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Results for "

cb1 antagonist 1

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    17
    TargetMol | Inhibitors_Agonists
CB1 antagonist 1
T10510890037-68-0
CB1 antagonist 1 is a CB1 receptor antagonist, used in the research of obesity and metabolic syndrome, neuroinflammatory disorders, cognitive disorders, and gastrointestinal disorders, psychosis, and cardiovascular.
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8-10 weeks
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Rimonabant hydrochloride
SR 151716A, SR 141716A
T1519158681-13-1
Rimonabant hydrochloride (SR 141716A) is a cannabinoid receptor antagonist, binding selectively to central cannabinoid receptors (CB1) with high affinity.
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AM251
T1915183232-66-8
AM251 is a effective CB1 receptor antagonist (IC50 Ki: 8 7.49 nM) that displays 306-fold selectivity over CB2 receptors; also effective GPR55 agonist (EC50: 39 nM).
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CB1-IN-1
DBPR211
T59961429239-98-4
CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.
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TargetMol | Inhibitor Sale
CB1 antagonist 4
T85111253641-65-4
CB1 antagonist 4 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.
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Taranabant racemate
MK-0364 racemate
T13081701977-00-6
Taranabant racemate is an antagonist and or inverse agonist of the Cannabinoid-1 (CB1) receptor.
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7-10 days
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CB1 antagonist 2
AM4113
T14881614726-85-1
CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.
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LH 21
T21811611207-11-5
LH-21 is a potent in vivo neutral cannabinoid CB1 receptor antagonist that reduces food intake and body weight gain in obese Zucker rats, resulting in a dose-dependent inhibition of feeding [1].
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6-8 weeks
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(s)-slv 319
T21914464213-10-3
Ibipinabant (SLV319) is a potent, selective, and orally active cannabinoid CB1 receptor antagonist, with a K_i of 7.8 nM and over 1000-fold selectivity for CB1 compared to CB2 (K_i = 7943 nM). It is utilized in obesity and diabetes research [1] [2] [3].
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6-8 weeks
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(r)-slv 319
T22140656827-86-0
(R)-SLV 319 is a potent and selective antagonist of cannabinoid receptor 1 (CB1) with a Ki value of 894 nM. It is the dextrorotatory counterpart of SLV 319 [1].
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6-8 weeks
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AM6545
AM-6545, AM 6545
T225631245626-05-4
AM6545 is a selective and potent peripheral restricted cannabinoid receptor 1 (CB1) antagonist that inhibits the CB2 receptor, ameliorates hypometabolic obesity and improves adipokine secretion in monosodium glutamate-induced obese mice, and may be useful in the study of obesity and diabetes.
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6-8 weeks
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o-2050
T230991883545-42-3
O-2050 is a high-affinity cannabinoid CB1 receptor antagonist with a Ki of 2.5 nM and inhibits the cannabinoid CB2 receptor with a Ki of 0.2 nM. O-2050 decreased food intake and stimulated locomotion in mice [1].
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8-10 weeks
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amauromine
T3656688360-87-6
Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.
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8-10 weeks
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Isopropyl dodec-11-enylfluorophosphonate
IDEFP
T78674623114-64-7
Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester that serves as a central cannabinoid receptor (CB1) antagonist and equally inhibits fatty acid amide hydrolase (FAAH), both with an IC50 value of 2 nM [1].
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8-10 weeks
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(R)-Monlunabant
(R)-MRI-1891
T835332765579-76-6
(R)-Monlunabant ((R)-MRI-1891) is a CB1 receptor antagonist used in obesity and metabolic disease research [1].
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8-10 weeks
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urb447
T844881132922-57-6
URB447, a peripherally restricted CB1 cannabinoid antagonist with IC50 values of 313 nM for rat CB1 receptor and 41 nM for human CB2 receptor, effectively reduces food intake and body weight gain in mice. It achieves these effects without penetrating the brain or antagonizing central CB1-dependent responses, making it a potential research tool for obesity studies [1].
  • Inquiry Price
8-10 weeks
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TM38837
T860111034264-77-1
CB1 antagonist 4 is an inverse agonist of cannabinoid receptor 1 (CB1) with an IC50 of 0.4 nM. It can reduce body weight, improve plasma inflammatory markers, and enhance glucose homeostasis [1].
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10-14 weeks
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