radioligand — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T79577	CB2 PET Radioligand 1		Cannabinoid Receptor
	CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.7 nM). It is synthesized via Cu-mediated 18F-fluorination an...		Cannabinoid Receptor
T21667	FAUC-365	FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide,FAUC-365 Benzo[b]thiophene-2-carboxylic acid {4-[4-(2,3-dichloro- phenyl)-piperazin-1-yl]-butyl}-amide	Dopamine Receptor
	FAUC-365 is a D3 dopamine receptor agonist.		Dopamine Receptor
T11894	Lusaperidone	R107474	Adrenergic Receptor
	Lusaperidone (R107474) is a potent α2-adrenergic receptor antagonist, a potential radioligand for the α (2)-adrenergic receptor, with inhibitory effects on α2A and α2C, with Ki values of 0.13 and 0.15 nM, respectively.		Adrenergic Receptor
T4727	Taurolithocholic acid sodium salt	Sodium taurolithocholate	Others , Calcium Channel
	Taurolithocholic acid sodium salt (Sodium taurolithocholate) is the major human metabolite, a bile acid which inhibits radioligand binding to muscarinic M1, but not to M2 or M3 receptors.		Others , Calcium Channel
T16140	MRS 1754		Adenosine Receptor
	MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a very low affinity for A1 and A3 receptors of both humans and rats.		Adenosine Receptor
T38205	3-Aminopropylphosphonic Acid		GABA Receptor
	3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding assay).		GABA Receptor
T30140	Arotinolol hydrochloride	Arotinolol HCl	5-HT Receptor , Adrenergic Receptor
	Arotinolol hydrochloride（Arotinolol HCl） is a non-selective α/β-adrenergic receptor blocker.Arotinolol hydrochloride inhibits the binding of the radioligand 125I-ICYP to the 5HT1B-hydroxytryptamine receptor. Arotinolol h...		5-HT Receptor , Adrenergic Receptor
T16115	MLi-2		LRRK2
	MLi-2 is a structurally novel, highly potent, and selective LRRK2 kinase inhibitor with central nervous system activity. MLi-2 exhibits exceptional potency in a purified LRRK2 kinase assay in vitro (IC50 = 0.76 nM), a ce...		LRRK2
T34243	R214127	R 214127,R-214127
	R214127 is a new type of mGlu1 receptor high-affinity radioligand.
T30253	AZD-2184	J2.698.897G,AZD2184
	AZD-2184 is a radioligand for detecting beta-amyloid deposits.
T34626	Setoperone	R-52245,R 52245,R52245
	Setoperone, as a sensitive radioligand, can be commonly used in position emission tomography (PET) imaging.
T29913	Altanserin	R-53200,R53200,R 53200
	Altanserin can binds to the 5-HT2A receptor. Labeled with the isotope fluorine-18 it is used as a radioligand in positron emission tomography (PET) studies of the brain.
T34483	Sadopine
	Sadopine is an excellent high affinity, high specific activity radioligand to label selectively the DHP receptor of L-type Ca2+ channels in tissue sections as well as in membrane fragments.
T26478	A-317920
	A-317920 is an inverse agonist radioligand.
T39069	UCB-J
	UCB-J is a radioligand for the synaptic vesicle protein 2A (SV2A), utilized in positron emission tomography (PET)[4].
T10371	Arotinolol		5-HT Receptor
	Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand 125I-ICYP to 5HT1B-serotonergic receptor sites. It is...		5-HT Receptor
T71186	ORM-13070
	ORM-13070 is a selective antagonist radioligand for the α2C adrenoceptor subtype. ORM-13070 C-11 is under investigation in clinical trial.
T34688	SP203	SP-203,SP 203
	SP203 is a radioligand for brain metabotropic glutamate receptor imaging.
T33277	Mefway F-18	18F-Mefway
	Mefway F-18 is a PET radioligand specific to serotonin-1A receptors.
T69100	A-349821
	A-349821 is an H3 receptor agonist radioligand.