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Search Results for "bace"

Targets

Compounds

Cat No. Product Name
T3161L BACE-IN-1 acetate BACE-IN-1 acetate (350228-37-4,Free base) BACE
BACE-IN-1 acetate 已被用作 BACE1 抑制剂测定中的 β 位淀粉样前体蛋白 (APP) 裂解酶-1 (BACE1) 抑制剂。 β-位点淀粉样前体蛋白 (APP) 切割酶-1 (BACE1)是一种天冬氨酸蛋白酶,属于蛋白酶...
T62181 BACE-IN-1
BACE-IN-1 是一种咪唑[1,2-a ]吡啶衍的生物,对 β 位点淀粉样蛋白前体蛋白切割酶 (BACE) 句有抑制作用。BACE-IN-1 具有研究涉及 BACE 疾病(如阿尔茨海默氏病)的潜力。
T62995 BACE-1 inhibitor 2
BACE-1 inhibitor 2 是一种有效的,可透过血脑屏障的BACE-1抑制剂,IC50为 1.5 nM。
T10449 BACE-1 inhibitor 1 Others
BACE-1 inhibitor 1 (Compound 8a) is an effective BACE-1 inhibitor (IC50: 56 nM).
T60691 AChE/BChE/BACE-1-IN-2
AChE/BChE/BACE-1-IN-2 (Compound 4o) 表现出显著的抗氧化潜力和对PAS-AChE 的强大的结合能力。AChE/BChE/BACE-1-IN-2 是口服有效的AChE、BACE-1和BChE 抑制剂,对 hA...
T61206 AChE/BChE/BACE-1-IN-1
AChE/BChE/BACE-1-IN-1 (Compound 4k) is an orally active inhibitor that targets acetylcholinesterase (AChE), butyrylcholi...
TN7076 Herbacetin-3,8-diglucopyranoside Linocinamarin,草质素-3,8-二葡萄糖苷 Others
herbacetin-3,8-diglucopyranoside 是一种天然产物。
T5S1331 Herbacetin c-Met/HGFR , Akt
Herbacetin 是一种亚麻籽中的天然类黄酮,具有多种药理活性,如抗氧化、抗炎、抗癌作用。 它是鸟氨酸脱羧酶Ornithine decarboxylase (ODC)变构抑制剂,能够直接与 ODC 上的 Asp44,Asp243 和 G...
T10450 BACE1-IN-1 BACE
BACE1-IN-1 is a high brain penetrant BACE1 inhibitor (IC50s: 32 and 47 nM for human BACE1 and BACE2).
T10451 BACE1-IN-2 BACE
BACE1-IN-2 is a BACE1 inhibitor (IC50: 22 nM).
T10453 BACE1-IN-5 Beta Amyloid , BACE
BACE1-IN-5 (Compound 15) 是一种 BACE1抑制剂,IC50为 9.1 nM。BACE1-IN-5还可抑制细胞 Aβ,IC50为 0.82 nM。并且,BACE1-IN-5 具有改善 hERG 抑制和 P-gp 外排...
T10452 BACE1-IN-4 BACE
BACE1-IN-4 is a potent and highly selective BACE1 inhibitor (IC50: 3.8 nM; Ki: 1.9 nM), more selective at BACE1 over BAC...
T39484 BACE1-IN-6 BACE1-IN-6
BACE1-IN-6 is a BACE1 inhibitor with an IC 50 value of 1.5 nM.
T13253 Umibecestat BACE
Umibecestat 是一种β-位点淀粉样前体蛋白裂解酶-1 (BACE-1) 抑制剂,对人 BACE-1 和小鼠 BACE-1 的 IC50 分别为 11 nM 和 10 nM,可用于阿尔茨海默病的研究。
T11175 Elenbecestat E2609 Beta-Secretase , BACE
Elenbecestat 是一种高效、有口服活性的,能透过 CNS 的 BACE-1抑制剂,它有用于阿尔茨海默病 (AD) 的研究潜力。
T2S1181 Aloenin Aloearbonaside,Aloenin A,芦荟宁 AChR , Beta-Secretase
Aloenin A 是一种具有清除过氧自由基作用的天然产物,对 β-分泌酶 (BACE) 具有中等抑制活性。
T6058 LY2886721 Beta-Secretase , BACE
LY2886721 是选择性的,口服活性的 β 位淀粉样蛋白前体蛋白裂解酶 1 抑制剂,对重组人 BACE1的 IC50=20.3 nM。它对 BACE1的选择性高于对组织蛋白酶 D、胃蛋白酶、肾素的选择性,但缺乏对 BACE2的选择性。它...
TMPY-03065 BACE2 Protein, Mouse, Recombinant (His Tag)
BACE2, also known as beta secretase 2, belongs to the peptidase A1 family. It is a protease known to be an important enz...
TMPY-00752 BACE1 Protein, Human, Recombinant (His Tag), HPLC-verified
Beta-site APP-cleaving enzyme 1 (BACE1) is an aspartic-acid protease important in the formation of myelin sheaths in per...
T62719 AChE/BACE1/GSK3β-IN-1
AChE/BACE1/GSK3β-IN-1 是一种口服具有活力的、可透过血脑屏障的、生物利用度适中的 AChE/BACE1/GSK3β的三重抑制剂。AChE/BACE1/GSK3β- IN -1 能够抑制 AChE (IC50: 1.0 μ...
BACE-IN-1 acetate
T3161L
synonym: BACE-IN-1 acetate (350228-37-4,Free base)
Target:
BACE-IN-1
T62181
synonym:
Target:
BACE-1 inhibitor 2
T62995
synonym:
Target:
BACE-1 inhibitor 1
T10449
synonym:
Target:
AChE/BChE/BACE-1-IN-2
T60691
synonym:
Target:
AChE/BChE/BACE-1-IN-1
T61206
synonym:
Target:
herbacetin-3,8-diglucopyranoside
TN7076
synonym: Linocinamarin,草质素-3,8-二葡萄糖苷
Target:
Herbacetin
T5S1331
synonym:
Target:
BACE1-IN-1
T10450
synonym:
Target:
BACE1-IN-2
T10451
synonym:
Target:
BACE1-IN-5
T10453
synonym:
Target:
BACE1-IN-4
T10452
synonym:
Target:
BACE1-IN-6
T39484
synonym: BACE1-IN-6
Target:
Umibecestat
T13253
synonym:
Target:
Elenbecestat
T11175
synonym: E2609
Target:
Aloenin
T2S1181
synonym: Aloearbonaside,Aloenin A,芦荟宁
Target:
LY2886721
T6058
synonym:
Target:
BACE2 Protein, Mouse, Recombinant (His Tag)
TMPY-03065
synonym:
Target:
BACE1 Protein, Human, Recombinant (His Tag), HPLC-verified
TMPY-00752
synonym:
Target:
AChE/BACE1/GSK3β-IN-1
T62719
synonym:
Target:
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