Home Tools
Log in
Products Inhibitors Libraries Kits Services Contact Us
Cart
Peptides Monoclonal Antibodies Dye Reagents PROTAC Virtual Screening Targetmol Kits Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails Natural Products Phenols Alkaloids Flavonoids
Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling
MAPK Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library

Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat. No. Product name CAS No. Purity Chemical Structure
TP1452L1 HAEGTFTSD acetate(926018-45-3 free base) TP1452L1 98%
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
T14130 Adomeglivant 1488363-78-5 98%
Adomeglivant is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
T11408 GLP-1 receptor agonist 1 2212020-52-3 98%
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
T35337 Teduglutide 197922-42-2 98%
T7364 NNC-0640 307986-98-7 98%
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
T12878 Semaglutide TFA (910463-68-2 free base) T12878 98%
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T11845 LGD-6972 1207989-09-0 98%
LGD-6972 is an antagonist of glucagon receptor.
TP1039 Secretin (33-59), rat 121028-49-7 98%
Secretin (33-59), rat is a 27-aa peptide, acts on secretin receptor, enhances the secretion of bicarbonate, enzymes, and K+ from the pancreas.
T36579 GLP-1R Agonist DMB 281209-71-0 98%
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
T9579L GLP-1 receptor agonist 9 citrate T9579L 98%
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
TP2071L Bay 55-9837 acetate 98%
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
T35337L Teduglutide acetate 98%
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
T37890L GLP-1(28-36)amide acetate T37890L 98%
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
TP1863L Glucagon (19-29), human acetate TP1863L 98%
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
TP1419L HAEGTFT acetate(926018-95-3 free base) TP1419L 100%
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
TP1796 Albiglutide TFA (782500-75-8 free base) TP1796 100%
Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
T22893 L-168049 191034-25-0 100%
L-168049 is a selective and non-competitive antagonist of human glucagon receptor with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine, respectiv...
TP1111L Tirzepatide Acetate(2023788-19-2 free base) TP1111L 97.3%
Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
TP1382L HAEGTFTSDVS acetate TP1382L 97.47%
HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.
TQ0124 BETP 1371569-69-5 97.92%
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
HAEGTFTSD acetate(926018-45-3 free base)
TP1452L1
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
Adomeglivant
T14130
Adomeglivant is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.
GLP-1 receptor agonist 1
T11408
GLP-1 receptor agonist 1 is a GLP-1 receptor agonist .
Teduglutide
T35337
NNC-0640
T7364
NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.
Semaglutide TFA (910463-68-2 free base)
T12878
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
LGD-6972
T11845
LGD-6972 is an antagonist of glucagon receptor.
Secretin (33-59), rat
TP1039
Secretin (33-59), rat is a 27-aa peptide, acts on secretin receptor, enhances the secretion of bicarbonate, enzymes, and K+ from the pancreas.
GLP-1R Agonist DMB
T36579
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
GLP-1 receptor agonist 9 citrate
T9579L
GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.
Bay 55-9837 acetate
TP2071L
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.
Teduglutide acetate
T35337L
Teduglutide acetate, a GLP-2 analogue, maximizes small intestinal mucosal hypertrophy. Teduglutide acetate partially restores small intestinal epithelial functio...
GLP-1(28-36)amide acetate
T37890L
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.
Glucagon (19-29), human acetate
TP1863L
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.
HAEGTFT acetate(926018-95-3 free base)
TP1419L
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.
Albiglutide TFA (782500-75-8 free base)
TP1796
Albiglutide TFA is a long acting GLP-1 receptor agonist for the treatment of type 2 diabetes mellitus (T2DM).
L-168049
T22893
L-168049 is a selective and non-competitive antagonist of human glucagon receptor with IC50s of 3.7 nM, 63 nM, and 60 nM for human, murine, and canine, respectiv...
Tirzepatide Acetate(2023788-19-2 free base)
TP1111L
Tirzepatide acetate is a dual GIP / GLP-1 receptor agonist.
HAEGTFTSDVS acetate
TP1382L
HAEGTFTSDVS acetate is the first N-terminal 1-11 residues of GLP-1 which stimulates insulin secretion from pancreatic β-cells.
BETP
TQ0124
BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
1 2 3
CORPORATE
About Us Privacy Notice Events & News Terms & Conditions
SUPPORT
Contact Us Worldwide Distributors Quality Control Technical Support
RESOURCE
Product Catalog Product Citations Signaling Pathways Solution Calculators
FOLLOW OUR
Social Network
Newsletter Subscription
Subscribe to receive our lastest product updates and special offers!
Corporate
Support
Resource
Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
Copyright © 2015-2022 TargetMol Chemicals Inc. All rights reserved.