adrenoreceptor

(±)-Befunolol is a blocking agent of β-adrenoceptor.

Higenamine hydrochloride (norcoclaurine HCl) has been demonstrated to be a β2 adrenoreceptor agonist. Adrenergic receptors, or adrenoceptors, belong to the class of G protein–coupled receptors, and are the most prominent receptors in the adipose membrane, besides also being expressed in skeletal muscle tissue.

Quetiapine (ICI204636) is used for the therapy of schizophrenia, and for the treatment of acute manic episodes associated with bipolar I disorder. The mechanism of quetiapine' action is thought by mediated through antagonist activity at serotonin and dopamine receptors. Specifically, the D1 and D2 dopamine, the α1 adrenoreceptor and α2 adrenoreceptor, and 5-HT1A and 5-HT2 serotonin receptor subtypes are antagonized. Quetiapine also can inhibit the histamine H1 receptor.

Procaterol is an intermediate-acting β2 adrenoreceptor agonist. It is used for the treatment of asthma.

Bufuralol hydrochloride (Ro 3-4787 hydrochloride) is a potent non-selective, orally active β-adrenoreceptor antagonist with partial agonist activity, which is also a CYP2D6 probe substrate [1] [2].

Fenoterol hydrobromide is an orally active and selective β2-adrenoceptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.

α2-adrenoreceptor antagonist

Broxaterol is a β2 adrenoreceptor agonist. It is part of a class of drugs that affect the smooth muscle receptors in the body.

L-Mabuterol HCl is a selective agonist of β2 adrenoreceptor.

Befunolol is a beta blocker with intrinsic sympathomimetic activity and also acts as a β adrenoreceptor partial agonist.

Hexoprenaline Sulfate is a selective beta2-adrenoreceptor agonist. Hexoprenaline Sulfate is active in man as a bronchodilator by the oral or intravenous routes and by inhalation. Hexoprenaline Sulfate is indicated for use in the treatment of bronchospasm

Mabuterol is a selective agonist of β2 adrenoreceptor with no beta 1-stimulation. Mabuterol inhibited the positive inotropic effect of isoprenaline at 10(-7) g/ml and decreased the maximum driving frequency at 3 X 10(-6) g/ml. Mabuterol was 3 times more p

Pirbuterol, a short-acting β2 adrenoreceptor agonist, has bronchodilating action used in the treatment of asthma.

Reproterol hydrochloride, a β2 adrenoreceptor agonist, is used to treat asthma and chronic obstructive pulmonary disease (COPD).

Ro 16-8714 is an agonist of beta-adrenoreceptor with antihyperglycemic and thermogenic properties.

Vatinoxan is a peripheral α2 adrenoreceptor antagonist.

Etiguanfacine(SSP-1871) is a agonist of α2-adrenoreceptor.

Fasobegron is a agonist of β3-adrenoreceptor .

Lubabegron(LY488756) is used as an agonist of β3-adrenoreceptor in veterinary.

Ronactolol is an aminopropanol derivative with beta-adrenoreceptor blocking activity.

Zoleprodolol is a antagonist of adrenoreceptor.

Povafonidine (PGE-6201204) is a potent alpha-2 adrenoreceptor agonist that constricts blood vessels and reduces mucosal congestion, making it useful for nasal congestion research [1].

Oxyfedrine is an orally active β-adrenoreceptor agonist. Oxyfedrine is a vasodilator that reduces coronary vessels tonicity that can be used in cardiovascular disease research[1] [2].

Aminomenthylnorepinephrine is a partial agonist of the beta-adrenoreceptor that causes irreversible inactivation.