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Compounds

Cat No. Product Name
T13206 Tris(2,4-di-tert-butylphenyl)phosphate Phospholipase
Tris(2,4-di-tert-butylphenyl)phosphate 是一种从 Vitex negundoL 中分离的活性化合物,能够通过分子对接抑制了分泌性磷脂酶 A2(sPLA2),具有抗炎作用。
T2044 Varespladib LY315920,伐瑞拉地,伐瑞拉迪 Phospholipase
Varespladib 是选择性group IIA, secretory phospholipase A2(sPLA2)抑制剂,其IC50=9 nM。它对大鼠,兔,豚鼠和人等各种物种血清的sPLA2活性具有明显的抑制作用,IC50分别为 8...
T6928 Pantoprazole SKF96022,BY1023,泮托拉唑 Autophagy , Proton pump , Apoptosis
Pantoprazole 是一种质子泵抑制剂,用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。
TN1419 Rhamnetin 鼠李素,beta-Rhamnocitrin Phospholipase , Others
Rhamnetin 是一种槲皮素衍生物,在芫荽中被发现,具有抗氧化和抗炎活性。Rhamnetin 可抑制分泌型磷脂酶 A2。
T0161 Pantoprazole Sodium Hydrate SKF96022 sodium hydrate,SKF96022 (sodium hydrate),泮托拉唑钠水合物,BY1023 (sodium hydrate) Apoptosis , Potassium Channel , Proton pump , Autophagy
Pantoprazole Sodium Hydrate 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑,是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。
T16865 SCH28080 ATPase , Proton pump
SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂,具有抗溃疡活性、抗分泌和细胞保护...
T6929 Pantoprazole sodium SKF96022 (sodium),泮托拉唑钠盐,泮托拉唑钠,BY1023 (sodium),SKF96022 sodium,Pantoloc,BY-1023 sodium,Pantecta Others , HIF , Proton pump , Autophagy , Apoptosis
Pantoprazole sodium 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生...
TCS1772 Dehydroabietic acid Dehydroabietate,脱氢枞酸;脱氢松香酸 Antifection
Dehydroabietic acid 是 EBV-EA 活化抑制剂。 它是食物衍生化合物,可通过降低血浆葡萄糖、胰岛素水平、血浆甘油三酯 (TG) 和肝 TG 水平来治疗肥胖相关疾病。它的衍生物在动物模型中表现出抗分泌和抗胃蛋白酶作用。
T27539 Hexocyclium metilsulfate AB-803,Traline,AB 803,AB803
Hexocyclium metilsulfate has anti-gastric secretory effects in humans.
T10008 BTM-1086 Others
BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.
T39465 (Z)-Lafutidine (Z)-Lafutidine,(Z)-FRG-8813
(Z)-Lafutidine ((Z)-FRG-8813) is a powerful histamine H2 receptor antagonist renowned for its anti-secretory and gastrop...
TN4659 Nimbin COX
Nimbin is an anti-pyretic, can be used to treat arthritis, hypoglycaemia, peptic ulcers, anti-secretory activity, and it...
TMPY-04912 PLA2G2A Protein, Mouse, Recombinant (His Tag)
Phospholipase A2, membrane associated, also known as Phosphatidylcholine 2-acylhydrolase 2A, Group IIA phospholipase A2,...
TMPY-01705 PLA2G2A Protein, Human, Recombinant (His Tag)
Phospholipase A2, membrane associated, also known as Phosphatidylcholine 2-acylhydrolase 2A, Group IIA phospholipase A2,...
T76320 FIZZ-1 (32-51) (mouse)
FIZZ-1 (32-51) (mouse) 是一种富含半胱氨酸的分泌蛋白,在过敏性气道炎症中,由巨噬细胞、支气管上皮和 II 型肺泡上皮细胞 (AEC) 高度表达。FIZZ1 (32-51) (mouse) 还对肺成纤维细胞有抗凋亡作用。...
TMPY-03120 Prostaglandin D2 Synthase Protein, Human, Recombinant (His Tag), HPLC-verified
PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s...
TMPY-02597 IL-37 Protein, Human, Recombinant
Interleukin 1 family member 7, or interleukin 37 (IL1F7 / IL37 / IL-1H4) is a secretory protein belonging to the Interle...
TMPY-05069 Prostaglandin D2 Synthase Protein, Rat, Recombinant (His Tag)
PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s...
TMPY-04624 Prostaglandin D2 Synthase Protein, Mouse, Recombinant (His Tag)
PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s...
TN5221 (-)-Variabilin
Variabilin, a novel inhibitor of human platelet aggregation, it is a potent RGD (Arg-Gly-Asp)-containing antagonist of t...
Tris(2,4-di-tert-butylphenyl)phosphate
T13206
synonym:
Target:
Varespladib
T2044
synonym: LY315920,伐瑞拉地,伐瑞拉迪
Target:
Pantoprazole
T6928
synonym: SKF96022,BY1023,泮托拉唑
Target:
Rhamnetin
TN1419
synonym: 鼠李素,beta-Rhamnocitrin
Target:
Pantoprazole Sodium Hydrate
T0161
synonym: SKF96022 sodium hydrate,SKF96022 (sodium hydrate),泮托拉唑钠水合物,BY1023 (sodium hydrate)
Target:
SCH28080
T16865
synonym:
Target:
Pantoprazole sodium
T6929
synonym: SKF96022 (sodium),泮托拉唑钠盐,泮托拉唑钠,BY1023 (sodium),SKF96022 sodium,Pantoloc,BY-1023 sodium,Pantecta
Target:
Dehydroabietic acid
TCS1772
synonym: Dehydroabietate,脱氢枞酸;脱氢松香酸
Target:
Hexocyclium metilsulfate
T27539
synonym: AB-803,Traline,AB 803,AB803
Target:
BTM-1086
T10008
synonym:
Target:
(Z)-Lafutidine
T39465
synonym: (Z)-Lafutidine,(Z)-FRG-8813
Target:
Nimbin
TN4659
synonym:
Target:
PLA2G2A Protein, Mouse, Recombinant (His Tag)
TMPY-04912
synonym:
Target:
PLA2G2A Protein, Human, Recombinant (His Tag)
TMPY-01705
synonym:
Target:
FIZZ-1 (32-51) (mouse)
T76320
synonym:
Target:
Prostaglandin D2 Synthase Protein, Human, Recombinant (His Tag), HPLC-verified
TMPY-03120
synonym:
Target:
IL-37 Protein, Human, Recombinant
TMPY-02597
synonym:
Target:
Prostaglandin D2 Synthase Protein, Rat, Recombinant (His Tag)
TMPY-05069
synonym:
Target:
Prostaglandin D2 Synthase Protein, Mouse, Recombinant (His Tag)
TMPY-04624
synonym:
Target:
(-)-Variabilin
TN5221
synonym:
Target:
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