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  • Melanin-concentrating Hormone Receptor (MCHR)
    (11)
  • GPCR
    (4)
  • 5-HT Receptor
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Results for "

melanin-concentrating hormone receptor

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    27
    TargetMol | Inhibitors_Agonists
  • Peptide Products
    7
    TargetMol | Peptide_Products
  • Recombinant Protein
    1
    TargetMol | Recombinant_Protein
TC-MCH 7c
T13101864756-35-4
TC-MCH 7c is an oral, selectable and blood-brain barrier penetrating MCH1R antagonist with IC50 performance of 5.6 nM against hMCH1R, and TC-MCH 7c is a phenylpyridone derivative with MCH1R Ki of 3.4 nM against human. In mice, MCH1R Ki was 3.0 nM.
  • Inquiry Price
6-8 weeks
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TargetMol | Inhibitor Sale
Melanin Concentrating Hormone, salmon acetate
MCH (salmon), Melanin Concentrating Hormone, salmon acetate(87218-84-6 free base)
TP1104L
Melanin Concentrating Hormone, salmon acetate (MCH (salmon)) is a 19 amino acid cyclic peptide, is largely expressed in the hypothalamus.
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ATC 0175 hydrochloride
T22591510733-97-8
ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective. ATC 0175 hydrochloride has affinity for MCH1R, MCH2R, MCH1, 5-HT2B receptors and 5-HT1A receptors with IC50s of 13.5 nM, >10,000 nM, 13 nM, 9.66 nM and 16.9 nM, respectively. ATC 0175 hydrochloride exhibits antidepressant and anxiolytic effects in animal models. aTC 0175 can be used to study depression and or anxiety disorders.
  • Inquiry Price
6-8 weeks
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QTY
TargetMol | Inhibitor Sale
SNAP 94847 hydrochloride
T80041781934-47-1
SNAP 94847 hydrochloride is a melanin-concentrating hormonereceptor1 (MCHR1) antagonist(Ki= 2.2 nM)
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Neuropeptide EI, rat acetate
Neuropeptide EI, rat acetate(125934-45-4 free base)
TP1578L
Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.
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SNAP-7941
SNAP7941
T28823387825-78-7
SNAP-7941 is a selective antagonist of the melanin concentrating hormone receptor MCH1 with promising anxiolytic, antidepressant and anorectic effects in initial animal studies.
  • Inquiry Price
10-14 weeks
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T-226296
T 226296,T226296
T28902331758-35-1
T-226296 is a antagonist of melanin concentrating hormone receptor 1 (MCHR1).
  • Inquiry Price
6-8 weeks
Size
QTY
SNAP 94847
SNAP-94847
T5406487051-12-7
SNAP 94847 (SNAP-94847) is a selective and competitive MCH1 receptor (MCH1-R) antagonist (Ki: 2.2 nM). It has anxiolytic and antidepressant activity and reduces food intake in mice.
  • Inquiry Price
1-2 weeks
Size
QTY
ATC0175
ATC 0175,ATC-0175
T26677509118-03-0
ATC0175 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
  • Inquiry Price
1-2 weeks
Size
QTY
GW-803430
GW3430, GW-3430, GW803430A, GW803430, GW 803430A
T15450515141-51-2
GW-803430 (GW-3430) is an orally active and selective melanin-concentrating hormone receptor 1 (MCH R1) antagonist used in the study of obesity.
  • Inquiry Price
8-10 weeks
Size
QTY
ALB-127158
T77491173154-32-9
ALB-127158(a) is a potent and selective melanin-concentrating hormone 1 (MCH 1) receptor antagonist that may potentially treat inflammatory bowel disease (IBD).
  • Inquiry Price
6-8 weeks
Size
QTY
AZ13483342
AZ-13483342,AZ 13483342
T26703645399-82-2
AZ13483342 is an antagonist of the melanin concentrating hormone receptor 1 (MCH1) with a potential diabetes therapeutic activity.
  • Inquiry Price
6-8 weeks
Size
QTY
NGD-4715
T16293476322-70-0
NGD-4715 is a selective, orally active antagonist of melanin-concentrating hormone receptor 1 (MCHR1).
  • Inquiry Price
6-8 weeks
Size
QTY
MCHR1 antagonist 1
T10173391610-37-0
MCHR1 antagonist 1 is a selective antagonist of the melanin-concentrating hormone-1 (MCH1) receptor with a Kb of 1 nM and a Ki of 4 nM at the human MCH1 receptor.
  • Inquiry Price
6-8 weeks
Size
QTY
ATC0065
ATC 0065,ATC-0065
T26676509145-82-8
ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.
  • Inquiry Price
6-8 weeks
Size
QTY
hMCH-1R antagonist 1
T76640353487-64-6
HMCH-1R Antagonist 1 (Compound 30) serves as an effective and selective antagonist for the human melanin-concentrating hormone receptor 1 (hMCHR1), exhibiting a K_B value of 3.6 nM. It possesses the ability to bind to hMCHR1 and hMCHR2, with IC_50 values of 65 nM and 49 nM, respectively. This compound is applicable in metabolic research [1].
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MCHR1 antagonist 3
T119651069622-60-1
MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.
  • Inquiry Price
8-10 weeks
Size
QTY
[Ala17]-MCH acetate
[Ala17]-MCH acetate(359784-84-2 free base)
TP1997L
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled). [Ala17]-MCH acetate shows selectivity over MCHR2 with Ki of 34 nM.
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ATC0065 HCl
T69170510732-84-0
ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.
  • Inquiry Price
6-8 weeks
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MCH(human, mouse, rat)
MCH (human, mouse, rat)
TP1996128315-56-0
MCH(human, mouse, rat) is a potent endogenous agonist at melanin-concentration hormone (MCH) receptors (IC50 values are 0.3 and 1.5 nM and EC50 values are 3.9 and 0.1 nM at MCH1 and MCH2 receptors respectively). Increases food intake in vivo.
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[Ala17]-MCH
TP1997359784-84-2
Potent melanin-concentrating hormone (MCH) receptor agonist (EC50 values are 17 and 54 nM at MCH1 and MCH2 receptors respectively). Displays some selectivity towards MCH1 over MCH2 (Ki values are 0.16 and 34 nM respectively).
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AZD1979
T143721254035-84-1
AZD1979 is an antagonist of Melanin-concentrating hormone receptor 1 (MCHr1) (IC50: 12 nM).
    7-10 days
    Inquiry
    SB-568849
    T16852395679-53-5
    SB-568849 is an antagonist of the melanin-concentrating hormone receptor 1 (pKi: 7.7).
    • Inquiry Price
    6-8 weeks
    Size
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    BMS-819881
    T146781197420-05-5
    BMS-819881, a melanin-concentrating hormone receptor 1 (MCHR1) antagonist, binds rat MCHR1 with a Ki of 7 nM, and is selective and potent for CYP3A4 activity with an EC50 of 13 μM.
    • Inquiry Price
    6-8 weeks
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