Home Tools
Log in
Cart

Search Result

Search Results for "nlrp3-in-2"

Compounds

Cat No. Product Name
T3230 NLRP3-IN-2 4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,NLRP3 Inflammasome Inhibitor I NOD-like Receptor (NLR) , NOD
NLRP3 Inflammasome Inhibitor I 是一种能够合成格列本脲的中间物,对心肌细胞中NLRP3炎症小体的形成具有抑制作用,在小鼠心肌缺血/再灌注后限制梗死面积,且对代谢无影响。
T60404 NLRP3/AIM2-IN-2 NOD
NLRP3/AIM2-IN-2是一种新型强效抑制剂,对依赖于 NLRP3和 AIM2炎症体的热扩散具有不同物种特异性影响,IC50为0.2392 ± 0.0233 μ M。
T6S1256 Ruscogenin NF-κB , NOS , NOD-like Receptor (NLR)
Ruscogenin 是一种重要甾体皂苷元,提取自麦冬。它能够抑制 TXNIP/NLRP3炎症体激活和 MAPK 途径,改善脑缺血诱导的血脑屏障功能障碍,具有显著抗血栓、抗炎作用。
T39552 NLRP3-IN-5 NLRP3-IN-5
NLRP3-IN-5, a compound disclosed in WO2016131098, is an inhibitor of NLRP3 inflammasome. It consists of the chemical str...
T62221 NLRP3-IN-8
NLRP3-IN-8 (compound 27) 是具有口服活性的、与 NLRP3直接结合的 NLRP3炎性体抑制剂,对 IL-1β 的 IC50值为1.23 μM. NLRP3-IN-8 对肝微粒体具有良好的代谢稳定性 (t1/2= 13...
T9655 NBC 6
NLRP3-IN-NBC6 是一种有效的选择性 NLRP3炎性小体抑制剂 ,IC50为574 nM,其作用独立于 Ca2+。NLRP3-IN-NBC6 抑制 Nigericin 诱导的 THP-1 细胞炎症反应和 Imiquimod 诱导...
T38106 JC-171
JC-171 is a selective NLRP3 inflammasome inhibitor, with an IC50 of 8.45 μM for inhibiting LPS/ATP-induced interleukin-1...
T72580 Isoandrographolide
Isoandrographolide 具有诱导细胞分化和保肝活性。Isoandrographolide 可抑制 NLRP3炎症小体激活并减轻小鼠矽肺。
NLRP3-IN-2
T3230
synonym: 4-[2-(5-氯-2-甲氧基苯甲酰氨基)乙基]苯磺酰胺,5-Chloro-N-(p-sulfamoylphenethyl)-o-anisamide,NLRP3 Inflammasome Inhibitor I
Target:
NLRP3/AIM2-IN-2
T60404
synonym:
Target:
Ruscogenin
T6S1256
synonym:
Target:
NLRP3-IN-5
T39552
synonym: NLRP3-IN-5
Target:
NLRP3-IN-8
T62221
synonym:
Target:
NBC 6
T9655
synonym:
Target:
JC-171
T38106
synonym:
Target:
Isoandrographolide
T72580
synonym:
Target: