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Drug Repurposing Compound Library

Catalog No. L9200
  Library Compound List   Excel SDF

Traditional de novo drug discovery and development involves an HTS campaign for de novo candidate hits and requires highly specialized screening facilities and compound libraries containing several million compounds. It is a time consuming and expensive process. As the regulation for drug safety and efficacy is increasingly getting complex, the cost of developing new drugs is keeping skyrocket. Drug repositioning, also known as old drugs for new uses, is an effective strategy to find new indications for existing drugs and has recently drawn attention and has led to several blockbuster drugs because of its high efficiency and low-cost. High-content screens, new biomarkers, noninvasive imaging techniques, and advanced in bioinformatics have created new opportunities for pursuing novel indications for approved compounds.

The Drug Repurposing Compound Library by TargetMol, containing 4630 approved and clinical drugs, which have undergone extensive preclinical studies and have well-characterized bioactivities, safety and bioavailability – properties which could dramatically accelerate drug development and optimization, is a good tool for drug repurposing and cell induction.

All products from TargetMol are for Research Use Only. Not for Human or Veterinary or Therapeutic Use.
Compound Libraries | TargetMol
Pack Size
1 mg
30 μL * 10 mM (in DMSO)
50 μL * 10 mM (in DMSO)
100 μL * 10 mM (in DMSO)
250 μL * 10 mM (in DMSO)
If the above compound libraries do not match your needs,
please contact our compound library specialist for a customized compound library at inquiry@targetmol.com
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Product Description

  • A unique collection of 4630 approved and clinical drugs for high throughput screening (HTS) and high content screening (HCS);
  • An effective tool for discovering new with old drugs, cell induction, and new drug target screening;
  • All approved drugs collected in this library are approved by Food and Drug Administration (FDA), the European Medicine Agency (EMA), or National Medical Products Administration (NMPA), or included in the US Pharmacopeia (USP) Dictionary, the British Pharmacopoeia (BP), the European Pharmacopoeia (EP), the Japanese Pharmacopoeia (JP), or Chinese Pharmacopoeia (CP) Dictionary;
  • Covers various research areas, such as cancer, cardiovascular disease, immunology, respiratory system, etc.
  • Covers various targets, such as 5-HT Receptor, Sodium Channel, p38 MAPK, PI3K, MEK, etc.
  • Detailed compound information with structure, target, activity, and brief introduction;
  • Structurally diverse, medicinally active, and cell permeable;
  • NMR and HPLC validated to ensure high purity and quality.

Library Customization

Targetmol Compound Libraries can be highly customized! Learn More

Packaging And Storage

  • Powder or pre-dissolved DMSO solutions in 96/384 well plate with optional 2D barcode
  • Shipped with blue ice
Request Library Compound List (L9200)

Publications Cited TargetMol Libraries

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Library Composition

Autophagy (458)
Antibacterial (435)
Apoptosis (433)
Antibiotic (389)
Endogenous Metabolite (323)
5-HT Receptor (206)
Adrenergic Receptor (175)
AChR (160)
COX (135)
Dopamine Receptor (128)
Histamine Receptor (127)
DNA/RNA Synthesis (118)
HIV Protease (117)
Parasite (117)
Antifungal (104)
Sodium Channel (100)
Calcium Channel (91)
Potassium Channel (90)
VEGFR (83)
EGFR (79)
Topoisomerase (77)
PDE (76)
PI3K (66)
Reactive Oxygen Species (63)
Glucocorticoid Receptor (60)
P450 (58)
Influenza Virus (57)
CDK (57)
FLT (57)
HCV Protease (55)
PPAR (55)
Estrogen/progestogen Receptor (55)
Dehydrogenase (54)
Ferroptosis (53)
NF-κB (53)
PDGFR (52)
SARS-CoV (52)
Microtubule Associated (50)
GABA Receptor (49)
c-Kit (49)
JAK (48)
FGFR (48)
HDAC (45)
RAAS (43)
Prostaglandin Receptor (42)
mTOR (41)
c-Met/HGFR (39)
Mitophagy (39)
Estrogen Receptor/ERR (38)
HBV (37)
Nucleoside Antimetabolite/Analog (35)
Src (35)
Reverse Transcriptase (34)
Tyrosine Kinases (33)
Serotonin Transporter (32)
iGluR (32)
Androgen Receptor (32)
Adenosine Receptor (32)
GPR (31)
HSV (31)
ribosome (30)
Virus Protease (30)
Proteasome (30)
Bcr-Abl (30)
BTK (29)
Raf (29)
Norepinephrine (28)
TNF (27)
MAO (27)
AChE (27)
NMDAR (27)
ATPase (26)
GluR (26)
Progesterone Receptor (26)
Opioid Receptor (25)
TRP/TRPV Channel (25)
PARP (25)
HER (25)
Phosphatase (25)
Akt (24)
Epigenetic Reader Domain (24)
Transferase (23)
HSP (23)
Antioxidant (23)
Carbonic Anhydrase (23)
Aurora Kinase (23)
Beta Amyloid (22)
p38 MAPK (22)
ROS (22)
Antifection (22)
MEK (21)
Proton pump (21)
HIF/HIF Prolyl-Hydroxylase (21)
PKC (21)
P-gp (21)
IL Receptor (20)
Antiviral (20)
Monoamine Oxidase (20)
DPP-4 (19)
ALK (19)
Thrombin (19)
Phospholipase (18)
MMP (18)
c-RET (18)
DNA Alkylator/Crosslinker (18)
Drug Metabolite (18)
ERK (18)
Interleukin (17)
Trk receptor (17)
AMPK (17)
Mitochondrial Metabolism (17)
Thyroid hormone receptor(THR) (17)
Histone Methyltransferase (16)
GSK-3 (16)
CXCR (16)
Endothelin Receptor (16)
Retinoid Receptor (16)
c-Fms (16)
BCL (16)
Caspase (15)
SGLT (15)
TAM Receptor (15)
TLR (15)
NO Synthase (14)
MRP (14)
CCR (14)
P2X Receptor (14)
Gamma-secretase (14)
PKA (14)
STAT (13)
Lipoxygenase (13)
CFTR (13)
DNA-PK (13)
E1/E2/E3 Enzyme (13)
S1P Receptor (13)
Syk (13)
ROCK (13)
Chk (13)
Integrin (12)
Cannabinoid Receptor (12)
p53 (12)
DNA Alkylation (12)
HMG-CoA Reductase (12)
NADPH (12)
LPL Receptor (12)
HIF (12)
GNRH Receptor (11)
Guanylate cyclase (11)
IGF-1R (11)
Antifolate (11)
Hedgehog/Smoothened (11)
DNA gyrase (11)
TGF-beta/Smad (11)
Nrf2 (11)
Wnt/beta-catenin (11)
DHFR (11)
Factor Xa (11)
FAK (11)
Amino Acids and Derivatives (11)
IAP (10)
Reductase (10)
FXR (10)
Serine Protease (10)
Glutathione Peroxidase (10)
P2Y Receptor (10)
Vasopressin Receptor (10)
Neurokinin receptor (10)
CSF-1R (10)
Kinesin (9)
CETP (9)
ABC (9)
ATM/ATR (9)
NOS (9)
Ras (9)
Histone Demethylase (9)
Hydroxylase (9)
DNA Methyltransferase (9)
Chloride channel (9)
PLK (9)
Glucosidase (9)
Tyrosinase (9)
S6 Kinase (9)
Indoleamine 2,3-Dioxygenase (IDO) (9)
CAT (8)
OX Receptor (8)
CaMK (8)
Casein Kinase (8)
Sirtuin (8)
RSV (8)
Mdm2 (8)
Smo (8)
JNK (8)
Sigma receptor (8)
ROS Kinase (8)
Glucokinase (7)
Xanthine Oxidase (7)
Cysteine Protease (7)
Aminopeptidase (7)
Pim (7)
Monoamine Transporter (7)
Leukotriene Receptor (7)
BACE (7)
Aryl Hydrocarbon Receptor (7)
Glucagon Receptor (7)
Beta-Secretase (7)
IRAK (6)
Ligand for E3 Ligase (6)
DNA (6)
Acyltransferase (6)
Isocitrate Dehydrogenase (IDH) (6)
AhR (6)
ROR (6)
RIP kinase (6)
Fatty Acid Synthase (6)
IκB/IKK (6)
PAK (6)
cholecystokinin (6)
Imidazoline Receptor (5)
GPCR19 (5)
Ephrin Receptor (5)
IDO (5)
CRFR (5)
Aromatase (5)
CaSR (5)
PGE Synthase (5)
Tie-2 (5)
Liver X Receptor (5)
Bradykinin Receptor (5)
GlyT (5)
FAAH (5)
LTR (5)
Gap Junction Protein (5)
Complement System (5)
IFNAR (5)
NADPH-oxidase (5)
Serine/threonin kinase (5)
NOD (5)
Lipid (5)
MT Receptor (5)
GHSR (5)
Melatonin Receptor (4)
LPA Receptor (4)
Wee1 (4)
DprE1 (4)
Neuropeptide Y Receptor (4)
Neprilysin (4)
Decarboxylase (4)
CGRP Receptor (4)
Acetyl-CoA Carboxylase (4)
PD-1/PD-L1 (4)
Anti-infection (4)
Annexin A (4)
KSP (4)
MAPK (4)
Molecular Glues (4)
NOD-like Receptor (NLR) (4)
Oxytocin Receptor (4)
Cell wall (4)
YAP (4)
Melanocortin Receptor (4)
UGT (4)
GST (3)
PDK (3)
Monocarboxylate transporter (3)
Adenosine deaminase (3)
Protease-activated Receptor (3)
Glutaminase (3)
Hexokinase (3)
STING (3)
Somatostatin (3)
Na-K-Cl cotransporter (3)
OAT (3)
Rho (3)
NAMPT (3)
Telomerase (3)
Myosin (3)
CRM1 (3)
Free radical scavengers (3)
LDL (3)
Arginase (3)
Epoxide Hydrolase (3)
DUB (3)
Taste receptor (2)
ATP Citrate Lyase (2)
PYK2 (2)
Stearoyl-CoA Desaturase (SCD) (2)
Aquaporin (2)
Thrombopoietin Receptor (2)
Galectin (2)
Ligands for Target Protein for PROTAC (2)
p97 (2)
GSNOR (2)
BCRP (2)
advanced glycation end products (2)
Phosphorylase (2)
VDA (2)
Glutathione reductase (2)
PKM (2)
PAI-1 (2)
Integrase (2)
GluCls (2)
PERK (2)
transporter (2)
Lipase (2)
CD73 (2)
PROTAC Linker (2)
Porcupine (2)
NEDD8 (2)
IRE1 (2)
MLK (2)
FLAP (2)
Discoidin Domain Receptor (DDR) (2)
TOPK (2)
AAK1 (AP2 associated kinase 1) (1)
Arrestin (1)
MELK (1)
GRK (1)
Na+/Ca2+ Exchanger (1)
DYRK (1)
N-Acetylglucosaminyltransferase (1)
BMI-1 (1)
MTH1 (1)
PAFR (1)
RAR/RXR  (1)
Adiponectin receptor (1)
Motilin Receptor (1)
Immunology/Inflammation related (1)
Stemness kinase (1)
Fas/FasL (1)
PAD (1)
LIM Kinase (1)
CRISPR/Cas9 (1)
Methionine Adenosyltransferase (MAT) (1)
Hippo pathway (1)
ASK (1)
Histone Acetyltransferase (1)
GTPase (1)
VDAC (1)
Dynamin (1)
Survivin (1)
MALT (1)
MNK (1)
PI4K (1)
KLF (1)
Hydrogenase (1)
NPC1L1 (1)
Anion Exchanger (1)
Hck (1)
Kisspeptin (1)
RXFP receptor (1)
cAMP (1)
ACK (1)
SGK (1)
Pyroptosis (1)
PROTACs (1)
Angiotensin-converting Enzyme (ACE) (1)
Platelet aggregation (1)
Adenylyl cyclase (1)
Thioredoxin (1)
HCN Channel (1)
c-Myc (1)

Library Information Sample

Empty 1000025-07-9 1000413-72-8 229005-80-5 1000787-75-6 946387-07-1 1000998-59-3 1175526-27-8 1001288-58-9 1001350-96-4 1001404-83-6 Empty
Vadadustat TAK875 TAK-779 Tegobuvir RN-1734 BMS-687453 AM211 FT011 BMS754807 AAI101
Empty 1001625-82-6 1001645-58-4 1001753-24-7 1001908-89-9 1002304-34-8 1002-84-2 100291-86-9 100299-08-9 10030-52-1 10040-45-6 Empty
RPW-24 SRT1720 hydrochloride INH6 SRT 2183 AMG208 Pentadecanoic acid Apiopaeonoside Pemirolast potassium L-Anserine nitrate salt Sodium Picosulfate
Empty 100427-26-7 1004316-88-4 10045-45-1 100462-37-1 1004990-28-6 100-51-6 1005-24-9 1005264-47-0 1005334-57-5 1005342-46-0 Empty
Lercanidipine Cobicistat 1-Ethyl-2-benzimidazolinone ROSIRIDIN PF-AKT400 Benzyl alcohol 1-Methylnicotinamide chloride MX69 CVT-10216 LCL161
Empty 1005491-05-3 100-55-0 1005504-62-0 1005883-72-6 100643-71-8 1007207-67-1 10075-50-0 1007647-73-5 100784-20-1 10083-24-6 Empty
Tirasemtiv Roniacol Rg3039 Z433927330 Desloratadine CH5132799 5-Bromoindole Smurf1-IN-A01 Halosulfuron-methyl Piceatannol
Empty 100872-83-1 100874-08-6 1009119-64-5 1009119-65-6 100929-71-3 1009298-09-2 1009298-59-2 100929-99-5 1009734-33-1 10097-84-4 Empty
ML346 SB 4 Daclatasvir Daclatasvir dihydrochloride NADPH (tetracyclohexanamine) AZD8055 Vistusertib PAβN dihydrochloride HZ1157 Rotundine
Empty 1009816-48-1 1009817-63-3 1009820-21-6 100986-85-4 101001-34-7 1010411-21-8 1010-60-2 1011244-68-0 1011301-27-1 1011529-10-4 Empty
Thiamet G B-AP15 Silmitasertib Levofloxacin Pamicogrel GSK369796 Dihydrochloride 2-Chloronaphthoquinone TFAP Tenovin3 Azvudine
Empty 101152-94-7 101155-02-6 1011557-82-6 1011-74-1 101-20-2 1012054-59-9 101-21-3 101-26-8 101303-98-4 1013101-36-4 Empty
Milnacipran hydrochloride BW-A78U Tenovin-6 DL-Normetanephrine hydrochloride Triclocarban CUDC101 Chlorpropham Mestinon Zacopride hydrochloride PF04691502
Empty 101-31-5 1013-69-0 1013750-77-0 1013753-99-5 10138-52-0 1013920-15-4 1013937-63-7 1014691-61-2 101477-54-7 101494-95-5 Empty
L-Hyoscyamine Noreugenin ML-030 BC-1382 Gadolinium chloride Vorolanib VTP-27999 TFA GSK0660 Lomerizine hydrochloride 8-CHLOROQUINAZOLIN-4(1H)-ONE
TargetMol