tinnitus

Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.

Caroverine hydrochloride (Caroverine HCL) is a potent, competitive and reversible antagonist of NMDA and AMPA glutamate receptor. It is also an antioxidant and calcium-blocking agent that exhibits vasorelaxant action, and can be used for the research of inner ear tinnitus.

Selurampanel (BGG492) is an orally active and selective competitive AMPA glutamate receptor antagonist, a quinazoline-dione sulfonamide. selurampanel is used in the study of epilepsy, migraine and tinnitus.

Necrostatin 2 is a necrotic protein and receptor-interacting protein kinase 1 (RIPK1) inhibitor used to study inner ear disorders such as sudden deafness, dizziness and tinnitus.

(S)-Baclofen has effects on excitation in the ascending auditory pathway leading to it a potential reagent for the treatment of hyperactive auditory disorders such as hyperacusis and tinnitus.

HCN2 modulator-8 is a pyrazolopyridine derivative and a selective HCN2 inhibitor. It can be utilized in research related to pain, tinnitus, central nervous system disorders, psychiatric conditions, and mood disorders.

HCN2 modulator-6 is an inhibitor of the HCN2 ion channel with an IC50 of 7 nM. It effectively suppresses the activity of HCN2 ion channels and can be used in research related to pain, inflammatory pain, neuropathic pain, tinnitus, central nervous system disorders, psychiatric disorders, and mood disorders.

HCN2 modulator-5 (S-configuration 39) is an inhibitor of the HCN2 ion channel. It effectively hinders the activity of HCN2 ion channels and is applicable in research focused on pain, inflammatory pain, neuropathic pain, tinnitus, central nervous system disorders, psychiatric conditions, and mood disorders.

HCN2-IN-4 is an orally active inhibitor of the HCN2 ion channel. It effectively suppresses HCN2 ion channel activity and is useful for research related to pain, tinnitus, and central nervous system disorders.

Hexylcaine HCl also called cyclaine or osmocaine, is a short-acting local anesthetic. It acts by inhibiting sodium channel conduction. Overdose can lead to headache, tinnitus, numbness and tingling around the mouth and tongue, convulsions, inability to breathe, and decreased heart function.

Neramexane Free Base is a drug related to memantine, which acts as an NMDA antagonist and has neuroprotective effects. It is being developed for various possible applications, including treatment of tinnitus, Alzheimer's disease, drug addiction and as an analgesic.

Gacyclidine hydrochloride is a N-methyl-D-aspartate (NMDA) receptor antagonist potentially for the treatment of tinnitus.

NK1 Receptor Antagonist 2, a compound targeting the NK1 receptor, holds potential for tinnitus and hearing loss research.