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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T8462 | Enoximone | PDE | |
Enoximone is a selective inhibitor of phosphodiesterase III (PDE3), with treatment of congestive heart failure. | |||
T6551 | Isosorbide | Devicoran,Isobide,Hydronol,Dianhydro-D-glucitol,D-Isosorbide | Others |
Isosorbide (Devicoran) is a heterocyclic compound that is derived from glucose, used as a diuretic. | |||
T0109 | Molsidomine | Morsydomine,SIN-10,Corvaton | NOD |
Molsidomine (Corvaton) is an orally active, long-acting vasodilating drug. It metabolizes in the liver to the active metabolite linsidomine, that releases nitric oxide (NO) upon decay as the actual vasodilating compound. | |||
T0903 | Cinnarizine | Stugeron,Cinarizine,Dimitronal,Stutgin | Calcium Channel , Histamine Receptor |
Cinnarizine (Stugeron) is a piperazine derivative having histamine H1-receptor and calcium-channel blocking activity with vasodilating and antiemetic properties but it induces PARKINSONIAN DISORDERS. | |||
TNU0864 | HUP30 | Potassium Channel , Calcium Channel | |
HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx. | |||
T0112 | Diltiazem hydrochloride | CRD-401,RG 83606 HCl,Diltiazem HCl | Calcium Channel |
Diltiazem hydrochloride (RG 83606 HCl) is a benzothiazepine calcium channel blocking agent with vasodilating action due to its antagonism of the actions of CALCIUM ion on membrane functions. | |||
T15130 | Dilazep dihydrochloride | Others | |
Dilazep dihydrochloride is an adenosine uptake inhibitor. It also inhibits ischemic damage, membrane transport of nucleosides, and platelet aggregation. It has cerebral and coronary vasodilating action through the enhanc... | |||
T2671 | Regadenoson | CVT-3146,Lexiscan | Adenosine Receptor |
Regadenoson (CVT-3146) is an adenosine derivative and selective A2A adenosine receptor agonist with coronary vasodilating activity. Upon administration, regadenoson selectively binds to and activates the A2A adenosine re... | |||
T26201 | Sorbinicate | LG10017,Sorbinicatum,LG10,017,LG-10017,LG 10017 | |
Sorbinicate is an antihypercholesterolaemic and vasodilating nicotinic acid ester. | |||
T70678 | Rwj 29009 | ||
Rwj 29009 is a potassium channel activator with prominent coronary and peripheral vasodilating actions. | |||
T30586 | Brefonalol | ||
Brefonalol is a vasodilating beta-adrenergic receptor blocker. | |||
T26081 | Ridazolol | Ridazololum | |
Ridazolol is a vasodilating and cardioselective beta adrenergic blocker. | |||
T30487 | BMS 180448 | BMS-180448,BMS180448 | |
BMS 180448 is a prototype mitochondrial ATP-sensitive K+ (Mitok (ATP)) channel opener with cardioprotective and vasodilating properties. | |||
T21047 | Apovincamine | cis-Apovincamine | |
Apovincamine is a vinca alkaloid and a chemical precursor of Vinpocetine, which is a derivative of Vincamine with vasodilating activity. | |||
T11609 | ICI 153110 | Others | |
ICI 153110 is an orally active phosphodiesterase inhibitor with both inotropic and vasodilating properties. It is designed for the treatment of congestive cardiac failure. | |||
T61495 | Medroxalol | ||
Medroxalol (RMI81968) is an orally active adrenergic receptor antagonist that effectively blocks both α- and β-adrenergic receptors, effectively producing antihypertensive and vasodilating effects [1]. | |||
T10371 | Arotinolol | 5-HT Receptor | |
Arotinolol is a nonselective α/β-adrenergic receptor blocker and a vasodilating β-blocker. Arotinolol also shows potency for inhibiting the binding of the radioligand 125I-ICYP to 5HT1B-serotonergic receptor sites. It is... | |||
T0879L | Niacin hydrochloride | ||
Niacin hydrochloride is a water-soluble vitamin of the B complex occurring in various animal and plant tissues. It is needed by the body for the formation of coenzymes NAD and NADP. It possesses PELLAGRA-curative, vasodi... | |||
T29213 | Zelandopam free base | YM-435,YM435,MYD-37,MYD37,Zelandopam | |
Zelandopam is a dopamine D1 agonist. Zelandopam is a potent stimulant of pancreatic exocrine secretion by acting on DA D1 receptors of the pancreas in dogs. Intravenous administration of Zelandopam produces renal vasodil... | |||
T68600 | Enoximone sulfoxide | ||
Enoximone sulfoxide is a selective phosphodiesterase III (PDE3) inhibitor with vasodilating and positive inotropic activity that does not cause changes in myocardial oxygen consumption. Enoximone prevents the degradation... |