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Search Result

Search Results for " gsk-3 "

Targets

GSK-3 Apoptosis GSK-3

105

Compounds

3

Natural Products

67

Recombinant Proteins

2

Libraries

Cat No. Product Name Synonyms Targets
T35554 GSK-3β inhibitor 3 Apoptosis , GSK-3
GSK-3β inhibitor 3 is a covalent inhibitor (IC50: 6.6 μM) of glycogen synthase kinase 3β (GSK-3β) that is potent, selective, and irreversible.GSK-3β inhibitor 3 can be used to study acute promyelocytic leukemia.
T77342 GSK-3 inhibitor 3 GSK-3 , Microtubule Associated
GSK-3 inhibitor 3 is a selective, orally active, brain-permeable GSK-3 inhibitor that inhibits GSK-3α and GSK-3β with IC50s of 0.35 nM and 0.25 nM, respectively.GSK-3 inhibitor 3 reduces the phosphorylation level of tau ...
T77341 GSK-3 inhibitor 4 GSK-3 , CDK
GSK-3 inhibitor 4 is an orally active and brain-permeable triple inhibitor of GSK-3, CDK2 and CDK5 with inhibitory effects on GSK-3β, GSK-3α, CDK2 and CDK5, with IC50 values of 0.56 nM, 0.45 nM, 0.47 μM, 0.68 μM, respect...
T1917 GSK 3 Inhibitor IX BIO,GSK 3 IX,6-BIO,6-Bromoindirubin-3'-oxime,MLS 2052,6-bromoindirubin-3-oxime Apoptosis , GSK-3 , Tyrosine Kinases , CDK
GSK 3 Inhibitor IX (6-BIO) is a selective reversible, ATP-competitive inhibitor of GSK-3α/β and CDK1-cyclinB complex. It inhibits (GSK-3α/β)/CDK1/CDK5 activity with IC50 values of 5 nM/320 nM/83 nM, respectively.
T77554 GSK-3 Inhibitor 5 4-Cyanophenacyl bromide GSK-3
GSK-3 Inhibitor 5 (4-Cyanophenacyl bromide) is a ketone derivative that is used as an intermediate in pharmaceuticals and organic synthesis, and inhibits glycogen synthase kinase 3 (GSK-3).
T78578 GSK-3 Inhibitor XIII GSK-3
GSK-3 Inhibitor XIII, an ATP-competitive GSK-3 inhibitor (Ki: 24 nM), can be used to study diabetes and obesity.
T35555 GSK-3/CDK5/CDK2-IN-1 GSK-3/CDK5/CDK2-IN-1
GSK-3/CDK5/CDK2-IN-1 is an imidazole derivative compound that inhibits cdk5, cdk2, and GSK-3.it has demonstrated applications in cancer research and the study of neurodegenerative diseases [1].
T11467 GSK-3β inhibitor 1 GSK-3
GSK-3β inhibitor 1 is an inhibitor of GSK-3β( IC50 of 4.9 nM) and demonstrates high antidiabetic efficacy.
T2073 GSK2636771 GSK 2636771,GSK-2636771 PI3K
GSK2636771, an effective, specific, orally bioavailable, PI3Kβ inhibitor, has been used in cancer, lymphoma, solid neoplasm, recurrent solid neoplasm, and advanced malignant neoplasm.
T9725 GSK-3β inhibitor 10 Others
GSK-3β inhibitor 10 has skin-whitening, anti-oxidizing and PPAR activities.
T6787 BIO-acetoxime BIA,GSK-3 Inhibitor X Apoptosis , GSK-3 , HSV
BIO-acetoxime (GSK-3 Inhibitor X) is a potent dual GSK3α/β inhibitor with IC50 of 10 nM, >240-fold selectivity over CDK5/p25, CDK2/cyclin A and CDK1/cyclin B.
T9178 (E/Z)-GSK-3β inhibitor 1 GSK-3β inhibitor 1 GSK-3
(E/Z)-GSK-3β inhibitor 1 is a glycogen synthase kinase 3β (GSK-3β) inhibitor and demonstrates high antidiabetic efficacy.
T11468 GSK-3 inhibitor 1 GSK-3
GSK-3 inhibitor 1 is a GSK-3 inhibitor.
T2357 GSK1059615 GSK 1059615,GSK-1059615 Apoptosis , PI3K , mTOR
GSK1059615 has been used in trials studying the treatment of Lymphoma, Solid Tumours, Endometrial Cancer, Solid Tumor Cancer, and Metastatic Breast Cancer.
T1861 Omipalisib GSK458,GSK2126458 PI3K , mTOR , Autophagy
Omipalisib (GSK2126458) is a small-molecule pyridylsulfonamide inhibitor of phosphatidylinositol 3-kinase (PI3K) with potential antineoplastic activity.
T22817 GSK 789472 hydrochloride GSK-789472 HCl,1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride,4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one Dopamine Receptor
GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
T6187 TDZD-8 GSK-3β Inhibitor I,NP 01139 GSK-3
TDZD-8 (NP 01139) is an inhibitor of GSK-3β, with an IC50 of 2 μM; minimal inhibitory effect observed on CDK1, casein kinase II, PKA and PKC.
T24111 GSK3i XIII GSK3 inhibitor XIII,GSK3iXIII,GSK3i-XIII GSK-3
GSK3i XIII (GSK3 inhibitor XIII) is a GSK-3 ATP-binding site inhibitor.
T1881 AR-A014418 AR 0133418,GSK-3beta Inhibitor VIII,AR 014418,GSK 3β inhibitor VIII GSK-3
AR-A014418 (GSK 3β inhibitor VIII) is an ATP-competitive, and selective GSK3β inhibitor.
T22820 GSK J5 HCl (1394854-51-3 free base) GSK J5 HCl Others
GSK J5 HCl is the hydrochloride form of GSK J5. GSK J5 is an inactive isomer of GSK J4 and a cell-permeable ester derivative of inactive control GSK J2.
T1965 Bikinin Abrasin Others , GSK-3
Bikinin (Abrasin), a potent inhibitor of plant GSK-3/Shaggy-like kinase, activates BR signaling downstream of the BR receptor.
T14066 9-ING-41 Apoptosis , GSK-3 , Autophagy
9-ING-41 is a glycogen synthase kinase-3 inhibitor.
T9987 GSK3-IN-1 GSK-3
GSK3-IN-1 is a GSK3B-glycogen synthase kinase-3 beta inhibitor.
T19840 GSK-F1 PI4KA inhibitor-F1 PI4K
GSK-F1 (PI4KA inhibitor-F1) is a novel potent PI4KA inhibitor.
T10202 A 1070722 GSK-3
A 1070722 is a potent and selective GSK-3 inhibitor, with a Ki of 0.6 nM for both GSK-3α and GSK-3β. It can penetrate the blood-brain barrier (BBB) and accumulates in brain regions, thus potential for PET radiotracer for...
T1741 AZD1080 GSK-3
AZD1080 is a selective, orally active, brain permeable GSK3 inhibitor.
T1957 AZD2858 GSK-3
AZD2858 is a selective GSK-3 inhibitor, inhibiting tau phosphorylation at the S396 site and activating Wnt signaling pathway.
T5956 VP3.15 dihydrobromide GSK-3 , PDE
VP3.15 dihydrobromide is a potent, orally bioavailable and CNS-penetrant dual phosphodiesterase (PDE7- glycogen synthase kinase (GSK)3 inhibitor(with IC50s of 1.59 μM , 0.88 μM,respectively.)
T1755 LY2090314 GSK-3
LY2090314, an effective GSK-3α/β inhibitor (IC50: 1.5 nM/0.9 nM), may improve the efficacy of platinum-based chemotherapy regimens. LY2090314 has been used in trials studying the treatment of Leukemia, Advanced Cancer, a...
T2166 TWS119 GSK-3 , Autophagy
TWS119 is a GSK-3β inhibitor; capable of inducing neuronal differentiation
T3077 SB 216763 SB216763 GSK-3 , Autophagy
SB 216763 (SB216763) is an effective and specific GSK-3α/β inhibitor (IC50: 34.3 nM).
T2261 IM-12 IM 12 GSK-3
IM-12, an effective GSK-3β inhibitor(IC50=53 nM), regulates Wnt signalling.
T21966 MeBIO GSK-3 , Aryl Hydrocarbon Receptor , CDK
MeBIO is an agonist of aryl hydrocarbon receptor, with IC50 of 44 and 55 μM for GSK-3 and CDK1/CyclinB, respectively. MeBIO does not affect GSK-3β.
T21956 GSK3β inhibitor II GSK-3
GSK3β inhibitor II is a GSK3β inhibitor. GSK3β inhibitor II exhibits the research potential of Alzheimer's disease (AD).
T3684 CP21R7 CP21 GSK-3 , PKC
CP21R7 (CP21) is an effective and specific GSK3β inhibitor. It is used as an activator of stem cells prior to the induction of differentiation of stem cells to smooth muscle and endothelial cells. CP21R7 can be combined ...
T7361 Verucerfont NBI77860,GSK561679 CRFR
Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .
T5200 Indirubin-3'-monoxime Indirubin-3'-oxime GSK-3 , Lipoxygenase , CDK
Indirubin-3'-monoxime (Indirubin-3'-oxime) is a potent inhibitor of GSK3β (IC50: 22 nM) and also inhibits CDKs ( (IC50s: 100/180/250 nM for Cdk5/p35, Cdk1/cyclin B, Cdk2/cyclin E).
T12664 (Rac)-BRD0705 Others
(Rac)-BRD0705 is a less active racemate of BRD0705. BRD0705 is an effective and selective inhibitor of GSK3α.
T9138 Indirubin-3′-oxime Indirubin-3'-monoxime GSK-3 , CDK , JNK
Indirubin-3′-oxime is an effective inhibitor of cyclin-dependent protein kinases, and may play an obligate role in neuronal apoptosis in Alzheimer's disease.
T10606 BRD0705 GSK-3
BRD0705 is a potent, paralog selective and orally active GSK3α inhibitor (IC50: 66 nM; Kd: 4.8 μM). BRD0705 displays increased selectivity for GSK3α (8-fold) versus GSK3β (IC50: 515 nM).
T3074 CHIR 98024 CHIR98014 GSK-3 , S6 Kinase
CHIR 98024 is a potent GSK-3α/β inhibitor with IC50 of 0.65 nM/0.58 nM in cell-free assays, with the ability to distinguish GSK-3 from its closest homologs Cdc2 and ERK2.
T2608 CHIR-98014 CHIR 98014,CT98014,CHIR98014 FGFR , GSK-3 , Src , S6 Kinase
CHIR-98014 (CT98014) is a selective GSK3 inhibitor; potentiate insulin activation of glucose transport and utilization in vitro and in vivo.
T15438 GSK3186899 3,3,3-trifluoro-N-[4-[[3-[(2R)-2-methylmorpholin-4-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]cyclohexyl]propane-1-sulfonamide,DDD-853651 Parasite
GSK3186899 is an inhibitor of Cdc2-related kinase 12 with an EC50 of 1.4 μM for L. donovani.
T9611 PF-04802367 GSK-3
PF-04802367 is a highly selective GSK-3 inhibitor with an IC50 of 2.1 nM based on a recombinant human GSK-3β enzyme assay and 1.1 nM based on ADP-Glo assay. It shows desirable central nervous system (CNS) properties and ...
T3067 Tideglusib NP-12,NP031112 GSK-3
Tideglusib (NP031112), a non-ATP competitive inhibitor of glycogen synthase kinase 3 (GSK-3), is with anti-inflammatory and neuroprotective activities.
T11447 GNF4877 GSK-3 , DYRK
GNF4877 is a potent DYRK1A and GSK3β inhibitor (IC50s: 6 nM and 16 nM). It leads to blockade of nuclear factor of activated T-cells (NFATc) nuclear export and increased β-cell proliferation cells.
T22012 7BIO FLT , DYRK , Aurora Kinase
7-bromoindirubin-3'-oxime (7BIO) is a caspase independent nonapoptotic cell death inducer. 7BIO is an inhibitor of FLT3, DYRK1A, DYRK2, Aurora B and Aurora C kinases.
T6659 SB 415286 SB415286 Apoptosis , GSK-3
SB 415286 is a potent GSK3α inhibitor with IC50/Ki of 78 nM/31 nM with equally effective inhibition of GSK-3β.
T10608 BRD5648 (R)-BRD0705 GSK-3
BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705. BRD0705 is a GSK3α inhibitor (IC50: 66 nM; Kd: 4.8 μM) and can be used in acute myeloid leukemia (AML) studies.
T2277 Losmapimod GSK-AHAB,GW856553X,GW856553,SB856553 p38 MAPK , Autophagy
Losmapimod (GSK-AHAB) (GW856553X; SB856553; GSK-AHAB) is a specific, potent, and orally active p38 MAPK inhibitor (pKi: 8.1/7.6 for p38α/β).

Compounds

GSK-3β inhibitor 3
T35554
Synonym:
Target: Apoptosis, GSK-3
GSK-3 inhibitor 3
T77342
Synonym:
Target: GSK-3, Microtubule Associated
GSK-3 inhibitor 4
T77341
Synonym:
Target: GSK-3, CDK
GSK 3 Inhibitor IX
T1917
Synonym: BIO,GSK 3 IX,6-BIO,6-Bromoindirubin-3'-oxime,MLS 2052,6-bromoindirubin-3-oxime
Target: Apoptosis, GSK-3, Tyrosine Kinases, CDK
GSK-3 Inhibitor 5
T77554
Synonym: 4-Cyanophenacyl bromide
Target: GSK-3
GSK-3 Inhibitor XIII
T78578
Synonym:
Target: GSK-3
GSK-3/CDK5/CDK2-IN-1
T35555
Synonym: GSK-3/CDK5/CDK2-IN-1
Target:
GSK-3β inhibitor 1
T11467
Synonym:
Target: GSK-3
GSK2636771
T2073
Synonym: GSK 2636771,GSK-2636771
Target: PI3K
GSK-3β inhibitor 10
T9725
Synonym:
Target: Others
BIO-acetoxime
T6787
Synonym: BIA,GSK-3 Inhibitor X
Target: Apoptosis, GSK-3, HSV
(E/Z)-GSK-3β inhibitor 1
T9178
Synonym: GSK-3β inhibitor 1
Target: GSK-3
GSK-3 inhibitor 1
T11468
Synonym:
Target: GSK-3
GSK1059615
T2357
Synonym: GSK 1059615,GSK-1059615
Target: Apoptosis, PI3K, mTOR
Omipalisib
T1861
Synonym: GSK458,GSK2126458
Target: PI3K, mTOR, Autophagy
GSK 789472 hydrochloride
T22817
Synonym: GSK-789472 HCl,1-phenyl-3-(piperidin-2-ylmethyl)imidazolidin-2-one hydrochloride,4,5-Dihydro-1-phenyl-3-(2-piperidinyl)methylimidazol-2(1H)-one
Target: Dopamine Receptor
TDZD-8
T6187
Synonym: GSK-3β Inhibitor I,NP 01139
Target: GSK-3
GSK3i XIII
T24111
Synonym: GSK3 inhibitor XIII,GSK3iXIII,GSK3i-XIII
Target: GSK-3
AR-A014418
T1881
Synonym: AR 0133418,GSK-3beta Inhibitor VIII,AR 014418,GSK 3β inhibitor VIII
Target: GSK-3
GSK J5 HCl (1394854-51-3 free base)
T22820
Synonym: GSK J5 HCl
Target: Others
Bikinin
T1965
Synonym: Abrasin
Target: Others, GSK-3
9-ING-41
T14066
Synonym:
Target: Apoptosis, GSK-3, Autophagy
GSK3-IN-1
T9987
Synonym:
Target: GSK-3
GSK-F1
T19840
Synonym: PI4KA inhibitor-F1
Target: PI4K
A 1070722
T10202
Synonym:
Target: GSK-3
AZD1080
T1741
Synonym:
Target: GSK-3
AZD2858
T1957
Synonym:
Target: GSK-3
VP3.15 dihydrobromide
T5956
Synonym:
Target: GSK-3, PDE
LY2090314
T1755
Synonym:
Target: GSK-3
TWS119
T2166
Synonym:
Target: GSK-3, Autophagy
SB 216763
T3077
Synonym: SB216763
Target: GSK-3, Autophagy
IM-12
T2261
Synonym: IM 12
Target: GSK-3
MeBIO
T21966
Synonym:
Target: GSK-3, Aryl Hydrocarbon Receptor, CDK
GSK3β inhibitor II
T21956
Synonym:
Target: GSK-3
CP21R7
T3684
Synonym: CP21
Target: GSK-3, PKC
Verucerfont
T7361
Synonym: NBI77860,GSK561679
Target: CRFR
Indirubin-3'-monoxime
T5200
Synonym: Indirubin-3'-oxime
Target: GSK-3, Lipoxygenase, CDK
(Rac)-BRD0705
T12664
Synonym:
Target: Others
Indirubin-3′-oxime
T9138
Synonym: Indirubin-3'-monoxime
Target: GSK-3, CDK, JNK
BRD0705
T10606
Synonym:
Target: GSK-3
CHIR 98024
T3074
Synonym: CHIR98014
Target: GSK-3, S6 Kinase
CHIR-98014
T2608
Synonym: CHIR 98014,CT98014,CHIR98014
Target: FGFR, GSK-3, Src, S6 Kinase
GSK3186899
T15438
Synonym: 3,3,3-trifluoro-N-[4-[[3-[(2R)-2-methylmorpholin-4-yl]-1H-pyrazolo[3,4-d]pyrimidin-6-yl]amino]cyclohexyl]propane-1-sulfonamide,DDD-853651
Target: Parasite
PF-04802367
T9611
Synonym:
Target: GSK-3
Tideglusib
T3067
Synonym: NP-12,NP031112
Target: GSK-3
GNF4877
T11447
Synonym:
Target: GSK-3, DYRK
7BIO
T22012
Synonym:
Target: FLT, DYRK, Aurora Kinase
SB 415286
T6659
Synonym: SB415286
Target: Apoptosis, GSK-3
BRD5648
T10608
Synonym: (R)-BRD0705
Target: GSK-3
Losmapimod
T2277
Synonym: GSK-AHAB,GW856553X,GW856553,SB856553
Target: p38 MAPK, Autophagy
1 2 3
Cat No. Product Name Synonyms Targets
T6S0653 Linarin Buddleoflavonoloside,Buddleoside,Acacetin-7-O-rutinoside,Acaciin,Linarine TNF , AChE
1. Linarin (Acacetin-7-O-rutinoside) (acacetin-7-O-β-d-rutinoside) shows selective dose dependent inhibitory effect on acetylcholinesterase. 2. Linarin alleviates GalN/LPS-induced liver injury by suppressing TNF-α-mediat...
TN1702 Glycycoumarin P450 , JNK , AMPK , Autophagy
Glycycoumarin is an estrogen agonist, it shows moderate inhibitory effects against CYP1A2 and CYP2B6.
T27977 Manzamine A Keramamine A
Manzamine A is a GSK-3 inhibitor and vacuolar ATPase uncoupler found in marine sponges. It inhibits autophagy and tumor growth in cancer models, suppresses foam cell formation in macrophages, prevents growth of gram nega...

Natural Products

Linarin
T6S0653
Synonym: Buddleoflavonoloside,Buddleoside,Acacetin-7-O-rutinoside,Acaciin,Linarine
Target: TNF, AChE
Glycycoumarin
TN1702
Synonym:
Target: P450, JNK, AMPK, Autophagy
Manzamine A
T27977
Synonym: Keramamine A
Target:

Recombinant Proteins

Species：
Human (60)
Mouse (6)
Canine (1)
Expression System：
HEK293 (49)
Baculovirus-Insect Cells (7)
Human Cells (7)
E. coli (4)
Tag：
His (24)
hFc (9)
Tag Free (6)
mFc (5)
C-Fc (4)
C-6His (3)
C-His-Avi (3)
C-Avi (2)
GST (2)
His,AVI (2)
Cat No. Product Name Species Expression System
TMPY-04439 GSK3B Protein, Mouse, Recombinant (His) Mouse Baculovirus-Insect Cells
GSK3B is a serine-threonine kinase, belonging to the glycogen synthase kinase subfamily. It Contains 1 protein kinase domain, and is expressed in the testis, thymus, prostate, and ovary and weakly expressed in the lung, ...
TMPY-04147 Frizzled 10 Protein, Human, Recombinant (His) Human HEK293
Frizzled-1, also known as Fz-1, CD35 and FZD1, is a multi-pass membrane protein which belongs to theG-protein coupled receptor Fz/Smo family. Frizzled-1 / FZD1 is abundantly expressed in the cerebellum, followed by ce...
TMPY-01797 Frizzled 10 Protein, Mouse, Recombinant (hFc) Mouse HEK293
Frizzled-1, also known as Fz-1, CD35 and FZD1, is a multi-pass membrane protein which belongs to theG-protein coupled receptor Fz/Smo family. Frizzled-1 / FZD1 is abundantly expressed in the cerebellum, followed by ce...
TMPY-01798 Frizzled 10 Protein, Mouse, Recombinant (His) Mouse HEK293
Frizzled-1, also known as Fz-1, CD35 and FZD1, is a multi-pass membrane protein which belongs to theG-protein coupled receptor Fz/Smo family. Frizzled-1 / FZD1 is abundantly expressed in the cerebellum, followed by ce...
TMPY-04140 Frizzled 10 Protein, Human, Recombinant (hFc) Human HEK293
Frizzled-1, also known as Fz-1, CD35 and FZD1, is a multi-pass membrane protein which belongs to theG-protein coupled receptor Fz/Smo family. Frizzled-1 / FZD1 is abundantly expressed in the cerebellum, followed by ce...
TMPY-04142 RANK/TNFRSF11A Protein, Human, Recombinant (hFc) Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small i...
TMPY-00132 Mesothelin Protein, Human, Recombinant Human HEK293
The megakaryocyte potentiating factor belongs to the mesothelin family. This family is comprised of several mammalian pre-pro-megakaryocyte potentiating factor precursor (MPF) or mesothelin proteins. Mesothelin is a glyc...
TMPY-00357 HNT/NTM Protein, Human, Recombinant (His) Human HEK293
NTM (Neurotrimin) is a Protein Coding gene. 4 alternatively spliced human isoforms have been reported. This gene encodes a member of the IgLON (LAMP, OBCAM, Ntm) family of immunoglobulin (Ig) domain-containing glycosylph...
TMPY-06986 FGF-8b Protein, Human, Recombinant Human E. coli
In mammalian embryos, transient Fgf8 expression defines the developing isthmic region, lying between the midbrain and the first rhombomere, but there has been uncertainty about the existence of a distinct isthmic segment...
TMPY-05748 CD45 Protein, Human, Recombinant (aa 26-577, His) Human HEK293
The cluster of differentiation (CD) system is commonly used as cell markers in Immunophenotyping. Different kinds of cells in the immune system can be identified through the surface CD molecules associating with the immu...
TMPY-04683 CD47 Protein, Human, Recombinant Human HEK293
CD47 contains 1 Ig-like V-type (immunoglobulin-like) domain and is a receptor for the C-terminal cell binding domain of thrombospondin. It may play a role in membrane transport and signal transduction. CD47 is also a mem...
TMPY-01020 Periostin/OSF-2 Protein, Human, Recombinant (His) Human HEK293
Periostin ( POSTN ), also known as OSF2 (osteoblast specific factor 2), is a heterofunctional secreted extracellular matrix (ECM) protein comprised of four fasciclin domains that promotes cellular adhesion and movement, ...
TMPY-01897 PRSS3 Protein, Human, Recombinant (His) Human HEK293
Trypsin-3, also known as Trypsin III, brain trypsinogen, Serine protease 3 and PRSS3, is a secreted protein that belongs to the peptidase S1 family. Trypsin-3 / PRSS3 is expressed is in pancreas and brain. It contains on...
TMPY-05191 CD47 Protein, Human, Recombinant, Biotinylated Human HEK293
CD47 contains 1 Ig-like V-type (immunoglobulin-like) domain and is a receptor for the C-terminal cell binding domain of thrombospondin. It may play a role in membrane transport and signal transduction. CD47 is also a mem...
TMPY-03763 Neuropilin-2 Protein, Human, Recombinant (hFc) Human HEK293
Neuropilin-2 (NRP-2) which is related to NRP-1, is a type I? transmembrane glycoprotein and has the structure characteristic with five main extracellular domains: two complement binding (CUB) domains, two coagulation fac...
TMPY-00892 Neuropilin-2 Protein, Human, Recombinant (His) Human HEK293
Neuropilin-2 (NRP-2) which is related to NRP-1, is a type I? transmembrane glycoprotein and has the structure characteristic with five main extracellular domains: two complement binding (CUB) domains, two coagulation fac...
TMPY-04935 CD47 Protein, Human, Recombinant (aa 1-139, His) Human HEK293
CD47 contains 1 Ig-like V-type (immunoglobulin-like) domain and is a receptor for the C-terminal cell binding domain of thrombospondin. It may play a role in membrane transport and signal transduction. CD47 is also a mem...
TMPY-00072 GITR/TNFRSF18 Protein, Human, Recombinant (His) Human HEK293
GITR, also known as TNFRSF18(CD357), belongs to the tumor necrosis factor receptor (TNF-R) superfamily. It is the receptor for TNFSF18. GITR plays a key role in dominant immunological self-tolerance maintained by CD25(+)...
TMPJ-01099 IL-15RA Protein, Human, Recombinant (hFc)（Human Cells） Human Human Cells
Interleukin 15 Receptor alpha (IL-15Rα) is a transmembrane glycoprotein that plays a pleiotropic role in immune development and function, including the positive maintenance of lymphocyte homeostasis. IL-15Rα chain can bi...
TMPY-04298 CDCP1 Protein, Human, Recombinant (His) Human HEK293
CDCP1 contains three extracellular CUB domains. It is a putative stem cell marker that is highly expressed in some human cancer cells and both, typical and atypical (cancerous) colons. It interacts with CDH2/N-cadherin, ...
TMPY-00480 NCAM1 Protein, Human, Recombinant (His) Human HEK293
NCAM1 (Neural Cell Adhesion Molecule 1, also known as CD56) is a Protein Coding gene. 3 alternatively spliced human isoforms have been reported. NCAM1 is a neural adhesion protein (NCAM) that belongs to the immunoglobuli...
TMPY-01180 CD86 Protein, Human, Recombinant (His) Human HEK293
CD86, also known as B-lymphocyte activation antigen B7-2 (referred to as B70), is a member of the cell surface immunoglobulin superfamily. B7-2 exists predominantly as a monomer on cell surfaces and interacts with two co...
TMPJ-01331 Frizzled-8 Protein, Human, Recombinant (His & Avi), Biotinylated Human Human Cells
Frizzled-8 is one of at least ten seven-transmembrane (7TM) glycoproteins of the Frizzled family of Wnt receptors. Frizzled proteins are thought to be G-protein-coupled. Wnt engagement, with low density lipoprotein recep...
TMPJ-01332 Frizzled-8 Protein, Human, Recombinant (His) Human Human Cells
Frizzled-8 is one of at least ten seven-transmembrane (7TM) glycoproteins of the Frizzled family of Wnt receptors. Frizzled proteins are thought to be G-protein-coupled. Wnt engagement, with low density lipoprotein recep...
TMPY-01165 FZD1/Frizzled 1 Protein, Mouse, Recombinant (His) Mouse HEK293
Frizzled-1, also known as FZD1, belongs to theG-protein coupled receptor Fz/Smo family. FZD1 contains a signal peptide, a cysteine-rich domain in the N-terminal extracellular region, 7 transmembrane domains, and a C-term...
TMPK-00447 CD45 Protein, Human, Recombinant (aa 26-577, hFc) Human HEK293
PTPRC (also known as CD45),T cells require the protein tyrosine phosphatase CD45 to detect and respond to antigen because it activates the Src family kinase Lck, which phosphorylates the T cell antigen receptor (TCR) com...
TMPY-03883 CD47 Protein, Human, Recombinant (hFc) Human HEK293
CD47 contains 1 Ig-like V-type (immunoglobulin-like) domain and is a receptor for the C-terminal cell binding domain of thrombospondin. It may play a role in membrane transport and signal transduction. CD47 is also a mem...
TMPY-04273 FGFR2 Protein, Human, Recombinant (aa 1-378, His) Human HEK293
FGFR2, also known as CD332, belongs to the fibroblast growth factor receptor subfamily where amino acid sequence is highly conserved between members and throughout evolution. FGFR2 acts as cell-surface receptor for fibro...
TMPY-03969 SUSD4 Protein, Human, Recombinant (mFc) Human HEK293
SUSD4, also known as sushi domain-containing protein 4, is a hypothetical cell surface protein whose tissue distribution and function are completely unknown. SUSD4 is detectable in murine brains, eyes, spinal cords, and ...
TMPK-00399 FGFR2 beta (IIIb) Domain Protein, Human, Recombinant (Avi), Biotinylated Human HEK293
Four distinct genes encoding closely related FGF receptors, FGF R1 - 4, are known. All four genes for FGF Rs encode proteins with an N-terminal signal peptide, three immunoglobulin (Ig)-like domains, an acid-box region c...
TMPJ-00899 HER3/ERBB3 Protein, Human, Recombinant (aa 20-331, hFc) Human Human Cells
Receptor tyrosine-protein kinase erbB-3 is an enzyme that in humans is encoded by the ERBB3 gene. This gene encodes a member of the epidermal growth factor receptor (EGFR) family of receptor tyrosine kinases. ERBB3 belon...
TMPY-01268 SMYD3 Protein, Human, Recombinant (GST) Human Baculovirus-Insect Cells
SET and MYND domain-containing protein 3, also known as Zinc finger MYND domain-containing protein 1, SMYD3, and ZMYND, is a member of the histone-lysine methyltransferase family. SMYD3 contains one MYND-type zinc finger...
TMPY-05590 NCAM1 Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293
NCAM1 (Neural Cell Adhesion Molecule 1, also known as CD56) is a Protein Coding gene. 3 alternatively spliced human isoforms have been reported. NCAM1 is a neural adhesion protein (NCAM) that belongs to the immunoglobuli...
TMPY-04157 RANK/TNFRSF11A Protein, Human, Recombinant (His) Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small i...
TMPY-01656 VEGF183 Protein, Human, Recombinant Human Baculovirus-Insect Cells
Vascular endothelial growth factor (VEGF), also known as vascular permeability factor (VPF) and VEGF-A, is a potent mediator of both angiogenesis and vasculogenesis in the fetus and adult. It is a member of the platelet-...
TMPJ-00390 FGFR2IIIb Protein, Human, Recombinant (hFc) Human Human Cells
FGFR2, also known as CD332, belongs to the fibroblast growth factor receptor subfamily where amino acid sequence is highly conserved between members and throughout evolution. FGFR2 acts as cell-surface receptor for fibro...
TMPY-05383 NKp30/NCR3 Protein, Human, Recombinant (hFc) Human HEK293
Natural Cytotoxicity Triggering Receptor 3, NCR3, also known as NKp30, or CD337, is a natural cytotoxicity receptor, expressed on subsets of human peripheral blood NK cells, involved in NK cell killing of tumor cells and...
TMPY-06411 GITR/TNFRSF18 Protein, Human, Recombinant (His & Avi), Biotinylated Human HEK293
GITR, also known as TNFRSF18(CD357), belongs to the tumor necrosis factor receptor (TNF-R) superfamily. It is the receptor for TNFSF18. GITR plays a key role in dominant immunological self-tolerance maintained by CD25(+)...
TMPY-03960 COL9A1 Protein, Human, Recombinant (His) Human HEK293
TMPY-05246 CD86 Protein, Human, Recombinant (His), Biotinylated Human HEK293
CD86, also known as B-lymphocyte activation antigen B7-2 (referred to as B70), is a member of the cell surface immunoglobulin superfamily. B7-2 exists predominantly as a monomer on cell surfaces and interacts with two co...
TMPY-03621 EphB2 Protein, Mouse, Recombinant (hFc) Mouse HEK293
Ephrin type-B receptor 2, also known as EphB2, belongs to the ephrin receptor subfamily of the protein-tyrosine kinase family which 16 known receptors (14 found in mammals) are involved: EPHA1, EPHA2, EPHA3, EPHA4, EPHA5...
TMPY-02691 IL-17RC Protein, Human, Recombinant(aa 1-454, hFc) Human HEK293
IL17RC (Interleukin 17 Receptor C) is a Protein Coding gene. This gene encodes a single-pass type I membrane protein that shares similarity with the interleukin-17 receptor (IL-17RA). IL17RC is widely expressed in the pr...
TMPJ-00391 FGFR2IIIb Protein, Human, Recombinant (aa 22-378, hFc) Human Human Cells
FGFR2, also known as CD332, belongs to the fibroblast growth factor receptor subfamily where amino acid sequence is highly conserved between members and throughout evolution. FGFR2 acts as cell-surface receptor for fibro...
TMPJ-00054 PLGF-2 Protein, Human, Recombinant (His) Human Human Cells
Placental growth factor is a protein that in humans is encoded by the PGF gene. It is a secreted protein and belongs to the PDGF/VEGF growth factor family. Alternate splicing results in at least three human mature PlGF f...
TMPY-00276 PLGF/PGF Protein, Human, Recombinant (mFc) Human HEK293
TMPY-03435 NCKIPSD Protein, Human, Recombinant (GST) Human E. coli
NCKIPSD is localized exclusively in the cell nucleus. It plays a role in signal transduction and may function in the maintenance of sarcomeres and the assembly of myofibrils into sarcomeres. NCKIPSD also plays an importa...
TMPK-00398 FGFR2 beta (IIIb) Domain Protein, Human, Recombinant (Avi) Human HEK293
Four distinct genes encoding closely related FGF receptors, FGF R1 - 4, are known. All four genes for FGF Rs encode proteins with an N-terminal signal peptide, three immunoglobulin (Ig)-like domains, an acid-box region c...
TMPY-05514 RANK/TNFRSF11A Protein, Human, Recombinant (mFc) Human HEK293
TNFRSF11A is a member of the TNF-receptor superfamily. In mouse, it is also known as CD265. TNFRSF11A contains 4 TNFR-Cys repeats and is widely expressed with high levels in skeletal muscle, thymus, liver, colon, small i...
TMPJ-01288 KLF6 Protein, Human, Recombinant Human E. coli
Krueppel-Like Factor 6 (KLF6) belongs to the krueppel C2H2-type zinc-finger protein family. KLF6 contains three C2H2-type zinc fingers and localizes in the nucleus. KLF6 expression is highest in the placenta followed by ...
TMPY-04386 EphB2 Protein, Human, Recombinant (aa 570-987, His & GST) Human Baculovirus-Insect Cells
Ephrin type-B receptor 2, also known as EphB2, belongs to the ephrin receptor subfamily of the protein-tyrosine kinase family which 16 known receptors (14 found in mammals) are involved: EPHA1, EPHA2, EPHA3, EPHA4, EPHA5...
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GSK3B Protein, Mouse, Recombinant (His)
TMPY-04439
Species: Mouse
Expression System: Baculovirus-Insect Cells
Frizzled 10 Protein, Human, Recombinant (His)
TMPY-04147
Species: Human
Expression System: HEK293
Frizzled 10 Protein, Mouse, Recombinant (hFc)
TMPY-01797
Species: Mouse
Expression System: HEK293
Frizzled 10 Protein, Mouse, Recombinant (His)
TMPY-01798
Species: Mouse
Expression System: HEK293
Frizzled 10 Protein, Human, Recombinant (hFc)
TMPY-04140
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (hFc)
TMPY-04142
Species: Human
Expression System: HEK293
Mesothelin Protein, Human, Recombinant
TMPY-00132
Species: Human
Expression System: HEK293
HNT/NTM Protein, Human, Recombinant (His)
TMPY-00357
Species: Human
Expression System: HEK293
FGF-8b Protein, Human, Recombinant
TMPY-06986
Species: Human
Expression System: E. coli
CD45 Protein, Human, Recombinant (aa 26-577, His)
TMPY-05748
Species: Human
Expression System: HEK293
CD47 Protein, Human, Recombinant
TMPY-04683
Species: Human
Expression System: HEK293
Periostin/OSF-2 Protein, Human, Recombinant (His)
TMPY-01020
Species: Human
Expression System: HEK293
PRSS3 Protein, Human, Recombinant (His)
TMPY-01897
Species: Human
Expression System: HEK293
CD47 Protein, Human, Recombinant, Biotinylated
TMPY-05191
Species: Human
Expression System: HEK293
Neuropilin-2 Protein, Human, Recombinant (hFc)
TMPY-03763
Species: Human
Expression System: HEK293
Neuropilin-2 Protein, Human, Recombinant (His)
TMPY-00892
Species: Human
Expression System: HEK293
CD47 Protein, Human, Recombinant (aa 1-139, His)
TMPY-04935
Species: Human
Expression System: HEK293
GITR/TNFRSF18 Protein, Human, Recombinant (His)
TMPY-00072
Species: Human
Expression System: HEK293
IL-15RA Protein, Human, Recombinant (hFc)（Human Cells）
TMPJ-01099
Species: Human
Expression System: Human Cells
CDCP1 Protein, Human, Recombinant (His)
TMPY-04298
Species: Human
Expression System: HEK293
NCAM1 Protein, Human, Recombinant (His)
TMPY-00480
Species: Human
Expression System: HEK293
CD86 Protein, Human, Recombinant (His)
TMPY-01180
Species: Human
Expression System: HEK293
Frizzled-8 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPJ-01331
Species: Human
Expression System: Human Cells
Frizzled-8 Protein, Human, Recombinant (His)
TMPJ-01332
Species: Human
Expression System: Human Cells
FZD1/Frizzled 1 Protein, Mouse, Recombinant (His)
TMPY-01165
Species: Mouse
Expression System: HEK293
CD45 Protein, Human, Recombinant (aa 26-577, hFc)
TMPK-00447
Species: Human
Expression System: HEK293
CD47 Protein, Human, Recombinant (hFc)
TMPY-03883
Species: Human
Expression System: HEK293
FGFR2 Protein, Human, Recombinant (aa 1-378, His)
TMPY-04273
Species: Human
Expression System: HEK293
SUSD4 Protein, Human, Recombinant (mFc)
TMPY-03969
Species: Human
Expression System: HEK293
FGFR2 beta (IIIb) Domain Protein, Human, Recombinant (Avi), Biotinylated
TMPK-00399
Species: Human
Expression System: HEK293
HER3/ERBB3 Protein, Human, Recombinant (aa 20-331, hFc)
TMPJ-00899
Species: Human
Expression System: Human Cells
SMYD3 Protein, Human, Recombinant (GST)
TMPY-01268
Species: Human
Expression System: Baculovirus-Insect Cells
NCAM1 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPY-05590
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (His)
TMPY-04157
Species: Human
Expression System: HEK293
VEGF183 Protein, Human, Recombinant
TMPY-01656
Species: Human
Expression System: Baculovirus-Insect Cells
FGFR2IIIb Protein, Human, Recombinant (hFc)
TMPJ-00390
Species: Human
Expression System: Human Cells
NKp30/NCR3 Protein, Human, Recombinant (hFc)
TMPY-05383
Species: Human
Expression System: HEK293
GITR/TNFRSF18 Protein, Human, Recombinant (His & Avi), Biotinylated
TMPY-06411
Species: Human
Expression System: HEK293
COL9A1 Protein, Human, Recombinant (His)
TMPY-03960
Species: Human
Expression System: HEK293
CD86 Protein, Human, Recombinant (His), Biotinylated
TMPY-05246
Species: Human
Expression System: HEK293
EphB2 Protein, Mouse, Recombinant (hFc)
TMPY-03621
Species: Mouse
Expression System: HEK293
IL-17RC Protein, Human, Recombinant(aa 1-454, hFc)
TMPY-02691
Species: Human
Expression System: HEK293
FGFR2IIIb Protein, Human, Recombinant (aa 22-378, hFc)
TMPJ-00391
Species: Human
Expression System: Human Cells
PLGF-2 Protein, Human, Recombinant (His)
TMPJ-00054
Species: Human
Expression System: Human Cells
PLGF/PGF Protein, Human, Recombinant (mFc)
TMPY-00276
Species: Human
Expression System: HEK293
NCKIPSD Protein, Human, Recombinant (GST)
TMPY-03435
Species: Human
Expression System: E. coli
FGFR2 beta (IIIb) Domain Protein, Human, Recombinant (Avi)
TMPK-00398
Species: Human
Expression System: HEK293
RANK/TNFRSF11A Protein, Human, Recombinant (mFc)
TMPY-05514
Species: Human
Expression System: HEK293
KLF6 Protein, Human, Recombinant
TMPJ-01288
Species: Human
Expression System: E. coli
EphB2 Protein, Human, Recombinant (aa 570-987, His & GST)
TMPY-04386
Species: Human
Expression System: Baculovirus-Insect Cells
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Cat No. Product Name
L1610 FDA-Approved Kinase Inhibitor Library

266 compounds
A unique collection of 266 kinase inhibitors/regulators for specific targeting of kinases, ready for high-throughput screening and high-content screening.
L1600 Kinase Inhibitor Library

2720 compounds
A unique collection of 2720 kinase inhibitors/regulators for high throughput screening and high content screening for drug discovery in kinase related diseases;

Libraries

FDA-Approved Kinase Inhibitor Library
L1610
Compounds: 266
Kinase Inhibitor Library
L1600
Compounds: 2720
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