T15702 |
Lactacystin
|
133343-34-7
|
98%
|
|
Lactacystin is an antibiotic Streptomyces spp. the metabolite and is an effective and selective proteasome inhibitor (IC50: 4.8 μM for 20S proteasome). Lactacyst...
|
T16568 |
PR-924
|
1416709-79-9
|
98%
|
|
PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM). PR-924 inhibits growth and triggers apoptosis in multiple...
|
T0242L |
Sitagliptin phosphate monohydrate
|
654671-77-9
|
98%
|
|
Sitagliptin phosphate is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.
|
T12561 |
Proteasome-IN-1
|
374080-21-4
|
98%
|
|
Proteasome-IN-1 is an inhibitor of proteasome.
|
T15678 |
KZR-504
|
1629052-78-3
|
98%
|
|
KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).
|
T11924 |
M3258
|
2285330-15-4
|
98%
|
|
LMP7-IN-1 may used in the research of inflammatory and autoimmune diseases, neurodegenerative diseases, proliferative diseases and cancer, is an inhibitor of imm...
|
T21617 |
MG-115
|
133407-86-0
|
98%
|
|
MG-115 is a potent and reversible proteasome inhibitor, with K i s of 21 nM and 35 nM for 20S and 26S proteasome, respectively. MG-115 specifically inhibit the c...
|
T7369L |
Gemigliptin Tartrate(911637-19-9 free base)
|
1374639-74-3
|
98%
|
|
Gemigliptin tartrate is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4). It has an IC50 of 10.3 nM for human recombina...
|
T10238 |
Aclacinomycin A hydrochloride
|
75443-99-1
|
98%
|
|
Aclacinomycin A (Aclarubicin) hydrochloride is a fluorescent molecule and the first described non-peptidic inhibitor showing discrete specificity for the CTRL (c...
|
T36902 |
RA375
|
|
98%
|
|
RA375 is a inhibitor of RPN13 (26S proteasome regulatory subunit). RA375 activates UPR signaling, ROS production and apoptosis. RA375 exhibits ten-fold greater a...
|
T39214L |
LXE408 fumarate
|
|
98%
|
|
LXE408 fumarate is an orally active, non-competitive and kinetoplastid-selective proteasome inhibitor. LXE408 fumarate has an IC50 of 0.04 μM for L. donovani pro...
|
T16169 |
N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride
|
4272-74-6
|
98%
|
|
N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride is an inhibitor of trypsin-like protease. N-alpha-Tosyl-L-lysine chloromethyl ketone hydrochloride exhib...
|
T1502 |
Vildagliptin
|
274901-16-5
|
|
|
Vildagliptin is a cyanopyrrolidine-based, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4), with hypoglycemic activity. Vildagliptin's cyano moiet...
|
T3359 |
Aprotinin
|
9087-70-1
|
|
|
Aprotinin a broad-spectrum serine protease inhibitor, inhibiting the activity of a number of different esterases and proteases, including trypsin, chymotrypsin, ...
|
T7814 |
Alloxan monohydrate
|
2244-11-3
|
|
|
Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
|
T2470 |
MDL-28170
|
88191-84-8
|
|
|
Calpain Inhibitor III is a Cysteine protease.
|
T7369 |
Gemigliptin
|
911637-19-9
|
|
|
Gemigliptin is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)
|
T8397 |
Ixazomib citrate
|
1239908-20-3
|
100%
|
|
Ixazomib citrate is a prodrug of Ixazomib (MMLN-2238). MLN9708 is an orally bioavailable second generation proteasome inhibitor (IC50 of 3.4 nM ) with potential ...
|
T6999 |
Teneligliptin hydrobromide
|
906093-29-6
|
100%
|
|
Teneligliptin is a novel, potent, and long-lasting dipeptidyl peptidase-4 inhibitor; competitively inhibited human plasma, rat plasma, and human recombinant DPP-...
|
T7133 |
Anagliptin
|
739366-20-2
|
100%
|
|
Anagliptin is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.
|