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cpt-1a

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  • Inhibitors & Agonists
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    TargetMol | Inhibitors_Agonists
Etomoxir sodium salt
(R)-Etomoxir sodium salt
T4535828934-41-4
Etomoxir sodium salt ((R)-Etomoxir sodium salt) is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that inhibits fatty acid oxidation (FAO). Etomoxir sodium salt has antitumor activity.
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Etomoxir
(R)-(+)-Etomoxir
T4535L124083-20-1
Etomoxir is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that inhibits fatty acid oxidation by inhibiting CPT-1a and inhibits palmitate oxidation in humans, rats, and guinea pigs. Etomoxir has an inhibitory effect on adenine nucleotide translocase and can inhibit macrophage polarization by disrupting CoA homeostasis.
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6-8 weeks
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TargetMol | Citations Cited