T12895 |
SHA 68
|
847553-89-3
|
98%
|
|
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respectivel...
|
T8456 |
GALNON
|
475115-35-6
|
98%
|
|
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
|
TP1137L |
Pancreatic Polypeptide (human) acetate
|
|
98%
|
|
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.
|
TP1140L |
Neuropeptide Y (29-64), amide, human acetate
|
|
98%
|
|
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.
|
TP1380 |
Galanin (1-16), mouse, porcine, rat
|
125118-77-6
|
98%
|
|
Galanin(1-16),mouse,porcine,rat(TFA) is a Galanin receptor agonist with a Kd value of 3nM..
|
TP1982L |
Neuropeptide S (Rat) acetate
|
TP1982L
|
98%
|
|
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor. Neuropeptide S (Rat) acetate can b...
|
TP1981L |
Neuropeptide S (Mouse) acetate
|
TP1981L
|
98%
|
|
Neuropeptide S (Mouse) acetate is a bioactive peptide. Neuropeptide S (Mouse) acetate, as a neurotransmitter/neuromodulator of 20 amino acids, can be used for th...
|
T14671 |
BMS-193885
|
186185-03-5
|
98%
|
|
BMS-193885 is a selective, brain-penetrant, and competitive antagonist of the neuropeptide Y1 receptor with a Ki of 3.3 nM, and an IC50 of 5.9 nM for hY1.
|
TP1044L |
Pancreatic Polypeptide, rat acetate
|
|
98%
|
|
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.
|
TP1993L |
M617 acetate
|
|
98%
|
|
M617 acetate is a selective agonist of galanin receptor 1 (GAL1). M617 acetate acts through central GAL1, promotes GLUT4 expression, and enhances GLUT4 content i...
|
TP1059 |
Peptide YY (PYY) (3-36), human
|
126339-09-1
|
98%
|
|
Peptide YY (PYY) (3-36), human is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.
|
TP2206 |
[Leu31,Pro34]-Neuropeptide Y (porcine)
|
125580-28-1
|
98%
|
|
High affinity neuropeptide Y Y1 receptor agonist
|
TP1994L |
M871 acetate
|
|
98%
|
|
M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive ef...
|
T24121 |
GW438014A
|
469861-49-2
|
98%
|
|
GW438014A is a potent and selective NPY-Y5 receptor antagonist.GW438014A inhibits food intake and reduces body weight gain in obese rodents.
|
T21646L |
AR-M 1896 Acetate
|
T21646L
|
98%
|
|
AR-M 1896 Acetate is the selective agonist of GalR2.
|
TP1930L1 |
Spexin acetate(1370290-58-6 free base)
|
TP1930L1
|
98%
|
|
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galani...
|
T1997 |
JNJ-31020028
|
1094873-14-9
|
98%
|
|
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold ...
|
TP1937L1 |
RFRP-1 (human) acetate(311309-25-8 free base)
|
TP1937L1
|
98%
|
|
RFRP-1 (human) acetate is a potent endogenous NPFF receptor agonist (EC50 values are 0.0011 and 29 nM for NPFF2 and NPFF1, respectively). Attenuates contractile ...
|
T21611L |
BWX 46 Acetate
|
T21611L
|
98%
|
|
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
|
T8963 |
CYM2503
|
1308833-36-4
|
98%
|
|
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthos...
|