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ENMD-1068 HCl

Name: ENMD-1068 HCl
Brand: TargetMol
SKU: T27267
Price: 50 USD
Availability: InStock
Rating: 5 (10 reviews)

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Catalog No. T27267Cas No. 789488-77-3

Alias ENMD-1068 hydrochloride, ENMD-1068 HCl, ENMD-1068, ENMD1068, ENMD 1068

ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis in a mouse model.

ENMD-1068 HCl

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Purity: 99.91%

Catalog No. T27267Alias ENMD-1068 hydrochloride, ENMD-1068 HCl, ENMD-1068, ENMD1068, ENMD 1068Cas No. 789488-77-3

ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis in a mouse model.

Pack Size	Price	USA Warehouse	Global Warehouse
10 mg	$50	-	In Stock
25 mg	$87	-	In Stock
50 mg	$137	-	In Stock
1 mL x 10 mM (in DMSO)	$50	-	In Stock

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In Stock Estimated shipping dateUSA Warehouse[1-2 days] Global Warehouse[5-7 days]

All TargetMol products are for research purposes only and cannot be used for human consumption. We do not provide products or services to individuals. Please comply with the intended use and do not use TargetMol products for any other purpose.

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Batch Information

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Purity:99.91%

Appearance:Viscous

Color:Yellow

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COA HNMR LCMS

Product Introduction

ENMD-1068 HCl AI Summary

ENMD-1068 HCl exhibits antagonist activity at protease-activated receptor 2 (PAR2) with an IC50 value of 5000 μM..

Note: Summary generated by AI. Data source: ChEMBL

Bioactivity

Description	ENMD-1068 HCl (ENMD 1068) is a PAR-2 antagonist. ENMD-1068 HCl inhibits the development of endometriosis in a mouse model.
Synonyms	ENMD-1068 hydrochloride, ENMD-1068 HCl, ENMD-1068, ENMD1068, ENMD 1068

Chemical Properties

Molecular Weight	283.41
Formula	C₁₅H₂₉N₃O₂
Cas No.	789488-77-3
Smiles	C(CC(C)C)(=O)N1CCN(C(CCCCCN)=O)CC1
Relative Density.	1.047 g/cm3 (Predicted)

Storage & Solubility Information

Storage

Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice/Shipping at ambient temperature.

Solubility Information

DMSO: 245 mg/mL (864.47 mM), Sonication is recommended.

Solution Preparation Table

DMSO

	1mg	5mg	10mg	50mg
1 mM	3.5285 mL	17.6423 mL	35.2846 mL	176.4229 mL
5 mM	0.7057 mL	3.5285 mL	7.0569 mL	35.2846 mL
10 mM	0.3528 mL	1.7642 mL	3.5285 mL	17.6423 mL
20 mM	0.1764 mL	0.8821 mL	1.7642 mL	8.8211 mL
50 mM	0.0706 mL	0.3528 mL	0.7057 mL	3.5285 mL
100 mM	0.0353 mL	0.1764 mL	0.3528 mL	1.7642 mL

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In Vivo Formulation Calculator (Clear solution)

Please enter your animal experiment information in the following box and click Calculate to obtain the stock solution preparation method and in vivo formula preparation method:

For example, if the intended dosage is 10 mg/kg for animals weighing 20 g , with a dosing volume of 100 μL per animal, TargetMol | Animal experiments

and a total of 10 animals are to be administered, using a formulation of TargetMol | reagent

10% DMSO+ 40% PEG300+ 5% Tween 80+ 45% Saline/PBS/ddH₂O , the resulting working solution concentration would be 2 mg/mL.

Stock Solution Preparation:

Dissolve 2 mg of the compound in 100 μL DMSO TargetMol | reagent to obtain a stock solution at a concentration of 20 mg/mL . If the required concentration exceeds the compound's known solubility, please contact us for technical support before proceeding.

Preparation of the In Vivo Formulation:

1) Add 100 μL of the DMSO TargetMol | reagent stock solution to 400 μL PEG300 and mix thoroughly until the solution becomes clear.

2) Add 50 μL Tween 80 and mix well until fully clarified.

3) Add 450 μL Saline,PBS or ddH₂O TargetMol | reagent and mix thoroughly until a homogeneous solution is obtained.

This example is provided solely to demonstrate the use of the In Vivo Formulation Calculator and does not constitute a recommended formulation for any specific compound. Please select an appropriate dissolution and formulation strategy based on your experimental model and route of administration.

All co-solvents required for this protocol, includingDMSO, PEG300/PEG400, Tween 80, SBE-β-CD, and Corn oil, are available for purchase on the TargetMol website.

Dose Conversion

You can also refer to dose conversion for different animals. More Dose Conversion

Tech Support

Please see Inhibitor Handling Instructions for more frequently ask questions. Topics include: how to prepare stock solutions, how to store products, and cautions on cell-based assays & animal experiments, etc