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diclofenac

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Diclofenac
T019615307-86-5
Diclofenac (Diclofenacum) is a nonsteroidal benzeneacetic acid derivative with anti-inflammatory activity. Diclofenac binds and chelates both isoforms of cyclooxygenase (COX-1 and-2), thereby blocking the conversion of arachidonic acid to pro-inflammatory-proprostaglandins.
  • $42
In Stock
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QTY
Diclofenac Acyl Glucuronide
T2716764118-81-6
Diclofenac Acyl Glucuronide (Diclofenac glucuronide) is an intestinal metabolite that accelerates intestinal ulcers.
  • $1,099
35 days
Size
QTY
Diclofenac Potassium
T647015307-81-0
Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.
  • $33
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Diclofenac Amide
T064315362-40-0
Diclofenac Amide is used as a intermediates of Diclofenac.
  • $55
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Diclofenac sodium
T155515307-79-6
Diclofenac sodium (GP 45840) is a non-steroidal anti-inflammatory agent (NSAID) with antipyretic and analgesic actions. It is primarily available as the sodium salt.
  • $45
In Stock
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Diclofenac diethylamine
T043278213-16-8
Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).
  • $56
In Stock
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4’-Hydroxy Diclofenac-d4 (Major)
TMID-02201382084-40-3
4’-Hydroxy Diclofenac-d4 (Major) is a deuterated compound of 4’-Hydroxy Diclofenac. 4’-Hydroxy Diclofenac has a CAS number of 64118-84-9. 4'-Hydroxydiclofenac is a diclofenac metabolite.
  • Inquiry Price
35 days
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4'-Hydroxy diclofenac
T1981964118-84-9
4'-Hydroxydiclofenac is a diclofenac metabolite.
  • $466
35 days
Size
QTY
4’-Hydroxy Diclofenac-d4
TMIJ-0128254762-27-1
4’-Hydroxy Diclofenac-d4 is a deuterated compound of 4’-Hydroxy Diclofenac. 4’-Hydroxy Diclofenac has a CAS number of 64118-84-9. 4'-Hydroxydiclofenac is a diclofenac metabolite.
  • Inquiry Price
20 days
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QTY
Diclofenac methyl ester
T3748215307-78-5
Diclofenac methyl ester is a hydrophobic prodrug form of the non-steroidal anti-inflammatory drug (NSAID) diclofenac . It is more soluble than diclofenac acid in isopropylmyristate. Diclofenac methyl ester does not permeate human epidermal membranes in vitro.
  • $35
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Diclofenac deanol
T6864081811-14-5
Diclofenac deanol is a nonsteroidal anti-inflammatory drug (NSAID) of the phenylacetic acid class with anti-inflammatory, analgesic, and antipyretic properties. Contrary to the action of many traditional NSAIDs, diclofenac inhibits cyclooxygenase (COX)-2 enzyme with greater potency than it does COX-1.
  • $1,520
1-2 weeks
Size
QTY
Diclofenac Epolamine
T22307119623-66-4
Diclofenac Epolamine (DHEP) is a non-steroidal anti-inflammatory agent (NSAID) with analgesic and antipyretic actions.
  • $30
In Stock
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5-hydroxy Diclofenac
T3791769002-84-2
5-hydroxy Diclofenac is a metabolite of the NSAID diclofenac formed by the cytochrome P450 (CYP) isoform CYP3A4. Diclofenac is a non-selective COX inhibitor. It inhibits human COX-1 and -2 with IC50 values of 0.9-2.7 and 1.5-20 μM, respectively. Diclofenac inhibits ovine COX-1 and -2 with IC50 values of 60 and 220 nM, respectively.
  • $293
35 days
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Diclofenac ethyl ester
T3748115307-77-4
Diclofenac ethyl ester can be used in related research in the field of life sciences. Its product number is T37481 and CAS number is 15307-77-4.
  • $198
35 days
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QTY
Diclofenac-d4
TMIJ-0127153466-65-0
Diclofenac-d4 is a deuterated compound of Diclofenac. Diclofenac has a CAS number of 15307-86-5. Diclofenac is a nonsteroidal benzeneacetic acid derivative with anti-inflammatory activity. Diclofenac binds and chelates both isoforms of cyclooxygenase (COX-1 and-2), thereby blocking the conversion of arachidonic acid to pro-inflammatory-proprostaglandins.
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20 days
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2,6-Dichlorodiphenylamine
T3824015307-93-4
2,6-Dichlorodiphenylamine, an analogue of Diclofenac Sodium, exhibits anti-Candida albicans activity. Diclofenac Sodium, a potent and nonselective COX inhibitor, has IC50 values of 4 and 1.3 nM for human COX-1 and COX-2 in CHO cells. [1]. Makoto Urai, et al. Potent Drugs That Attenuate anti-Candida albicans Activity of Fluconazole and Their Possible Mechanisms of Action. J Infect Chemother. 2014 Oct;20(10):612-5.
  • $34
In Stock
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BPC 157 acetate
TP25141628202-19-6
Body Protection Compound 157 (BPC 157) is a pentadecapeptide derived from BPC, identified in gastric juice, exhibiting diverse biological activities. At 2 µg/ml, BPC 157 enhances primary rat tendon fibroblast cell migration and F-actin formation. Furthermore, doses of 0.01 and 10 µg/kg, intraperitoneally (i.p.), mitigate paw swelling, bone erosion, and mononuclear cell infiltration in the joints of rats with rheumatoid arthritis induced by complete Freund's adjuvant (CFA). It also diminishes gastric ulcer size in rats caused by indomethacin, aspirin, or diclofenac at these doses. Additionally, BPC 157 reduces catalepsy duration and tremor severity in a mouse model of Parkinson's disease triggered by MPTP.
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1,3-Distearoyl Glycerol
T85080504-40-5
1,3-Distearoyl glycerol, a diacylglycerol with stearic acid at the sn-1 and sn-3 positions, is present in wheat bran extract. It is utilized in creating prodrug versions of NSAIDs (ibuprofen, naproxen, and diclofenac) with decreased ulcerogenicity.
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8-10 weeks
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AS 1892802
T22037928320-12-1
AS 1892802 is a potent and selective inhibitor of ROCK. AS 1892802 exibits IC50 values of 52nM, 57nM and 122 nM for human ROCK2, rat ROCK2 and human ROCK1, respectively. The onset of antinociceptive effect of AS 1892802 is as fast as those of Tramadol and Diclofenac.
  • $44
In Stock
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Urease-IN-10
T875971012205-70-7
Urease-IN-10 (Conjugate 4), a competitive inhibitor of urease, exhibits an IC50 of 3.59±0.07 μM and a Ki of 7.45 μM. This compound is a conjugate of Diclofenac and Sulfanilamide. The combination of Diclofenac-sulfanilamide effectively inhibits Jack bean urease (JBU) through competitive inhibition [1].
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10-14 weeks
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ATB-337
T21939912758-00-0
S-Diclofenac is a novel NSAID formed by linking diclofenac to an H2S-releasing moiety. S-Diclofenac spares the gastric mucosa of injury despite markedly suppressing prostaglandin synthesis [1].
  • $88
35 days
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