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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T73618 | Adenylate | ||
Adenylate (Adk), also known as myokinase, is a phosphotransferase enzyme that catalyzes the interconversion of adenosine phosphates, playing a crucial role in the regulation of phosphate nucleotide levels and cellular en... | |||
T35031 | Valyl adenylate | Valyladenylate,Valyl-adenylate | |
Valyl adenylate is a peptide. | |||
T34961 | Tryptophyl adenylate | ||
Tryptophyl adenylate is a bioactive chemical. | |||
T34018 | Phenylalanyl adenylate | Phe-pA | |
Phenylalanyl adenylate is a bioactive chemical. | |||
T32903 | L-Seryl-amp | Seryl-adenylate | |
L-Seryl-amp is a peptide. | |||
T14129 | Adenylosuccinic acid | Aspartyl adenylate,Adenylosuccinate | Others |
Adenylosuccinic acid (Adenylosuccinate; Aspartyl adenylate) is a purine ribonucleoside monophosphate and plays a role in nucleotide cycle metabolite. Adenylosuccinic acid has the potential for the study of duchenne muscu... | |||
T80069 | PACAP (6-27) (human, ovine, rat) | Pituitary adenylate cyclase-activating peptide (6-27) | |
PACAP (6-27) (human, ovine, rat) serves as an antagonist for the PACAP receptor, inhibiting the catecholamine response of the canine adrenal gland to vasoactive intestinal peptide (VIP). This compound holds promise for r... | |||
T15658 | KH7 | cAMP , AChR | |
KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific. It has IC50s of 3-10 μM toward both recombinant purified human sACt protein and heterologously expressed sACt in cellular assays. KH7 is also a cAMP inhibito... | |||
TP1054 | PACAP (1-38), human, ovine, rat TFA | Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA) | |
PACAP (1-38), a novel neuropeptide isolated from the bovine hypothalamus is more active than vasoactive intestinal peptide (VIP) in stimulating adenylate cyclase (EC50=7 nM). PACAP 1-38 (10-9 M) increased substance P (SP... | |||
T16938 | ST034307 | Adenylyl cyclase | |
ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM). | |||
TP1878 | PACAP (1-38), human, ovine, rat | Pituitary Adenylate Cyclase Activating Polypeptide 38,PACAP 1-38 | PACAP |
PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues. | |||
T60003 | AC1-IN-1 | Adenylyl cyclase | |
AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM). | |||
T0322 | Fipexide | Dopamine Receptor , AChR | |
Fipexide (Attentil, Vigilor), a psychoactive drug of the piperazine chemical class, was developed in Italy in 1983. It was served as a nootropic drug in France and Italy, mainly for the therapy of senile dementia, but is... | |||
T10066 | 2',5'-Dideoxyadenosine | Adenylyl cyclase , Adrenergic Receptor , AChR | |
2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM). | |||
T0830 | Bithionol | Actamer | cAMP , Parasite |
Bithionol (Actamer), formerly marketed as an active ingredient in various topical drug products, was shown to be a potent photosensitizer with the potential to cause serious skin disorders. Approvals of the NDA's for bit... | |||
T16275 | NB001 | HTS 09836 | Adenylyl cyclase |
NB001 (HTS 09836) is an inhibitor of adenyl cyclase 1 exhibiting effects on neural and non-neural pain. | |||
T2939 | Forskolin | Coleonol,Colforsin | FXR , Adenylyl cyclase , AChR , Autophagy |
Forskolin (Coleonol) is a natural product, an adenylate cyclase activator (EC50=0.5 μM). Forskolin increases cAMP levels, activates PXR and FXR, and induces autophagy. Forskolin produces positive inotropic effects in the... | |||
T8702 | SKF-83566 | Dopamine Receptor , 5-HT Receptor , AChR | |
SKF-83566 is a blood-brain permeable and orally active antagonist of D1-like dopamine receptor and a weaker competitive 5-HT2 receptor antagonist with Ki of 11 nM | |||
T2172 | SQ22536 | 9-(tetrahydrofuran-2-yl)-9h-purin-6-amine,SQ 22536 | AChR |
SQ22536 (9-(tetrahydrofuran-2-yl)-9h-purin-6-amine) , the adenosine analogue 9-(Tetrahydro-2-furyl)adenine, inhibited adenylate cyclase activity of crude membrane preparations from catfish (Ictalurus melas) and rat isola... | |||
T11918 | Lysipressin | Lysine vasopressin,[Lys8]-Vasopressin | Others |
Lysipressin ([Lys8]-Vasopressin), Induces contraction of the rabbit urinary bladder smooth muscle, activate adenylate-cyclase. Lysipressin is Antidiuretic hormone that have been found in pigs and some marsupial families. |