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Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
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Glucagon Receptor

The glucagon receptor is a 62 kDa protein that is activated by glucagon and is a member of the class B G-protein coupled family of receptors, coupled to G alpha i, Gs and to a lesser extent G alpha q. Stimulation of the receptor results in activation of adenylate cyclase and increased levels of intracellular cAMP. In humans, the glucagon receptor is encoded by the GCGR gene.
Cat. No. Product name CAS No. Purity Chemical Structure
T63166 LSN3318839 2764704-18-7 98%
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be...
T60047 V-0219 878453-71-5 98%
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
TP2252 GLP-1 (9-36) amide 161748-29-4 98%
antagonist at the human GLP-1 receptor
TP1976L Oxyntomodulin acetate 98%
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
TP1148L Glucagon-like peptide 1 (1-37), human acetate 98%
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
TP1452L1 HAEGTFTSD acetate(926018-45-3 free base) TP1452L1 98%
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
T12878 Semaglutide TFA (910463-68-2 free base) T12878 98%
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
T35337 Teduglutide 197922-42-2 98%
T9226 CCG-143140 891016-02-7 98%
CCG-143140 is a GLP-1 receptor inverse agonists.
TP1469 Lixisenatide acetate (320367-13-3 free base) 1997361-87-1 98%
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
T3984 GLP-1(7-36), amide 107444-51-9 98%
GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
T3967 Exendin-4 141758-74-9 98%
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...
T63166L (S, R)-LSN 3318839 2765539-92-0 98%
(S, R)-LSN 3318839 is an allosteric modulator of the glucagon-like peptide-3318839 receptor (GLP-1R) that has demonstrated powerful hypoglycemic effects in anima...
T19850 Semaglutide 910463-68-2 98%
Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
T36579 GLP-1R Agonist DMB 281209-71-0 98%
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
T8876 PF-06882961 Tris 2230198-03-3 98%
PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
T8355 Exenatide acetate 141732-76-5 98%
Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
T3896 Shanzhiside methyl ester 64421-28-9 98%
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 ...
TQ0239 PF-06291874 1393124-08-7 98%
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
T12431 PF-06882961 2230198-02-2 98%
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
LSN3318839
T63166
LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can be...
V-0219
T60047
V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.
GLP-1 (9-36) amide
TP2252
antagonist at the human GLP-1 receptor
Oxyntomodulin acetate
TP1976L
Oxyntomodulin acetate, a 37-amino acid peptide hormone, is a glucagon-like peptide 1 (GLP-1) receptor agonist[1].
Glucagon-like peptide 1 (1-37), human acetate
TP1148L
Glucagon-like peptide 1 (1-37), human acetate is a highly potent the GLP-1 receptor agonist.
HAEGTFTSD acetate(926018-45-3 free base)
TP1452L1
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted from in...
Semaglutide TFA (910463-68-2 free base)
T12878
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 diabetes treatment.
Teduglutide
T35337
CCG-143140
T9226
CCG-143140 is a GLP-1 receptor inverse agonists.
Lixisenatide acetate (320367-13-3 free base)
TP1469
Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).
GLP-1(7-36), amide
T3984
GLP-1 (7-36) amide is a peptide hormone released from intestinal L-cells upon nutrient consumption. It binds the GLP-1 receptor in the pancreas and displays vari...
Exendin-4
T3967
Exendin-4 is a glucagon-like peptide-1 receptor (GLP-1) agonist (IC50: 3.22 nM). Exenatide is a 39 amino acid peptide. Compared to GLP-1, exenatide has a longer ...
(S, R)-LSN 3318839
T63166L
(S, R)-LSN 3318839 is an allosteric modulator of the glucagon-like peptide-3318839 receptor (GLP-1R) that has demonstrated powerful hypoglycemic effects in anima...
Semaglutide
T19850
Semaglutide is a glucagon-like peptide 1 receptor (GLP-1R) agonist(EC50 of 6.2 pM in a reporter assay using BHK cells expressing the human receptor).
GLP-1R Agonist DMB
T36579
GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).
PF-06882961 Tris
T8876
PF-06882961 Tris is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
Exenatide acetate
T8355
Exendin-4 is a glucagon-like protein-1 (GLP-1) receptor agonist
Shanzhiside methyl ester
T3896
Shanzhiside methylester reduces neuropathic pain by activating spinal GLP-1 receptors and subsequently stimulating microglial β-endorphin expression via the p38 ...
PF-06291874
TQ0239
PF-06291874 (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.
PF-06882961
T12431
PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.
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