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Perfluorinated SAHA is an HDAC inhibitor for use in cancer treatment regimens, with demonstrated greater antiproliferative properties than SAHA . PFSAHA has also been shown to have higher selectivity for PA3774, an HDAC-like enzyme from P. aeruginosa, as well as other HDACs, which may prove beneficial for developing novel chemotherapeutic treatments for cancer.

KSI-3716 is a c-Myc inhibitor used as a bladder chemotherapy agent. It blocks the formation of the c-MYC MAX complex with the target gene promoter and induces cell cycle arrest and apoptosis. It can be used for bladder cancer research.

KSI-6666 is an orally effective competitive antagonist of sphingosine 1-phosphate receptor 1 (S1PR1), with an IC50 value of 6.4 nM. It exhibits anti-inflammatory activity in models of autoimmune encephalomyelitis and T-cell transfer-induced colitis.

3,7-O-Diacetylpinobanksin is a natural product of Pinus, Pinaceae. The catalog number is TN2910 and the CAS number is 103553-98-6. 3,7-O-Diacetylpinobanksin can be used as a reference standard.

Pinobanksin 3-O-propanoate is a natiral product from forest trees.

The compound AVSEHQLLHDKGKSIQDLRRRFFLHHLI-{Aib}-EIHTAYRFGG facilitates bone ossification and has potential applications in the study of conditions associated with osteogenic insufficiency or diminished bone mineral density (BMD), including osteoporosis [1].

PKSI-527 is an inhibitor of plasma kallikrein (Ki = 0.81 μM). It is selective for plasma kallikrein over glandular kallikrein, plasmin, thrombin, urokinase, and Factor Xa (Kis = >500, 390, >500, 200, and >500 μM, respectively). PKSI-527 reduces bradykinin generation induced by kaolin and λ-carrageenan ex vivo in human plasma. It also prolongs partial thromboplastin and euglobulin clot lysis times. In vivo, PKSI-527 (300 mg/kg per day) reduces hyperplasia, pannus formation, and infiltration of inflammatory cells in the tarsal joint of mice with collagen-induced arthritis.

Dihydroperaksine is a natural product of Rauvolfia, Apocynaceae. The catalog number is TN3860 and the CAS number is 16100-84-8. Dihydroperaksine can be used as a reference standard.

Pinobanksin 5-methyl ether can induce detoxification genes.

Peraksine is a natural product of Rauvolfia, Apocynaceae. The catalog number is TN6030 and the CAS number is 15527-80-7. Peraksine can be used as a reference standard.

Pinobanksin is a natural flavonoid that induces apoptosis in B-cell lymphoma cell lines and SH-SY5Y cells. It is a potent antioxidant that inhibits the peroxidation of low-density lipoprotein (LDL) and is able to occupy the catalytic center of xanthine oxidase (XO) and thus inhibit it. Pinobanksin also exhibits antimicrobial, anti-inflammatory, antiparasitic, anti-mutagenic, anti-proliferative, and anti-angiogenic effects.

Pinobanksin 3-(2-methyl)butyrate is a Pinobanksin derivative. pinobanksin is a apoptosis inducer that can induce apoptosis of F6 cells.

Pinobanksin 3-acetate (3-O-Acetylpinobanksin), a flavonoid derivative, is a strong antioxidant found in sunflowers and honey that inhibits LDL peroxidation.

10-Hydroxydihydroperaksine is a natural product of Rauvolfia, Apocynaceae. The catalog number is TN2568 and the CAS number is 451478-47-0. 10-Hydroxydihydroperaksine can be used as a reference standard.

KS I is a gonadotropin antagonist and is a cyclolignan isolated from extracts of Lycopus and Lithosperum after oxidation with caffeic acid.