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Aromatase

Aromatase is the enzyme that catalyzes a key aromatization step in the synthesis of estrogen. It converts the enone ring of androgen precursors such as testosterone, to a phenol, completing the synthesis of estrogen.

  • Aminoglutethimide
    T1103125-84-8
    Aminoglutethimide (BA-16038), an aromatase inhibitor, is used in the therapy of advanced BREAST Y.
    • $54
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  • Vorozole
    T26322129731-10-8In house
    Vorozole (R83842) is an orally active, potent, and selective nonsteroidal aromatase inhibitor.Vorozole exhibits antitumor activity in vivo and may be used in the study of breast cancer.
    • $191
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  • Letrozole
    T1590112809-51-5
    Letrozole (CGS 20267) is an Aromatase Inhibitor. The mechanism of action of letrozole is as an Aromatase Inhibitor.
    • $31
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    TargetMol | Citations Cited
  • Anastrozole
    T0393120511-73-1
    Anastrozole (ZD1033)(ZD1033), a potent and highly selective aromatase (CYP19) inhibitor (IC50 = 15 nM), has no obvious effect on adrenocorticoid hormone synthesis.
    • $45
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  • Finrozole
    T27320160146-17-8In house
    Finrozole (MPV 2213ad) is a novel selective aromatase inhibitor that is partially reversible for breast development.
    • $130
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  • (-)-Vorozole
    T26322L132042-69-4In house
    (-)-Vorozole is an orally active non-steroidal aromatase inhibitor with potency and selectivity. (-)-Vorozole has demonstrated antitumor activity in in vivo experiments. (-)-Vorozole is used in the study of breast cancer.
    • $195
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    TargetMol | Inhibitor Sale
  • Androsta-1,4,6-triene-3,17-dione
    T10321633-35-2In house
    Androsta-1,4,6-triene-3,17-dione is a lipophilic and specific aromatase inhibitor (Ki: 0.18 μM). It inhibits estrogen biosynthesis and shows antifertility effects. It induces impairment of spatial memory.
      6-8 weeks
      Inquiry
      TargetMol | Inhibitor Sale
    • Endoxifen
      T4281110025-28-0
      (E/Z)-Endoxifen ((E/Z)-Endoxifen) is an active metabolite of tamoxifen produced by the sequential action of cytochrome P450 (CYP) isoforms, including CYP2D6. It is a strong anti-estrogen, as it has an approximately 100-fold greater affinity for estrogen receptors than tamoxifen. As the efficient conversion of tamoxifen to endoxifen depends on CYP2D6, polymorphisms in this CYP isoform can impact the effectiveness of TMX treatment.
      • $41
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      TargetMol | Citations Cited
    • Eriodictyol chalcone
      TN398714917-41-0
      Eriodictyol chalcone has anti-plasmodial effects on P. falciparum growth.
      • $290
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      TargetMol | Inhibitor Sale
    • 3-(3,4-Dimethoxyphenyl)propanoic acid
      T16922107-70-2
      3-(3,4-Dimethoxyphenyl)propanoic acid (3,4-Dimethoxyhydrocinnamic acid) is an orally active short-chain fatty acid (SCFAs). It promotes γ-globin gene expression and erythropoiesis in vivo and can be used in beta hemoglobinopathies and other anemias.
      • $29
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      TargetMol | Inhibitor Sale
    • Minamestane
      T71708105051-87-4
      Minamestane is a novel irreversible aromatase inhibitor.Minamestane induces time-dependent inhibition of human placental aromatase with a half-life of 4 minutes and a K of 59 nM.Minamestane has antitumor activity.
      • $128
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    • LY 43578
      T2791826766-35-8
      LY 43578 is an orally active aromatase inhibitor. LY43578 could inhibit O-demethylation of P-450-dependent p-nitroanisole and N-demethylation of ethylmorphine (IC50 of 0.3 and 5 μm, respectively) in rat liver microsomes. LY 43578 can be used to study neurological and cardiovascular diseases.
      • $30
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    • YM 511
      T23549148869-05-0
      YM 511 is a highly specific non-steroidal aromatase inhibitor. YM 511 inhibits aromatase activities in microsomes from rat ovary and human placenta competitively (IC50s of 0.4 and 0.12 nM, respectively). YM 511 slightly inhibits production of other steroid hormones. YM 511 has the potential for suppressing estrogen-dependent action research without affecting serum levels of other steroid hormones.
      • $54
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    • Fadrozole
      T7197102676-47-1
      Fadrozole is a nonsteroidal aromatase inhibitor with potential antineoplastic activity(IC50 : 6.4 nM)
      • $45
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    • alpha-Naphthoflavone
      T2O2744604-59-1
      alpha-Naphthoflavone (7,8-benzoflavone), a synthetic flavonoid, is a potent inhibitor of aromatase with an I50 value of 0.5 μM.
      • $39
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    • Calceolarioside B
      T3899105471-98-5
      Calceolarioside B (Desrhamnosyl isoacteoside) displays inhibition of aromatase. Calceolarioside B displays inhibition of human recombinant PKCalpha.
      • $51
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    • Org30958
      T1231999957-90-1
      Org30958 is a potent inhibitor of aromatase in vivo.
      • $1,520
      Backorder
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    • Oleuropein
      T691732619-42-4
      Oleuropein is an antioxidant polyphenol isolated from olive leaf.
      • $43
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    • Exemestane
      T1587107868-30-4
      Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.
        Inquiry
      • Flavanone
        T0530487-26-3
        Flavanone (2-Phenylchroman-4-one)s from citrus fruits have also been shown to exert beneficial effects on human vascular function. In particular, chronic interventions with orange juice, or the pure flavanone hesperidin, resulted in a decrease in blood pressure in overweight volunteers and acute improvements in microvascular reactivity.
        • $40
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      • Fadrozole hydrochloride
        T7556102676-31-3
        Fadrozole hydrochloride (CGS 16949A) is a model aromatase inhibitor that has been shown to suppress estrogen production in the ovaries of fish.
        • $42
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      • Obacunone
        T3390751-03-1
        Obacunone has cytotoxicity in androgen-dependent human prostate Y cells. Obacunone exerts an antivirulence effect on S. Typhimurium and may serve as a lead compound for development of antivirulence strategies for S. Typhimurium. Obacunone may have the pot
        • $100
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