T13206 |
Tris(2,4-di-tert-butylphenyl)phosphate
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Phospholipase
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Tris(2,4-di-tert-butylphenyl)phosphate 是一种从 Vitex negundoL 中分离的活性化合物,能够通过分子对接抑制了分泌性磷脂酶 A2(sPLA2),具有抗炎作用。 |
T2044 |
Varespladib
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LY315920,伐瑞拉地,伐瑞拉迪 |
Phospholipase
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Varespladib 是选择性group IIA, secretory phospholipase A2(sPLA2)抑制剂,其IC50=9 nM。它对大鼠,兔,豚鼠和人等各种物种血清的sPLA2活性具有明显的抑制作用,IC50分别为 8... |
T6928 |
Pantoprazole
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SKF96022,BY1023,泮托拉唑 |
Autophagy
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Proton pump
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Apoptosis
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Pantoprazole 是一种质子泵抑制剂,用于短期治疗由胃食管反流病引起的食管糜烂和溃疡。它联合阿霉素可显著增加肿瘤生长延迟。它是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。 |
TN1419 |
Rhamnetin
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鼠李素,beta-Rhamnocitrin |
Phospholipase
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Others
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Rhamnetin 是一种槲皮素衍生物,在芫荽中被发现,具有抗氧化和抗炎活性。Rhamnetin 可抑制分泌型磷脂酶 A2。 |
T0161 |
Pantoprazole Sodium Hydrate
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SKF96022 sodium hydrate,SKF96022 (sodium hydrate),泮托拉唑钠水合物,BY1023 (sodium hydrate) |
Apoptosis
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Potassium Channel
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Proton pump
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Autophagy
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Pantoprazole Sodium Hydrate 是一种具有口服活性的质子泵抑制剂。它是取代的苯并咪唑,是H+/K+-ATPase 抑制剂。它可改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生长延迟。 |
T16865 |
SCH28080
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ATPase
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Proton pump
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SCH28080 是一种可逆且具有 K+ 竞争性的胃 H+/K+-ATP 酶 (H+/K+-ATPase) 抑制剂,IC50 值为 20 nM (家兔微粒体膜)。SCH28080 在体内是有效的酸分泌抑制剂,具有抗溃疡活性、抗分泌和细胞保护... |
T6929 |
Pantoprazole sodium
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SKF96022 (sodium),泮托拉唑钠盐,泮托拉唑钠,BY1023 (sodium),SKF96022 sodium,Pantoloc,BY-1023 sodium,Pantecta |
Others
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HIF
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Proton pump
,
Autophagy
,
Apoptosis
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Pantoprazole sodium 是一种具有口服活性的质子泵抑制剂,是一种取代的苯并咪唑,是H+/K+-ATPase 抑制剂,IC50为 6.8 μM。它可以改善 pH 值稳定性,具有抗分泌和抗溃疡的作用。它联合阿霉素可显著增加肿瘤生... |
TCS1772 |
Dehydroabietic acid
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Dehydroabietate,脱氢枞酸;脱氢松香酸 |
Antifection
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Dehydroabietic acid 是 EBV-EA 活化抑制剂。 它是食物衍生化合物,可通过降低血浆葡萄糖、胰岛素水平、血浆甘油三酯 (TG) 和肝 TG 水平来治疗肥胖相关疾病。它的衍生物在动物模型中表现出抗分泌和抗胃蛋白酶作用。 |
T27539 |
Hexocyclium metilsulfate
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AB-803,Traline,AB 803,AB803 |
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Hexocyclium metilsulfate has anti-gastric secretory effects in humans. |
T10008 |
BTM-1086
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Others
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BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent. |
T39465 |
(Z)-Lafutidine
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(Z)-Lafutidine,(Z)-FRG-8813 |
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(Z)-Lafutidine ((Z)-FRG-8813) is a powerful histamine H2 receptor antagonist renowned for its anti-secretory and gastrop... |
TN4659 |
Nimbin
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COX
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Nimbin is an anti-pyretic, can be used to treat arthritis, hypoglycaemia, peptic ulcers, anti-secretory activity, and it... |
TMPY-04912 |
PLA2G2A Protein, Mouse, Recombinant (His Tag)
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Phospholipase A2, membrane associated, also known as Phosphatidylcholine 2-acylhydrolase 2A, Group IIA phospholipase A2,... |
TMPY-01705 |
PLA2G2A Protein, Human, Recombinant (His Tag)
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Phospholipase A2, membrane associated, also known as Phosphatidylcholine 2-acylhydrolase 2A, Group IIA phospholipase A2,... |
T76320 |
FIZZ-1 (32-51) (mouse)
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FIZZ-1 (32-51) (mouse) 是一种富含半胱氨酸的分泌蛋白,在过敏性气道炎症中,由巨噬细胞、支气管上皮和 II 型肺泡上皮细胞 (AEC) 高度表达。FIZZ1 (32-51) (mouse) 还对肺成纤维细胞有抗凋亡作用。... |
TMPY-03120 |
Prostaglandin D2 Synthase Protein, Human, Recombinant (His Tag), HPLC-verified
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PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s... |
TMPY-02597 |
IL-37 Protein, Human, Recombinant
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Interleukin 1 family member 7, or interleukin 37 (IL1F7 / IL37 / IL-1H4) is a secretory protein belonging to the Interle... |
TMPY-05069 |
Prostaglandin D2 Synthase Protein, Rat, Recombinant (His Tag)
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PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s... |
TMPY-04624 |
Prostaglandin D2 Synthase Protein, Mouse, Recombinant (His Tag)
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PTGDS, also known as L-PGDS, belongs to the calycin superfamily, lipocalin family. Lipocalins share limited regions of s... |
TN5221 |
(-)-Variabilin
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Variabilin, a novel inhibitor of human platelet aggregation, it is a potent RGD (Arg-Gly-Asp)-containing antagonist of t... |