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Protease-activated Receptor

Protease-activated receptors (PAR) are a subfamily of related G protein-coupled receptors that are activated by cleavage of part of their extracellular domain. They are highly expressed in platelets, and also on endothelial cells, myocytes and neurons.
Cat. No. Product name CAS No. Purity Chemical Structure
T7573 TFLLR-NH2 197794-83-5 98%
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7623L PAR-4 Agonist Peptide, amide acetate T7623L 98%
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
T7380 Protease-Activated Receptor-4 245443-52-1 98%
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
TP1046 SLIGRL-NH2 171436-38-7 98%
PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
T7496 Thrombin Receptor Activator for Peptide 5 (TRAP-5) 141685-53-2 98%
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
T4186 AC-264613 1051487-82-1 98%
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
T1986L Atopaxar Hydrobromide 474550-69-1 98%
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
T27267 ENMD-1068 HCl 789488-77-3 98%
ENMD-1068 is a PAR-2 antagonist. ENMD-1068 inhibits the development of endometriosis in a mouse model.
T22933L LRGILS-NH2 acetate 98%
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
T7623 PAR-4 Agonist Peptide, amide 352017-71-1 98%
PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4).
T7674 Thrombin Receptor Activator for Peptide T7674 98%
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
TP1065 PAR-4 Agonist Peptide, amide TFA 1228078-65-6 98%
PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked...
T7513 Protease-Activated Receptor-2, amide 190383-13-2 98%
Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
T7625 TRAP-6 141136-83-6 98%
TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
TP1925L TcY-NH2 TFA(327177-34-4 free base) TP1925L 98%
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
TP1378 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) TP1378 98%
2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist.
T7573L TFLLR-NH2 2TFA(197794-83-5(free base)) T7573L 98%
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
T7137 I-191 1690172-25-8 98%
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
T38836L Protease-Activated Receptor-1, PAR-1 Agonist acetate 98%
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
TQ0012 AZ3451 2100284-59-9 98%
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
TFLLR-NH2
T7573
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
PAR-4 Agonist Peptide, amide acetate
T7623L
PAR-4 Agonist Peptide, amide acetate is an agonist of proteinase-activated receptor-4 (PAR-4).
Protease-Activated Receptor-4
T7380
Protease-Activated Receptor-4 is the proteinase-activated receptor-4 (PAR4) agonist, with Antiplatelet Therapy
SLIGRL-NH2
TP1046
PAR-2 Activating Peptide is an agonist of Protease-Activated Receptor-2 (PAR-2)
Thrombin Receptor Activator for Peptide 5 (TRAP-5)
T7496
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
AC-264613
T4186
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5 and decreases interleukin-12p40 pro...
Atopaxar Hydrobromide
T1986L
Atopaxar, a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling. Atopaxar has been investigated for the treatment of Coronary Arter...
ENMD-1068 HCl
T27267
ENMD-1068 is a PAR-2 antagonist. ENMD-1068 inhibits the development of endometriosis in a mouse model.
LRGILS-NH2 acetate
T22933L
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.
PAR-4 Agonist Peptide, amide
T7623
PAR-4 Agonist Peptide, amide is an agonist of proteinase-activated receptor-4 (PAR-4).
Thrombin Receptor Activator for Peptide
T7674
Thrombin Receptor Activator for Peptide is also called Coagulation Factor II Receptor (1-5) or Proteinase Activated Receptor 1 (1-5), used in the research of cor...
PAR-4 Agonist Peptide, amide TFA
TP1065
PAR-4 Agonist Peptide, amide TFA is a proteinase-activated receptor-4 (PAR-4) agonist, which has no effect on either PAR-1 or PAR-2 and whose effects are blocked...
Protease-Activated Receptor-2, amide
T7513
Protease-Activated Receptor-2, amide is an agonist of PAR2 (IC50 : 10.4 M)
TRAP-6
T7625
TRAP-6(2TFA) is an agonist of protease-activated receptor 1 (PAR1).
tcY-NH2 TFA(327177-34-4 free base)
TP1925L
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
TP1378
2-Furoyl-LIGRLO-amide is a potent and selective protease-activated receptor 2 (PAR2) agonist.
TFLLR-NH2 2TFA(197794-83-5(free base))
T7573L
TFLLR-NH2(2TFA) is an agonist of PAR1 (EC50 :1.9 μM).
I-191
T7137
I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.
Protease-Activated Receptor-1, PAR-1 Agonist acetate
T38836L
Protease-Activated Receptor-1, PAR-1 Agonist acetate is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 ...
AZ3451
TQ0012
AZ3451 is an allosteric antagonist of protease-activated receptor-2 (PAR2, IC50: 23 nM).
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