Home Tools
Log in
Cart

Glutaminase

Glutaminase (glutaminase I, L-glutaminase, glutamine aminohydrolase) is an amidohydrolase enzyme that generates glutamate from glutamine. Glutaminase has tissue-specific isoenzymes. Glutaminase has an important role in glial cells.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T78892 Glutaminase C-IN-2 98%
Glutaminase C-IN-2
Glutaminase C-IN-2 (compound 11), an allosteric inhibitor of glutaminase C (GAC), exhibits potent inhibitory activity with an IC50 of 10.64 nM. By disrupting glu...
T79340 GLS1 Inhibitor-7 98%
GLS1 Inhibitor-7
GLS1 Inhibitor-7 (compound 4d) serves as a GLS1 antagonist with an IC50 value of 46.7 μM, demonstrating potential applications in anticancer, antiaging, and anti...
T72679 GLS1 Inhibitor-4 2768599-97-7 98%
GLS1 Inhibitor-4
GLS1 Inhibitor-4 (compound 41e) is a powerful GLS1 inhibitor, demonstrating an IC50 of 11.86 nM. It exhibits antiproliferative effects, substantial metabolic sta...
T6797 Telaglenastat 1439399-58-2 99.89%
Telaglenastat
Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.
T3964 Glutaminase C-IN-1 311795-38-7 99.82%
Glutaminase C-IN-1
Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.
T17289 ZED-1227 1542132-88-6 99.04%
ZED-1227
ZED-1227 (TAK-227) is an orally active, selective and potent transglutaminase 2 (TG2) inhibitor with anticancer activity that blocks inflammation-induced TG2 exp...
T37385 Glutaminase-IN-3 1439399-45-7 98.51%
Glutaminase-IN-3
Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
T67865 BJJF078 2531244-56-9 98.19%
BJJF078
BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 an...
T6791 BPTES 314045-39-1 98.06%
BPTES
BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.
T62560 Sirpiglenastat 2079939-05-0 98.01%
Sirpiglenastat
Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by inhibiting glutamine metabolism and stimulating the in...
T17206 UPGL00004 1890169-95-5 97.44%
UPGL00004
UPGL00004 is a potent glutaminase C (GAC) inhibitor with an IC50 of 29 nM. Kd of UPGL00004 for GAC was 27 nM. UPGL00004 has a strong inhibitory effect on the pro...
T20121 L-Albizziin 1483-07-4 100%
L-Albizziin
L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.
T3968 GK921 1025015-40-0
GK921
GK921 is a transglutaminase 2 (TGase) inhibitor.
T8373 6-Diazo-5-oxo-L-nor-Leucine 157-03-9 98%
6-Diazo-5-oxo-L-nor-Leucine
6-Diazo-5-oxo-L-nor-Leucine (L-6-Diazo-5-oxonorleucine) is an antagonist of glutaminases (Ki : 6 μM). It is an antineoplastic antibiotic produced by an unidentif...
Glutaminase C-IN-2
T78892
Glutaminase C-IN-2 (compound 11), an allosteric inhibitor of glutaminase C (GAC), exhibits potent inhibitory activity with an IC50 of 10.64 nM. By disrupting glu...
GLS1 Inhibitor-7
T79340
GLS1 Inhibitor-7 (compound 4d) serves as a GLS1 antagonist with an IC50 value of 46.7 μM, demonstrating potential applications in anticancer, antiaging, and anti...
GLS1 Inhibitor-4
T72679
GLS1 Inhibitor-4 (compound 41e) is a powerful GLS1 inhibitor, demonstrating an IC50 of 11.86 nM. It exhibits antiproliferative effects, substantial metabolic sta...
Telaglenastat
T6797
Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.
Glutaminase C-IN-1
T3964
Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.
ZED-1227
T17289
ZED-1227 (TAK-227) is an orally active, selective and potent transglutaminase 2 (TG2) inhibitor with anticancer activity that blocks inflammation-induced TG2 exp...
Glutaminase-IN-3
T37385
Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.
BJJF078
T67865
BJJF078, an aminopiperidine derivative, is a potent inhibitor of recombinant human and mouse glutamine aminotransferase (TG2) activity, with IC50 values of 41 an...
BPTES
T6791
BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.
Sirpiglenastat
T62560
Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by inhibiting glutamine metabolism and stimulating the in...
UPGL00004
T17206
UPGL00004 is a potent glutaminase C (GAC) inhibitor with an IC50 of 29 nM. Kd of UPGL00004 for GAC was 27 nM. UPGL00004 has a strong inhibitory effect on the pro...
L-Albizziin
T20121
L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.
GK921
T3968
GK921 is a transglutaminase 2 (TGase) inhibitor.
6-Diazo-5-oxo-L-nor-Leucine
T8373
6-Diazo-5-oxo-L-nor-Leucine (L-6-Diazo-5-oxonorleucine) is an antagonist of glutaminases (Ki : 6 μM). It is an antineoplastic antibiotic produced by an unidentif...
TargetMol