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Search Result

Search Results for "thyroid hormone receptor"

Targets

Thyroid hormone receptor(THR)

Compounds

Cat No. Product Name
T12073 ML-109 TSH Receptor
ML-109 是一种促甲状腺激素受体的有效激动剂，EC50值为 40 nM。
T5360 Eprotirome 伊罗替罗,KB2115 Thyroid hormone receptor(THR)
Eprotirome 是一种肝脏选择性甲状腺激素受体 (thyroid hormone receptor, TR) 激动剂。它对 TRβ的亲和力略高于TRα。它降低了低密度脂蛋白 (LDL) 胆固醇的浓度，可用于研究血脂异常和肥胖症。
T3595 Resmetirom VIA-3196,MGL3196 Thyroid hormone receptor(THR)
MGL-3196 是一种高度选择性的THR-β激动剂(EC50:0.21 μM)。
T40548 NH-3 Thyroid hormone receptor(THR)
NH-3 is a potent orally active thyroid hormone receptor (THR) antagonist which exhibits reversible behavior, demonstrate...
T5313 Sobetirome QRX-431,IACS-010759 Thyroid hormone receptor(THR)
Sobetirome 是一种甲状腺激素受体 β (TRβ) 激动剂，能够选择性的结合到TRβ-1(EC50:0.16 μM)。
T1653 Liothyronine 三碘甲状腺原氨酸,碘噻罗宁,Lyothyronine,L-3,3',5-Triiodothyronine,Triiodothyronine,Tresitope,O-(4-Hydroxy-3-iodophenyl)-3,5-diiodo-L-tyrosine,3,3',5-Triiodo-L-thyronine Thyroid hormone receptor(THR) , Endogenous Metabolite
O-(4-Hydroxy-3-iodophenyl)-3,5-diiodo-L-tyrosine 是一种有效的甲状腺激素，能够激活 β1 甲状腺激素受体 (TRβ1)。
T13492 3,5-Diiodothyropropionic acid 3,5-二碘甲腺丙酸,Ditpa cpd,C082182 Thyroid hormone receptor(THR)
3,5-Diiodothyropropionic acid 是一种甲状腺激素类似物，能够诱导 α-肌球蛋白重链 mRNA 表达。它可与甲状腺激素受体结合，作用于 TRα1 (Ka:2.40 M-1) 和 TRβ1 (Ka:4.06 M-1)...
T22355 L-Thyroxine sodium Levothyroxine sodium,L-T4 sodium,左旋甲状腺素钠,LT4 sodium Thyroid hormone receptor(THR)
Levothyroxine sodium 是一种合成的甲状腺激素，用于研究甲状腺功能减退症。DIO 酶能够将Levothyroxine 转化成具有生物活性的三碘甲状腺氨酸 (T3)。
T5383 D3-βArr NCGC00379308 TSH Receptor
D3-βArr 是一种促甲状腺激素受体正变构调节剂，通过直接激活促甲状腺激素受体启动 β-Arr 1 的易位，EC50为 11.6 μM。它还可增强促甲状腺激素介导的体外成骨细胞分化。
T1604 Tiratricol 替拉曲可,3,3',5-Triiodothyroacetic acid Thyroid hormone receptor(THR)
Tiratricol 是 T3 和 T4 甲状腺激素的代谢物；促进高脂血症、局部脂肪营养不良和肥胖。它已用于研究 Allan-Herndon-Dudley 综合征治疗的试验。
T12192 NCGC00229600 TSH Receptor , Others
NCGC00229600 是促甲状腺激素受体 (TSHR) 的变构反向激动剂。 NCGC00229600 抑制 TSH 和刺激 TSHR 的内源性激活抗体，可用于格雷夫斯病的研究。
T13072 Taltirelin acetate TA-0910 acetate Thyroid hormone receptor(THR)
Taltirelin acetate 是促甲状腺激素释放激素受体(TRH-R)超激动剂(IC50:910 nM)，能够刺激细胞溶质Ca2+浓度增加 (Ca2+释放) ，其EC50值为 36 nM。
T23673 AH-3960 AH3960 Thyroid hormone receptor(THR)
AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。
T1669 Liothyronine sodium 三碘代甲状腺素钠盐,Sodium L-3,3',5-triiodothyronine,Cytomel,T3 Sodium salt,Triostat,3,3',5-Triiodo-L-thyronine sodium Thyroid hormone receptor(THR)
Liothyronine sodium 是甲状腺激素，能够结合并激活 β1 甲状腺激素受体。
T8672 2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE 双酚0PPA,BisOPP-A Thyroid hormone receptor(THR)
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE 是针对促甲状腺激素受体（人）。
T0864 L-Thyroxine T4,NSC 36397,L-甲状腺素,Levothyroxine Thyroid hormone receptor(THR) , Endogenous Metabolite
L-Thyroxine (T4)是一种合成的甲状腺激素，用于甲状腺功能减退症的研究。在 DIO 酶作用下， L-Thyroxine (T4)转化成具有生物特性的三碘甲状腺氨酸 (T3)。
T36715 Tetrac
Tetrac (Tetraiodothyroacetic acid) is a thyrointegrin receptor antagonist derived from L-thyroxine (T4). It effectively ...
T7578 REVERSE T3 碘塞罗宁,3,3',5'-triiodo-L-thyronine Thyroid hormone receptor(THR)
Reverse T3 是由甲状腺素原脱碘后产生的甲状腺激素。它可抑制由其它甲状腺激素类似物引起的新生大鼠心肌细胞中钠电流增加的作用。
T16442 PCO371 2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl- Thyroid hormone receptor(THR)
PCO371 是口服具有活性的甲状旁腺激素受体 1 的完全激动剂，对 PTHR2 无作用
T6956 Protirelin Thyroliberin,TRH,Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,TRF,普罗瑞林 Endogenous Metabolite , Thyroid hormone receptor(THR)
Protirelin 是高度保守的神经肽，具有促甲状腺激素水平的激素控制作用，及神经调节功能。
ML-109
T12073
synonym:
Target:
Eprotirome
T5360
synonym: 伊罗替罗,KB2115
Target:
Resmetirom
T3595
synonym: VIA-3196,MGL3196
Target:
NH-3
T40548
synonym:
Target:
Sobetirome
T5313
synonym: QRX-431,IACS-010759
Target:
Liothyronine
T1653
synonym: 三碘甲状腺原氨酸,碘噻罗宁,Lyothyronine,L-3,3',5-Triiodothyronine,Triiodothyronine,Tresitope,O-(4-Hydroxy-3-iodophenyl)-3,5-diiodo-L-tyrosine,3,3',5-Triiodo-L-thyronine
Target:
3,5-Diiodothyropropionic acid
T13492
synonym: 3,5-二碘甲腺丙酸,Ditpa cpd,C082182
Target:
L-Thyroxine sodium
T22355
synonym: Levothyroxine sodium,L-T4 sodium,左旋甲状腺素钠,LT4 sodium
Target:
D3-βArr
T5383
synonym: NCGC00379308
Target:
Tiratricol
T1604
synonym: 替拉曲可,3,3',5-Triiodothyroacetic acid
Target:
NCGC00229600
T12192
synonym:
Target:
Taltirelin acetate
T13072
synonym: TA-0910 acetate
Target:
AH-3960
T23673
synonym: AH3960
Target:
Liothyronine sodium
T1669
synonym: 三碘代甲状腺素钠盐,Sodium L-3,3',5-triiodothyronine,Cytomel,T3 Sodium salt,Triostat,3,3',5-Triiodo-L-thyronine sodium
Target:
2,2-BIS(2-HYDROXY-5-BIPHENYLYL)PROPANE
T8672
synonym: 双酚0PPA,BisOPP-A
Target:
L-Thyroxine
T0864
synonym: T4,NSC 36397,L-甲状腺素,Levothyroxine
Target:
Tetrac
T36715
synonym:
Target:
REVERSE T3
T7578
synonym: 碘塞罗宁,3,3',5'-triiodo-L-thyronine
Target:
PCO371
T16442
synonym: 2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl-
Target:
Protirelin
T6956
synonym: Thyroliberin,TRH,Lopremone,pGlu-His-Pro-NH2,Synthetic thyrotropin-releasing hormone,TRF,普罗瑞林
Target:
1 2
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