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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T23087 | NPY 5RA972 | Neuropeptide Y Receptor | |
neuropeptide Y Y5 receptor antagonist | |||
TP2194L | Neuropeptide Y (scrambled) Acetate | Pro-Neuropeptide Y (scrambled) Acetate,NPY (scrambled) Acetate | Others |
Neuropeptide Y (scrambled) Acetate (Pro-Neuropeptide Y (scrambled) Acetate) is a scrambled peptide of Neuropeptide Y that has been implicated in Alzheimer's disease (AD) and may have neuroprotective effects. | |||
T83677 | Neuropeptide Y (porcine, bovine) TFA | NPY (porcine, bovine) | |
Neuropeptide Y (NPY), a neuropeptide, plays roles in regulating appetite, vasoconstriction, cardiac contractility, and intestinal secretion, acting as an agonist for NPY receptors Y1, Y2, and Y5. Expressed ubiquitously, ... | |||
T71749 | SF-22 | Neuropeptide Y Receptor | |
SF-22 is a neuropeptide Y receptor (Y2R) antagonist that crosses the blood-brain barrier and has potential anti-inflammatory activity for the study of diseases associated with neurological disorders. | |||
T23094 | NTNCB hydrochloride | Others , Neuropeptide Y Receptor | |
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor. | |||
TQ0286 | MK-0557 | Neuropeptide Y Receptor | |
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM). | |||
TP2206 | [Leu31,Pro34]-Neuropeptide Y (porcine) | Neuropeptide Y Receptor | |
High affinity neuropeptide Y Y1 receptor agonist | |||
T10539 | BIBO3304 TFA | Neuropeptide Y Receptor | |
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 receptor). | |||
T8963 | CYM2503 | Neuropeptide Y Receptor | |
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by ... | |||
T5455 | HT-2157 | SNAP37889,SNAP-37889 | Neuropeptide Y Receptor |
HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target. | |||
T17222 | Velneperit | S2367 | Neuropeptide Y Receptor |
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity. | |||
T5587 | CGP71683 hydrochloride | CGP71683A | Neuropeptide Y Receptor |
CGP71683 hydrochloride (CGP71683A) is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes. | |||
TP1380 | Galanin (1-16), mouse, porcine, rat | Neuropeptide Y Receptor | |
Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons. | |||
T1997 | JNJ-31020028 | JNJ 31020028 | Neuropeptide Y Receptor |
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold selectivity for Y2 versus human Y1/Y4/Y5 receptors. | |||
TP1059 | Peptide YY (PYY) (3-36), human | Peptide YY (3-36) | Neuropeptide Y Receptor |
Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite. | |||
T8456 | GALNON | Neuropeptide Y Receptor | |
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties | |||
T12895 | SHA 68 | Neuropeptide Y Receptor | |
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respectively). | |||
T4445 | Tolfenpyrad | Antibacterial | |
Tolfenpyrad is an effective insecticide[1], used against pests that are resistant to existing insecticides such as organophosphates and carbamates.[2] | |||
T0435 | Sulfinpyrazone | (+/-)-Sulfinpyrazone,G-28315,NSC 75925 | COX |
Sulfinpyrazone (NSC-75925) is a uricosuric drug that is used to reduce the serum urate levels in gout therapy. It lacks anti-inflammatory, analgesic, and diuretic properties. | |||
T4446 | Tebufenpyrad | Pyranica,MK239,Comanche | Mitochondrial Metabolism |
Tebufenpyrad (Comanche) (mitochondrial complex-1 inhibitors) is an agro-chemically important acaricide that functions like the known mitochondrial toxicant rotenone. |