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GPCR/G Protein CaSR

CaSR

The calcium-sensing receptor (CaSR) is a Class C G-protein coupled receptor which senses extracellular levels of calcium ion. It is primarily expressed in the parathyroid gland and the renal tubules of the kidney.
Cat No. product name
T22795 Gadolinium chloride Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
T10666 Calhex 231 hydrochloride Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
T15261 Evocalcet Evocalcet has an activating effect on the calcium-sensing receptor (CaSR).
T8403 Cinacalcet Cinacalcet is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .
TP1236 Etelcalcetide hydrochloride (1262780-97-1 free base) Etelcalcetide hydrochloride is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide hydrochloride is effecti...
T4967 NPS-2143 HCL NPS-2143 is a selective potent calcium ion-sensing receptor antagonist.
T2406 Cinacalcet hydrochloride Cinacalcet hydrochloride is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-sensing receptors to seru...
Gadolinium chloride
T22795CAS 10138-52-0
Gadolinium chloride is a calcium-sensing receptor (CaSR) agonist
Calhex 231 hydrochloride
T10666CAS 2387505-78-2
Calhex 231 hydrochloride is a CaSR inhibitor with the potential for diabetic cardiomyopathy treatment. It blocks Ca2+-induced accumulation of [3H]inositol phosph...
Evocalcet
T15261CAS 870964-67-3
Evocalcet has an activating effect on the calcium-sensing receptor (CaSR).
Cinacalcet
T8403CAS 226256-56-0
Cinacalcet is an orally active, allosteric Ca receptor (CaR) agonist, treatment of cardiovascular disease .
Etelcalcetide hydrochloride (1262780-97-1 free base)
TP1236CAS 1334237-71-6
Etelcalcetide hydrochloride is a synthetic peptide as an allosteric modulator of the calcium (Ca)-sensing receptor (CaSR). Etelcalcetide hydrochloride is effecti...
NPS-2143 HCL
T4967CAS 324523-20-8
NPS-2143 is a selective potent calcium ion-sensing receptor antagonist.
Cinacalcet hydrochloride
T2406CAS 364782-34-3
Cinacalcet hydrochloride is a naphthalene derivative and CALCIMIMETIC AGENT that increases the sensitivity of PARATHYROID GLAND calcium-sensing receptors to seru...