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Results for "

androgenic

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    33
    TargetMol | Inhibitors_Agonists
  • Natural Products
    5
    TargetMol | Natural_Products
  • Isotope Products
    7
    TargetMol | Isotope_Products
Finasteride
MK-906
T048898319-26-7
Finasteride (MK-906) is an oral inhibitor of active testosterone 5-alpha-reductase and Ki value is 10 nM.
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CRTh2 antagonist 2
T10889780763-95-3In house
CRTh2 antagonist 2 is a selective and potent CRTH2 antagonist, IC50≤10 nM. CRTh2 antagonist 2 can be used to study the direction of androgenic alopecia.
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6-8 weeks
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TargetMol | Inhibitor Sale
EN3356
AS N001, ASN-001
T301611429329-63-4In house
EN3356 is an orally available and selective inhibitor of steroidal 17-alpha-hydroxylase C17,20 cleavage enzyme (CYP17A1 or CYP17), a non-steroidal cleavage enzyme-selective compound with potential anti-androgenic and anti-tumor activity.
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TargetMol | Inhibitor Sale
4-Diethylaminobenzaldehyde
T10140120-21-8
4-Diethylaminobenzaldehyde, a reversible aldehyde dehydrogenase (ALDH) inhibitor (Ki: 4 nM for ALDH1), exhibits a potent anti-androgenic effect (IC50: 1.71 μM).
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Megestrol acetate
SC10363, BDH1298
T1284595-33-5
Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the progestogens in general. Megestrol acetate also has anti-androgenic properties. It is given by mouth in the palliative treatment or as an adjunct to other therapy in endometrial carcinoma and in breast cancer. Megestrol acetate has been approved to treat anorexia and cachexia.
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Norethindrone
Norethisterone
T151468-22-4
Norethindrone (Norethisterone) is a synthetic progestational hormone with actions similar to those of PROGESTERONE but functioning as a more potent inhibitor of ovulation. It has weak estrogenic and androgenic properties. The hormone has been used in treating amenorrhea, functional uterine bleeding, endometriosis, and for contraception.
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Adrenosterone
11-ketoandrostenedione, 11-oxoandrostenedione, Reichstein's substance G
T2207382-45-6
Adrenosterone (11-ketoandrostenedione) is a steroid hormone isolated from the adrenal cortex.
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2-Isopropyl Thioxanthone
T79575495-84-1
2-Isopropyl Thioxanthone has potential anti-estrogenic and anti-androgenic properties.
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TargetMol | Inhibitor Sale
Germacrone
T29456902-91-6
Germacrone is extracted from Curcuma zedoaria and has anti-inflammatory, anti-androgenic and antiviral activities. It also inhibits the proliferation of glioma cells by promoting apoptosis.
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Bifluranol
BX341
T1484334633-34-6
Bifluranol (BX341) has anti-androgenic activity and has shown significant anti-prostatic activity in in vivo studies for the treatment of benign prostatic hyperplasia (BPH).
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6-8 weeks
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TargetMol | Inhibitor Sale
GLPG0492
T11410L1215085-92-9
GLPG0492 is a novel selective androgen receptor modulator. After oral dosing, it showed anabolic activity on muscle, strongly dissociated from the androgenic activity on the prostate.
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6-8 weeks
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1,3,5-Trihydroxyxanthone
T197166732-85-0
1,3,5-Trihydroxyxanthone is a highly cytotoxic natural compound. It against a range of bacteria and yeasts.Anti-androgenic.
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Nomegestrol
TX 066 free base
T1981158691-88-6
Nomegestrol (TX 066 free base) is an orally available, selective and potent full agonist of the progesterone receptor with potent anti-estrogenic, partial anti-androgenic and anti-gonadotropic activity.Nomegestrol is also a contraceptive progestin and is used in the study of endometriosis and meningiomas.
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Tigestol
1WAE0P123G
T202579896-71-9
Tigestol, as a derivative of Estrone, exhibits properties that promote muscle growth and possess androgenic and progestogenic effects.
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GTx-027
T204549928122-40-1
GTx-027 is a non-steroidal selective androgen receptor modulator (SARM) known for its androgen receptor (AR) transcription activation, with an EC50 of 2.8765 nM. It selectively promotes muscle mass (anabolic) without affecting secondary sexual organs (androgenic).
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10-14 weeks
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Vinclozolin
Vorlan, Ronilan, Ornalin
T2070850471-44-8
Vinclozolin (Ornalin) is a fungicide with anti-androgenic activity and is commonly used in agriculture.
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Finasteride acetate
T21668222989-99-3
Finasteride (MK-906) acetate is a potent and competitive 5α-reductase inhibitor with an IC50 of 4.2 nM for type II 5α-reductase, demonstrating approximately 100-fold higher affinity for type II than type I. Finasteride acetate can be used for research on benign prostatic hyperplasia (BPH) and androgenic alopecia [1] [2] [3].
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1-2 weeks
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Demegestone
R-2453,Lutionex,R 2453,RU 2453,R2453
T2530410116-22-0
Demegestone is a progestin, or a synthetic progestogen, and hence is a progesterone receptor agonist, the biological target of progestogens like progesterone. It has no androgenic activity. Previously used to treat luteal insufficiency.
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6-8 weeks
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Piperophos
Rilof
T2596124151-93-7
Piperophos is an organophosphate with anti-androgenic activities.
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6-8 weeks
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2α-Methyl androsterone
T408096961-54-2
2α-Methyl androsterone, a metabolite of mesterolone and drostanolone, is classified as an anabolic androgenic steroid.
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Cyprodinil
T41331121552-61-2
Cyprodinil, an anilinopyrimidine broad-spectrum fungicide, inhibits methionine biosynthesis in phytopathogenic fungi, effectively limiting cell growth of B. cinerea, P. herpotrichoides, and H. oryzae on amino acid-free media with IC 50 values of 0.44, 4.8, and 0.03 μM, respectively. Additionally, in the absence of the androgen receptor (AR) agonist DHT, Cyprodinil acts as an AR agonist (EC 50 =1.91 μM) and counters DHT's androgenic effects (IC 50 =15.1 μM).
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6-8 weeks
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TP0427736 hydrochloride
T610292459963-17-6
TP0427736 hydrochloride can be used in the androgenic alopecia (AGA) research. TP0427736 hydrochloride inhibits the phosphorylation of Smad2 3 in A549 cells induced by TGF-β1 with an IC50 value of 8.68 nM. TP0427736 hydrochloride is a potent ALK5 kinase inhibitor with an IC50 value of 2.72 nM which is 300-fold more potent than inhibitory effect against ALK3 of 836 nM [1].
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6-8 weeks
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Tebuconazole-d9
T711421246818-83-6
Tebuconazole-d9 is intended for use as an internal standard for the quantification of tebuconazole by GC- or LC-MS. Tebuconazole is a triazole fungicide that is active against both seed and foliar fungi. It inhibits 14α-demethylase isolated from U. maydis and S. bicolor with IC50 values of 0.05 and 0.16 nM, respectively. It inhibits the androgenic effect of the androgen receptor agonist DHT (IC20 = 2.89 µM) and is cytotoxic (EC20 = 38.9 µM) in an MDA-kb2 assay. Tebuconazole (50 and 100 mg kg per day) administered during gestation reduces testosterone levels and increases testicular levels of progesterone and 17α-hydroxyprogesterone in male rat fetuses. It has a feminizing effect on male pups and a virializing effect on female pups. When administered to rats gestationally through postnatal day 42, tebuconazole (20 and 60 mg kg per day) leads to cell death of pyramidal cells in the CA3-4 region of the hippocampus and layer V of the cortex concomitant with impairment in learning......
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6-8 weeks
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7β-Hydroxy-epi-androsterone
T7367125848-69-5
7β-Hydroxy-epi-androsterone (7β-Hydroxy-EpiA) is an endogenous androgenic derivative of dehydroepiandrosterone that binds to ERβ and exhibits anti-inflammatory and neuroprotective properties [1] [2] [3].
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