fumarate — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T22746	Tesmilifene fumarate	DPPE fumarate	Histamine Receptor
	Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。		Histamine Receptor
T0147	Clemastine fumarate	HS-592 (fumarate),Meclastine fumarate,Meclastine (fumarate)	Autophagy , Histamine Receptor
	Clemastine fumarate (Meclastine (fumarate)) is a synthetic ethanolamine with anticholinergic, sedative, and histamine H1 antagonistic properties.		Autophagy , Histamine Receptor
T35346	Tiamulin fumarate	Thiamutilin fumarate	Antibacterial
	Tiamulin fumarate （Thiamutilin fumarate） is a semisynthetic diterpenoid antibiotic with antibacterial activity and inhibition of protein synthesis, which can be used to study pneumocystis.		Antibacterial
T0001	Iron(II) fumarate	Ferrous fumarate,Iron Fumarate	Others
	Iron(II) fumarate (Iron Fumarate) is the iron(II) salt of fumaric acid, a reddish-orange powder, applied to supply iron intake.		Others
T13241	UB 165 fumarate	UB-165 fumarate,UB165 fumarate	AChR
	UB 165 fumarate is an agonist of the nAChR, a partial agonist of the α4β2 subtype, and a full agonist of the α3β2 subtype, with a Ki value of 0.27 nM for binding to [3H]-nicotine measured in rat brain.		AChR
T27047	Clovoxamine fumarate	DU23811 fumarate,DU 23811 fumarate,DU-23811 fumarate	5-HT Receptor , Serotonin Transporter , Norepinephrine
	Clovoxamine fumarate (DU 23811 fumarate) is a 5-hydroxytryptamine reuptake, serotonin and norepinephrine inhibitor with antidepressant and anticonvulsant activity.		5-HT Receptor , Serotonin Transporter , Norepinephrine
T39214L	LXE408 fumarate	LXE408 fumarate (1799330-15-6 Free base)	Proteasome
	LXE408 fumarate is an orally active, non-competitive and kinetoplastid-selective proteasome inhibitor. LXE408 fumarate has an IC50 of 0.04 μM for L. donovani proteasome and an EC50 of 0.04 μM for L. donovani. LXE408 fuma...		Proteasome
T6541	Ibutilide Fumarate	Corvert Fumarate,U70226E	Calcium Channel , Sodium Channel
	Ibutilide Fumarate (U70226E) is the fumarate salt form of ibutilide, a class III antiarrhythmic agent. Ibutilide exerts its effect by activating a slow, inward, predominately sodium current rather than by blocking outwar...		Calcium Channel , Sodium Channel
T41249	Tenofovir alafenamide fumarate	GS-7340 fumarate	HIV Protease
	Tenofovir alafenamide fumarate (GS-7340 fumarate) is an orally available Tenofovir precursor compound Tenofovir alafenamide fumarate has anti-HIV activity and can be used to prevent HIV infection.		HIV Protease
T30098	Aplindore Fumarate	Aplindore,DAB-452 Fumarate,DAB-452	Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
	Aplindore Fumarate (DAB-452) is a small molecule dopamine D2 receptor partial agonist.Aplindore Fumarate exhibits high affinity for dopamine D2 and D3 receptors, and low affinity for dopamine D4, 5-hydroxytryptophan (5-H...		Dopamine Receptor , 5-HT Receptor , Adrenergic Receptor
T13385	Zamifenacin fumarate	UK-76654 fumarate	AChR
	Zamifenacin fumarate (UK-76654 fumarate) is a potent and gut-selective antagonist of muscarinic M3 receptor.		AChR
T0994	Ketotifen fumarate	HC 20511 fumarate	PDE , Histamine Receptor
	Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.		PDE , Histamine Receptor
T2769	3-Aminopropionitrile fumarate (2:1)	Di-β-aminopropionitrile fumarate,3-Aminopropionitrile fumarate,β-Aminopropionitrile fumarate,3-Aminopropionitrile fumarate 2:1,Beta-Aminopropionitrile fumarate,β-Ammoniumpropionitrile hemifumarate	Others
	3-Aminopropionitrile fumarate (2:1) (β-Aminopropionitrile fumarate) is an organic compound and antirheumatic agent used in veterinary medicine.		Others
T37807	JTV 519 fumarate
	Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo. Hunt et al (2007) K201 (JTV519) suppresses spontaneous Ca2+ release and [3H]r...
T28453L	Propiram fumarate HCl	Propiram fumarate HCl(15686-91-6 Free base)	Opioid Receptor
	Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.		Opioid Receptor
T2409L	Tenofovir Disoproxil Fumarate	GS-1278 Disoproxil Fumarate,Tenofovir DF	HBV , HIV Protease , Reverse Transcriptase
	Tenofovir Disoproxil Fumarate (GS-1278 Disoproxil Fumarate) is a pro-drug, fumaric acid salt form of tenofovir, a nucleoside reverse transcriptase inhibitor analog of adenosine. Tenofovir disoproxil fumarate is prescribe...		HBV , HIV Protease , Reverse Transcriptase
T13324	VUF11207 fumarate		CXCR , Arrestin
	VUF11207 fumarate is an agonist of CXCR7 and a high-potency ligand of CXCR7 (pKi: 8.1).		CXCR , Arrestin
T17038	Tepilamide fumarate	XP-23829	Others
	Tepilamide fumarate (XP-23829) is an oral fumaric acid ester and is used in the research of moderate to severe chronic plaque psoriasis.		Others
T11071	Dofequidar fumarate	MS-209	P-gp
	Dofequidar fumarate (MS-209)(MS-209 fumarate), a quinoline-based compound administered orally, is known for counteracting multidrug resistance (MDR) through the inhibition of ABCB1/P-glycoprotein (P-gp) and ABCC1/MDR-ass...		P-gp
T22810	GR 89696 fumarate		Opioid Receptor
	GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.		Opioid Receptor