...
T16553	Pneumadin, rat	PNM	Others
	Pneumadin, rat (PNM) exerts a marked antidiuretic effect in animals has a functional AVP system. Pneumadin, rat (PNM) is a decapeptide, which possesses a potent stimulating effect on arginine-vasopressin (AVP) release.		Others
T83501	[Deamino-Pen1,Val4,D-Arg8]-vasopressin		Vasopressin Receptor
	[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP). It effectively reduces plasma aldosterone concentration in rats and is utilized in studying the growth and steroidogenic capa...		Vasopressin Receptor
T29178	YM 471	YM-471,YM471
	YM 471 is a non-peptide arginine vasopressin (AVP) V1A and V2 receptor antagonist with oral activity.
T80133	Pro8-Oxytocin		Oxytocin Receptor
	Pro8-Oxytocin, a modified oxytocin (OXT) ligand, elicits more potent and efficacious responses at primate OXTR and induces stronger behavioral effects compared to the standard mammalian OXT ligand (Leu8-Oxytocin). It dem...		Oxytocin Receptor
T76509	Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
	Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent agonist at the pituitary corticotrope receptor [1].
T80134	Pro8-Oxytocin TFA		Oxytocin Receptor
	Pro8-Oxytocin TFA, a modified oxytocin (OXT) ligand, exhibits greater potency and efficacy than the standard mammalian OXT ligand, Leu8-Oxytocin, at primate OXTR and elicits more pronounced behavioral effects. Compared t...		Oxytocin Receptor
T75708	Argipressin diacetate
	Argipressin (diacetate) (AVP (diacetate), also known as antidiuretic hormone (ADH)), is a nine-amino acid neuropeptide produced by the posterior pituitary gland. It plays a crucial role in maintaining fluid balance, osmo...