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Results for "Casein Kinase" in TargetMol Product Catalog
  • Inhibitor Products
    74
    TargetMol | Activity
  • Recombinant Protein
    19
    TargetMol | inventory
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    4
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TBCA
T21915934358-00-6In house
TBCA (Casein Kinase II Inhibitor III, TBCA) is a highly selective CK2 (casein kinase II) inhibitor, IC50 = 110 nM, Ki = 77 nM. TBCA shows selectivity for CK2 over CK1, DYRK1A and a panel of 27 other kinases.
  • $45
In Stock
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Casein Kinase II Inhibitor IV
T10687863598-09-8In house
Casein Kinase II Inhibitor IV is an inducer of epidermal keratinocyte differentiation.
  • $79
In Stock
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TBB
T269517374-26-4
TBB (NSC-231634)(NSC-231634) is a highly selective, ATP/GTP-competitive inhibitor of casein kinase-2 (CK2).
  • $38
In Stock
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TargetMol | Citations Cited
Casein kinase 1δ-IN-9
T64376854355-54-7
Casein kinase 1δ-IN-9 is a Quinone reductase 2 inhibitor with IC50 of 0.6μM.
  • $147
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Casein Kinase 2 Substrate Peptide
T76411132176-35-3
Casein Kinase 2 Substrate Peptide, a widely recognized CK2 substrate, is synthesized with its C-terminus conjugated to 5-[(2-aminoethyl)amino]naphthalene-1-sulfonic acid (EDANS). This peptide serves as a tool for determining protein kinase CK2 activity [1].
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Casein kinase 1δ-IN-14
T77648793722-88-0
Casein kinase 1δ-IN-14 (WAY-637081) can be used to study atherosclerosis-related cardiovascular disease.
  • $39
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Casein kinase 1δ-IN-7
T77708764694-25-9
Casein kinase 1δ-IN-7 is a Casein kinase 1δ inhibitor for neurodegenerative diseases such as Alzheimer's disease.
  • $39
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Casein kinase 1δ-IN-8
T77709851396-73-1
Casein kinase 1δ-IN-8 is an inhibitor of casein kinase 1δ and is used to treat neurodegenerative diseases such as Alzheimer's disease type.
  • $64
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Casein kinase 1δ-IN-3
T64350349438-77-3
Casein kinase 1δ-IN-3 (Casein kinase 1δ-IN-3) (Compound 23a) is a casein kinase 1 delta (CK1d) inhibitor with a pIC50 of 6.5376 M.
  • $67
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Casein kinase 1δ-IN-6
T775001579991-01-7
Casein kinase 1δ-IN-6 is a potent and selective inhibitor of the protein kinase CK-1δ with an IC50 of 23 nM.Casein kinase 1δ-IN-6 shows neuroprotective and anti-inflammatory activity in both in vitro and in vivo assays.Casein kinase 1δ-IN-6 can be used to study neurodegenerative diseases.
  • $129
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Casein Kinase inhibitor A86
T394822079069-01-3
Casein Kinase inhibitor A86 is a highly effective and orally bioavailable inhibitor of casein kinase 1α (CK1α). Additionally, it displays inhibitory actions towards CDK7 (TFIIH) and CDK9 (P-TEFb). Furthermore, Casein Kinase inhibitor A86 demonstrates the ability to induce apoptosis in leukemia cells, portraying substantial anti-leukemic effects.
    5 days
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    Casein kinase 1δ-IN-4
    T79127851168-98-4
    Casein kinase 1δ-IN-4 (compound 567) is a potent inhibitor of casein kinase 1δ with potential application in Alzheimer's disease research [1].
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    Casein Kinase II Substrate
    T7647595651-74-4
    Casein Kinase II Substrate, a peptide substrate, is selectively phosphorylated by casein kinase II (CK2) [1].
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    Casein kinase 1δ-IN-1
    T60295851871-94-8
    Casein kinase 1δ-IN-1 (WAY-643895) is an inhibitor of casein kinase 1δ (CK1δ), which inhibits CK1δ. Casein kinase 1δ-IN-1 can be used in the study of neurodegenerative diseases such as Alzheimer's disease.
    • $47
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    Casein kinase 1δ-IN-5
    T791541579991-10-8
    Casein kinase 1δ-IN-5 is a potent and selective CK-1δ inhibitor, exhibiting an IC50 of 47 nM, and demonstrates neuroprotective and anti-inflammatory effects in vitro, with potential applications in neurodegenerative disease research.
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    DMAT
    T7390749234-11-5
    DMAT (Casein kinase II Inhibitor) is a potent and specific inhibitor of CK2(IC50 value of 130 nM).
    • $56
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    D4476
    T2449301836-43-1
    D4476 (Casein Kinase I Inhibitor) is an effective, selective, and cell-permeant CK1 (casein kinase 1) inhibitor( IC50=300 nM in a cell-free assay).
    • $36
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    Casein Kinase inhibitor A51
    T91752079068-74-7
    Casein Kinase inhibitor A51 is an orally active casein kinase 1α (CK1α) inhibitor with anticancer activity that induces apoptosis in leukemia cells, and may be used in the study of neck cancers, acute myeloid leukemia, breast and prostate cancers.
    • $399
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    Casein kinase 1δ-IN-10
    T79697332074-85-8
    Casein kinase 1δ-IN-10 is an inhibitor of casein kinase 1δ (CK1δ).
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    Casein Kinase II Receptor Peptide
    T76383198481-81-1
    Casein Kinase II Receptor Peptide, a substrate for casein kinase II, exhibits a Km value of 500 µM. It is utilized to measure the activity of casein kinase II in crude enzyme preparations [1].
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    Casein Kinase II Inhibitor IV Hydrochloride
    T10687L2320347-54-2
    Casein Kinase II Inhibitor IV Hydrochloride is a small-molecule inducer of epidermal keratinocyte differentiation that lead to novel therapeutic approaches for the treatment of skin hyperproliferative disorders.
    • $1,520
    10-14 weeks
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    Casein Kinase Substrates 3
    TP1509154444-97-0
    Casein Kinase Substrates 3 is a substrate of casein kinase.
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    LY294002
    T2008154447-36-6
    LY294002 (SF 1101) is a broad-spectrum inhibitor of PI3K, inhibiting PI3Kα, PI3Kδ, and PI3Kβ (IC50=0.5/0.57/0.97 μM). LY294002 is also an inhibitor of DNA-PK (IC50=1.4 μM) and an inhibitor of CK2 (IC50=98 nM). LY294002 activates apoptosis and autophagy.
    • $34
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    TargetMol | Inhibitor Hot
    TargetMol | Citations Cited
    CK2/ERK8-IN-1
    T108271085822-09-8In house
    CK2/ERK8-IN-1 (TMCB) is a dual inhibitor of casein kinase 2 (CK2) (Ki: 0.25 µM) and ERK8 (IC50s: 0.50 μM) with pro-apoptotic efficacy. CK2/ERK8-IN-1 also binds to PIM1, DYRK1A, and HIPK2 (Kis: 8.65 µM, 11.9 µM, and 15.25 µM).
    • $30
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    LY-294002 hydrochloride
    T4079934389-88-5
    LY-294002 hydrochloride (NSC 697286) is a synthetic molecule inhibitor of PI3Kα/δ/β (IC50: 0.5/0.57/0.97 μM, in cell-free assays); more stable than Wortmannin in solution, and also is a blocker of autophagosome formation.
    • $37
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    Silmitasertib
    T22591009820-21-6
    Silmitasertib (CX-4945) is a potent, orally bioavailable inhibitor of casein kinase 2 (CK2; Ki: 0.38 nM).
    • $34
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    TargetMol | Citations Cited
    CK1-IN-3
    T60005349438-74-0
    CK1-IN-3 is casein kinase 1 (CK1) inhibitor and can be used for research on the treatment or prevention of diseases associated with circadiantiazol rhythm, inflammation diseases.
    • $68
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    Ellagic acid (hydrate)
    T8305314041-08-2
    Ellagic acid (hydrate) is a natural antioxidant and acts as a potent and ATP-competitive CK2 inhibitor (IC50:40 nM, Ki: 20 nM).
    • $76
    Backorder
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    H-89
    T11524127243-85-0
    H-89 is a selective inhibitor of cyclic AMP-dependent protein kinase (protein kinase A; IC50: 48 nM). H-89 has weak inhibition on PKG, Casein Kinase, PKC, and other kinases.
      5 days
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      TargetMol | Citations Cited
      TAK-715
      T6150303162-79-0
      TAK-715 is a p38 MAPK inhibitor for p38α.
      • $34
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      BRD4/CK2-IN-1
      T63991
      BRD4/CK2-IN-1 is the first potent, orally active dual-target inhibitor of BRD4/CK2 (bromodomain-containing protein 4/casein kinase 2), acting on both BRD4 (IC50: 180 nM) and CK2 (IC50: 230 nM). In triple-negative breast cancer (TNBC), BRD4/CK2-IN-1 induces apoptosis and autophagy-related cell death.
      • $1,490
      10-14 weeks
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      CK1-IN-1
      T53931784751-20-7
      CK1-IN-1 (PUN51207) is a casein kinase 1 (CK1) inhibitor. CK1-IN-1 has IC50s of 15 nM, 16 nM, 73 nM for CK1δ, and CK1ε, p38σ MAPK, respectively.
      • $42
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      PF-05236216 hydrochloride
      T708121383376-93-9
      PF-05236216 hydrochloride is a brain penetrant, potent and selective inhibitor of casein kinase 1 delta/epsilon (CK1δ/ε) that modulates circadian rhythms in mice.
      • $1,970
      8-10 weeks
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      TDZD-8
      T6187327036-89-5
      TDZD-8 (NP 01139) is an inhibitor of GSK-3β, with an IC50 of 2 μM; minimal inhibitory effect observed on CDK1, casein kinase II, PKA and PKC.
      • $42
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      SR-3029
      T39721454585-06-8
      SR-3029 is a potent and highly specific CK1δ/CK1ε inhibitor.
      • $39
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      Pyrvinium Iodide
      T6937335648-29-4
      Pyrvinium Iodide is a casein kinase 1α-dependent inhibitor of Wnt/β-Catenin.
      • $1,520
      6-8 weeks
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      QLT0267
      T84998866409-68-9
      QLT0267 is an inhibitor targeting integrin-linked kinase (ILK; IC50= 26 nM), showing over 10-fold selectivity against cyclin-dependent kinases 1, 2, and 5 (Cdk1, Cdk2, and Cdk5), and over 1,000-fold selectivity against C-terminal Src kinase (CSK), DNA-PK, Pim-1, Akt, PKC, and casein kinase 2 (CK2) at a concentration of 10 mg/ml. This compound effectively inhibits the proliferation of NPA187 papillary thyroid cancer cells with an IC50 of approximately 3 µM and induces apoptosis in NPA187, DRO, and K4 cancer cell lines. In vivo studies reveal that QLT0267, administered at 100 mg/kg, significantly reduces tumor growth in a DRO mouse xenograft model and diminishes both tumor volume and intratumoral vascularization in a U87MG glioblastoma mouse xenograft model, showcasing its potential for therapeutic applications in cancer treatment.
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      TMX-4113
      T60740
      TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].
      • $1,400
      10-14 weeks
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      PF 4800567 hydrochloride
      T231381391052-28-0
      casein kinase 1ε inhibitor
      • $690
      35 days
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      Epiblastin A
      T898716470-02-3
      Epiblastin A is an inhibitor of Casein Kinase 1 (CK1). Epiblastin A engages CK1 isoenzymes in cell lysate and induces efficient conversion of epiblast stem cells (EpiSCs) into embryonic stem cells (cESCs).
      • $48
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      Umbralisib
      T49761532533-67-7
      Umbralisib (TGR 1202) is a PI3Kδ inhibitor.
      • $41
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      TTP 22
      T1828329907-28-0
      TTP 22 is a high affinity, ATP-competitive casein kinase 2 (CK2) inhibitor with IC50/Ki of 0.1 uM/40 nM, and shows selectivity >250-fold for CK2 over JNK3, ROCK1, and MET(IC50> 10 uM).
      • $32
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      IWP-2
      T2702686770-61-6
      IWP-2, an inhibitor of Wnt processing and secretion (IC50=27 nM) in a cell-free assay, selectively blocks Porcn-mediated Wnt palmitoylation.
      • $43
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      LH846
      T1877639052-78-1
      LH846 is a selective inhibitor of CK1δ (IC50 values are 290 nM, 1.3 uM and 2.5 uM for CK1δ, ε and α); exhibits no inhibitory activity at CK2.
      • $58
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      TMX-4116
      T617542766385-56-0
      TMX-4116, a casein kinase 1α (CK1α) degrader, preferentially degrades CK1α in MOLT4, Jurkat, and MM.1S cells, exhibiting degradation concentration 50s (DC50s) below 200 nM. TMX-4116 is utilized in the research of multiple myeloma [1].
      • $1,650
      10-14 weeks
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      Benazoline oxalate salt
      T716001021868-82-5
      Benazoline oxalate salt is a pharmacological active compound that inhibits casein kinase Iε (CKIε) or CKIδ phosphorylation of the PER2 protein.
      • $1,520
      6-8 weeks
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      TA-01
      T46451784751-18-3
      TA-01 is a potent CK1 and p38 MAPK inhibitor, with IC50s of 6.4 nM, 6.8 nM, 6.7 nM for CK1ε, CK1δ and p38 MAPK, respectively.
      • $45
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      IN-1130
      T15572868612-83-3
      IN-1130 is a selective inhibitor of ALK5 with IC50 values of 5.3 nM, 36 nM, and 4.3 μM for phosphorylation of ALK5-mediated Smad3, ALK5 phosphorylation of casein and p38α mitogen-activated protein kinase.
      • $48
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      A-3 hydrochloride
      T1406978957-85-4
      A-3 hydrochloride is a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases. A-3 hydrochloride also inhibits PKC and casein kinase I with Ki values of 47 µM and 80 µM, respectively[1]. A-3 hydrochloride against P
      • $30
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      CKI-7 free base
      T10829120615-25-0
      CKI-7 free base is a potent and ATP-competitive inhibitor of casein kinase 1 (CK1; IC50: 6 μM; Ki: 8.5 μM) and a selective Cdc7 kinase inhibitor. CKI-7 free base also inhibits SGK, ribosomal S6 kinase-1 (S6K1), and MSK1.
      • $88
      5 days
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