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  • Neuropeptide Y Receptor
    (12)
  • Androgen Receptor
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    (10)
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Results for "

y5 receptor

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    30
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    9
    TargetMol | Peptide_Products
Neuropeptide Y5 receptor ligand-1
T74654322723-35-3
Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].
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L 152804
T156796508-43-6
L 152804 is a specific antagonist of the neuropeptide Y Y5 receptor and modulates food intake and energy expenditure thus causing weight loss in diet-induced obese mice.
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JNJ-31020028
JNJ 31020028
T19971094873-14-9
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold selectivity for Y2 versus human Y1 Y4 Y5 receptors.
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GW438014A
GW 438014 A, GW-438014-A
T24121469861-49-2
GW438014A is a potent, selective antagonist of the NPY-Y5 receptor, effectively inhibiting food consumption and curbing body weight gain in obese rodents.
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6-8 weeks
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Pancreatic Polypeptide (human) acetate
TP1137L
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4 Y5 receptor agonist.
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MK-0557
TQ0286328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
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FR252384
T10514447405-11-0
FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).
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3-6 months
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JNJ-5207787
T15620683746-68-1
JNJ-5207787 is a penetrates the blood-brain barrier neuropeptide Y Y2 receptor (Y2) antagonist. It is >100-fold selective versus human Y1, Y4, and Y5 receptors. JNJ-5207787 suppresses the binding of peptide YY with pIC50s of 7.0 and 7.1 for the human Y2 r
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Velneperit
S2367
T17222342577-38-2
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
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AR antagonist 10
T2054203068489-78-8
AR antagonist 10 (Compound Y5) is a potent, orally active androgen receptor (AR) antagonist with an IC50 value of 0.04 μM. It demonstrates a dual mechanism of action: antagonizing AR by disrupting AR dimerization and inducing AR degradation through the ubiquitin-proteasome pathway. This compound shows excellent activity against various resistant AR mutants and effectively inhibits the growth of LNCaP xenograft tumors. AR antagonist 10 is applicable for research in resistant prostate cancer.
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10-14 weeks
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LU AA33810
T22935304008-29-5
LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.
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NPY 5RA972
T23087439861-56-0
neuropeptide Y Y5 receptor antagonist
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ntncb hydrochloride
T23094191931-56-3
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
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6-8 weeks
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S 25585
T23287263849-50-9
S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.
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FMS586
FMS-586,FMS 586
T27345302556-51-0
FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.
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j-115814
UNII-81DP93CF8M, J-115814, (+ -)-
T32246329716-61-2
J-115814 is a potent feeding stimulant.
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BIIE 0246 hydrochloride
T36481
Potent, selective and competitive nonpeptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM). Displays > 650-fold selectivity for NPY Y2 over Y1, Y4 and Y5 receptors. Active in vivo.
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CGP71683 hydrochloride
CGP71683A
T5587192322-50-2
CGP71683 hydrochloride (CGP71683A) is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes.
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GW438014 free base
T69220469861-48-1
GW438014A is a selective NPY-Y5 receptor antagonist.
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6-8 weeks
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BIIE-0246 HCl
T69621246146-31-6
BIIE-0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor. BIIE-0246 displays > 650-fold selectivity over Y1, Y4 and Y5 receptors.
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10-14 weeks
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GR231118 TFA
T75910
GR231118 TFA, a neuropeptide Y C-terminus analogue, acts as a potent, competitive, and relatively selective antagonist at the human neuropeptide YY receptor, exhibiting a pKi of 10.4. It serves as a strong agonist at the human neuropeptide YY4 receptor with a pEC50 of 8.6 and a pKi of 9.6, while demonstrating weak agonistic activity at both human and rat neuropeptide YY2 and YY5 receptors. Additionally, this compound shows high affinity for the mouse neuropeptide YY6 receptor, with a pKi value of 8.8 [1].
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[D-Trp34]-Neuropeptide Y TFA
T75911
[D-Trp34]-Neuropeptide Y TFA is a potent and selective agonist for the neuropeptide Y (NPY) Y5 receptor, demonstrating significantly lower potency at the NPY Y1, Y2, Y4, and Y6 receptors. It significantly increases food intake in rats [1] [2].
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[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA
T75912
[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA acts as a specific agonist for the neuropeptide Y Y1 receptor and also activates Y4 and Y5 receptors, elevating blood pressure in anesthetized rats and enhancing food intake [1] [2].
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[cpp1-7,npy19-23,ala31,aib32,gln34]-hpancreatic polypeptide tfa
T75913
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide is a potent and selective neuropeptide Y Y5 receptor agonist, exhibiting a binding affinity with an IC50 of 0.24 nM for the hY5 receptor, and significantly stimulates food intake [1].
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