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Polyinosinic-polycytidylic acid sodium (Poly(I:C) sodium) is a synthetic analog of double-stranded RNA and an agonist of toll-like receptor 3 (TLR3) and retinoic acid inducible gene I (RIG-I)-like receptors (RIG-I and MDA5).

Benproperine phosphate (Pirexyl phosphate) is a cough suppressant.

Thioproperazine (RP 7843) is an orally effective antipsychotic also used as a tranquilizer and antiemetic for the treatment of schizophrenia and the manic phase of bipolar disorder, acting as a histamine and adrenergic receptor blocker.

Clenproperol, a β2-adrenergic agonist, is a chemical compound commonly used in veterinary medicine to treat respiratory diseases in animals.

Benproperine is a bioactive molecule with antineoplastic properties.

Properdistatin, a peptide originating from the thrombospondin 1 (TSP-1) domain of properdin, exhibits angiogenesis inhibition and vascular function enhancement capabilities, showing promise for melanoma research [1].

Clenproperol-d7 is a deuterated compound of Clenproperol.

Clenproperol (Standard) is the standard substance of Clenproperol, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Clenproperol is a β2-adrenergic agonist.

Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.

1-Dodecylimidazole (N-Dodecylimidazole) is a chemical compound that acts as a cytotoxic agent and lysosomotropic detergent, inducing cell death through acid-dependent lysosomal accumulation, disrupting the lysosomal membrane, and releasing cysteine proteases into the cytoplasm. It also exhibits hypocholesterolemic and broad-spectrum antifungal activities.

Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist. Pericyazine is a first-generation antipsychotic drug that is used as an adjunct to the short-term management of severe anxiety states and psychosis.

AAL-993 is a potent VEGFR inhibitor with IC50s of 130 nM, 23 nM and 18 nM for VEGFR1, VEGFR2 and VEGFR3, respectively. AAL993 has a weak inhibitory effect on other tyrosine kinases. AAL993 also shows potent antiangiogenic and antitumor activities.

Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.

Hispidin is a polyphenol originally, including antioxidant, anti-inflammatory, and cytoprotective properties

PF-9601N showed high potency and selectivity as a MAO-BI (monoamine oxidase type B inhibitor) and also demonstrated remarkable neuroprotective properties in several in vivo and cellular models of PD.

Mesdopetam hemitartrate (IRL790 hemitartrate) is an antagonist of dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM for human recombinant D3 receptor). It has psychomotor stabilizing properties.

N-Benzyllinoleamide ((9Z,12Z)-N-Benzyloctadeca-9,12-dienamide) is a natural product isolated from Lepidium meyenii Walp, has pharmaceutical property against exercise-induced fatigue.

L-Proline (proline) is a nonessential amino acid in humans. It is an essential component of collagen and is important for proper functioning of joints and tendons. It also helps maintain and strengthen heart muscles.

1-Methylindazole-3-carboxylic acid is an excellent solvent with a proper boiling point.

7-Keto-27-hydroxycholesterol is a significant bioactive compound known for its ability to activate the smoothened (SMO) protein within the Hedgehog (Hh) signaling pathway, which is crucial for proper cell differentiation in embryonic tissues.

Rhodblock 1a is an inhibitor of the Rho kinase signaling pathway, which disrupts the localization and function of proteins within the Rho pathway. This interference hinders the proper formation of the cleavage furrow during cell division, leading to some cells either failing to form the cleavage furrow or forming a ruptured furrow, resulting in binucleated cells. Rhodblock 1a can be utilized for investigating cell division mechanisms and holds potential for research into cardiovascular diseases and cancer.

DNJ-20 is an α-glucosidase inhibitor with an IC50 of 55.3 μg/mL. It exhibits broad-spectrum activity against SARS-CoV-2. By interfering with the endoplasmic reticulum-associated glycoprotein folding process (ERQC), DNJ-20 hinders the proper processing of viral glycoproteins, thus blocking the formation and infection of viral particles. It is effective against several SARS-CoV-2 variants, as well as HCoV-229E and HCoV-0C43, with IC50 values reaching up to 1.49 μM. DNJ-20 can be utilized for pan-coronavirus research.

Tubulozole is a microtubule inhibitor. It inhibits microtubule dynamics required for proper mitotic function, effectively blocking cell cycle progression and resulting in apoptosis.

BuChE-IN-2 is an excellent inhibitor of butylcholinesterase (BuChE) with IC50 values of 1.28 μM for BuChE and 0.67 μM for NO. It inhibits Aβ aggregation, ROS formation, and Cu2+ chelation, shows proper blood-brain barrier (BBB) penetration, and is suitable for Alzheimer's disease research.