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  • Cholecystokinin Receptor
    (16)
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Results for "

cck-a

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    64
    TargetMol | Inhibitors_Agonists
  • Compound Libraries
    1
    TargetMol | Compound_Libraries
  • Peptide Products
    16
    TargetMol | Peptide_Products
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    3
    TargetMol | Natural_Products
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    2
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    1
    TargetMol | Inhibitors_Agonists
CCK-A receptor inhibitor 1
T12404137004-80-9In house
CCK-A receptor inhibitor 1 is a potent cholecystokinin A (CCK-A) receptor inhibitor (IC50: 340 nM) and can be used to study digestive system-related diseases.
  • Inquiry Price
6-8 weeks
Size
QTY
(Iso)-FK-480
CHEMBL333994
T10055167820-10-2In house
(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.
  • Inquiry Price
6-8 weeks
Size
QTY
Gastrin/CCK antagonist 1
T13260162271-52-5In house
Gastrin CCK antagonist 1 is a potent gastrin CCK antagonist for the study of metabolic system-related diseases.
  • Inquiry Price
8-10 weeks
Size
QTY
A-65186
A 65186, A65186
T26483119295-94-2In house
A-65186 is an A-type glutamatergic cholecystokinin (CCK) antagonist used to study inflammation and gastrointestinal tract injury.
  • Inquiry Price
6-8 weeks
Size
QTY
itriglumide
CR-2945, CR2945, CR 2945
T27640201605-51-8In house
Itriglumide (CR-2945) is a cholecystokinin (CCK)-2 receptor antagonist with antisecretory and antiulcerogenic properties.
  • Inquiry Price
6-8 weeks
Size
QTY
Proglumide
T10526620-60-6
Proglumide (Binoside) is a cholecystokinin antagonist, which blocks both the CCKA and CCKB subtypes. Proglumide is a drug that exerts an inhibitory effect on gastric secretion and reduces gastrointestinal motility. It is used clinically in the drug therapy of gastrointestinal ulcers.
  • Inquiry Price
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N-Cbz-DL-tryptophan
T934313058-16-7
N-Cbz-DL-tryptophan is a cholecystokinin receptor antagonist, abolished the response of the isolated heart to CCK-8.
  • Inquiry Price
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TargetMol | Inhibitor Sale
Sincalide
SQ19844, Cholecystokinin octapeptide, CCK-8
TP119725126-32-3
Sincalide (CCK-8) is a cholecystokinetic drug administered by injection to aid in diagnosing disorders of the gallbladder and pancreas. It is the 8-amino acid C-terminal fragment of cholecystokinin.
  • Inquiry Price
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QTY
TargetMol | Inhibitor Sale
WAY-620645
T9991742116-45-6
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
  • Inquiry Price
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TargetMol | Inhibitor Sale
CCK-B Receptor Antagonist 2
T10707155412-88-7
CCK-B Receptor Antagonist 2 is a potent and orally active antagonist of Gastrin CCK-B (IC50: 0.43 nM). It also inhibits gastrin CCK-A activity (IC50: 1.82 μM).
  • Inquiry Price
6-8 weeks
Size
QTY
Proglumide hemicalcium
T1254485068-56-0
Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A B receptors, has antiepileptic and antioxidant activities.
  • Inquiry Price
3-6 months
Size
QTY
Tarazepide
T13084141374-81-4
Tarazepide is a potent and specific antagonist of the CCK-A receptor.
  • Inquiry Price
8-10 weeks
Size
QTY
CCK-B Receptor Antagonist 1
T13261168161-71-5
CCK-B Receptor Antagonist 1 is a cholecystokinin B (CCK-B) receptor agonist and has the potential of reducing the secretion of gastric acid.
  • Inquiry Price
7-10 days
Size
QTY
Ceruletide Ammonium acetate
FI-6934 Ammonium acetate, Ceruletide Ammonium acetate (17650-98-5 free base), Caerulein Ammonium acetate
T14932L
Ceruletide Ammonium acetate (FI-6934 Ammonium acetate) is a cholecystokinin (CCK) receptor agonist. Ceruletide Ammonium acetate is a safe and effective cholecystokinetic agent and small bowel and exocrine pancreatic stimulant.
  • Inquiry Price
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Devazepide
L-364,718, MK-329
T15101103420-77-5
Devazepide is a competitive and orally active nonpeptide antagonist of cholecystokinin (CCK) receptor (IC50s: 81 pM, 45 pM, and 245 nM for rat pancreatic, bovine gallbladder and guinea pig brain CCK receptors, respectively).
  • Inquiry Price
7-10 days
Size
QTY
Dexloxiglumide
T15105119817-90-2
Dexloxiglumide, an active enantiomer of Loxiglumide, inhibits smooth muscle cell contractions induced by cholecystokinin-octapeptide (CCK-8). It is a selective antagonist of cholecystokinin type A (CCKA) receptors.
  • Inquiry Price
7-10 days
Size
QTY
Sograzepide
YF476, YF 476, YM220, YM-220, Netazepide
T16906155488-25-8
Sograzepide (Netazepide) is an orally active, selective and highly potent gastrin CCK-B antagonist that inhibits gastrin CCK-A activity and pappalysin 2 expression in type 1 gastric neuroendocrine tumors, and can induce regression of type 1 gastric neuroendocrine tumors.
  • Inquiry Price
6-8 weeks
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QTY
YM022
T17274145084-28-2
YM022 is a highly effective and selective gastrin cholecystokinin (CCK)-B receptor antagonist. YM022 can inhibit gastrin-induced gastric acid secretion and histidine decarboxylase activation in vivo. YM022 shows the Ki values of 68 pM and 63 nM for CCK-B and CCK-A receptor, respectively.
  • Inquiry Price
6-8 weeks
Size
QTY
Nastorazepide hemicalcium
Z-360 hemicalcium
T201854343326-69-2
Nastorazepide (Z-360) hemicalcium is a selective, orally-administered 1,5-benzodiazepine derivative that functions as a receptor antagonist for gastrin cholecystokinin 2 (CCK-2), exhibiting potential antitumor activity.
  • Inquiry Price
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Cholecystokinin (27-32)-amide
Cholecystokinin (27-32)-NH2
T2388686367-90-0
Cholecystokinin (27-32)-amide is a CCK receptor antagonist.
  • Inquiry Price
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DA-3934
UNII-J353803KRG
T23946183176-50-3
DA-3934 has a high affinity for gastrin/CCK-B receptors and high selectivity over CCK-A receptors. DA-3934 and its methyl ester derivative inhibited pentagastrin-induced gastric acid secretion in rats in a dose-dependent manner.
  • Inquiry Price
8-10 weeks
Size
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L 365031
L 365,031,L365031,L-365,031,L-365031,L365,031
T24287111035-59-7
L 365031 is a CCK antagonist.
  • Inquiry Price
6-8 weeks
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ARL 15849XX
FPL-15849, FPL15849, FPL 15849, ARL-15849XX, ARL15849XX
T25108152548-39-5
ARL 15849XX, a CCK-8 analog, is a novel anti-obesity agent.
  • Inquiry Price
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BC 197
Boc-asp-tyr(SO3H)-ahx-lys-trp-ahx-asp-phe-NH2, BC-197, BC197
T25139115295-08-4
BC 197 is a selective CCK-B agonist.
  • Inquiry Price
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