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Thyroid hormone receptor(THR)

The thyroid hormone receptor (TR) is a type of nuclear receptor that is activated by binding thyroid hormone.TRs act as transcription factors, ultimately affecting the regulation of gene transcription and translation. These receptors also have non-genomic effects that lead to second messenger activation, and corresponding cellular response.
Cat. No. Product name CAS No. Purity Chemical Structure
T11101 DS08210767 2376334-75-5 98%
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.
T29011 Triiodothyronine Sulfate 31135-55-4 98%
Triiodothyronine Sulfate is a prodrug to the Conventional Hormone Therapy of Hypothyroidism. Triiodothyronine sulfate is the main metabolite of thyroid hormone t...
T25455L Glutaurine aceate T25455L 98%
Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid. Glutaurine aceate, as a hormone, is isolated from par...
T15699 L-Thyroxine sodium salt pentahydrate 6106-07-6 98%
L-Thyroxine sodium salt pentahydrate is a synthetic hormone for the research of hypothyroidism. DIO enzymes convert biologically active thyroid hormone (Triiodot...
T15644 KAT681 373641-87-3 98%
KAT681 is a liver selective thyromimetic.
T7590 Taltirelin 103300-74-9 98%
Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ conc...
T1309 Propylthiouracil 51-52-5 98%
Propylthiouracil is a thyroid peroxidase inhibitor and also a 5' -deiodinase inhibitor.
T13072 Taltirelin acetate 1549593-23-8 98%
Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic ...
T13492 3,5-Diiodothyropropionic acid 1158-10-7 98%
3,5-Diiodothyropropionic acid is a thyroid hormone analog. It induces α-myosin heavy chain mRNA expression, binds to thyroid hormone receptor (Ka: 2.40/M and 4.0...
T1653 Liothyronine 6893-02-3 98%
Liothyronine is an active form of thyroid hormone, binding to β1 thyroid hormone receptor (TRβ1), and activates its activity.
T0952 Carbimazole 22232-54-8 98%
Carbimazole is an Imidazolium thyroid antagonist, which is rapidly transformed into MMI in vivo and can be converted into methidazole in vitro, and can be used i...
T1604 Tiratricol 51-24-1 98%
Tiratricol is a metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials s...
T3595 Resmetirom 920509-32-6 98%
MGL-3196 is a highly selective thyroid hormone receptor β (THR-β) agonist.
T5313 Sobetirome 211110-63-3 98%
Sobetirome is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).
T0864 L-Thyroxine 51-48-9 98%
Levothyroxine is the major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (MONOIODOTYROSINE) and the coupling o...
T23673 AH-3960 862907-48-0 98%
AH-3960 is an thyroid hormone receptor-1 (PTHR1) agonist.
T5360 Eprotirome 355129-15-6 98%
Eprotirome, a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.
T1669 Liothyronine sodium 55-06-1 98%
Liothyronine Sodium is the sodium salt form of liothyronine, a synthetic form of the levorotatory isomer of the naturally occurring thyroid hormone triiodothyron...
T7578 REVERSE T3 5817-39-0 98%
reverse T3 inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.
T9691L (D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate 98%
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate is a highly potent antagonist of parathyroid hormone (PTH) The Ki value is 69 nM in bovine renal cortical membr...
DS08210767
T11101
DS08210767 is a highly potent, orally bioavailable PTHR1 antagonist with IC50 of 90 nM.
Triiodothyronine Sulfate
T29011
Triiodothyronine Sulfate is a prodrug to the Conventional Hormone Therapy of Hypothyroidism. Triiodothyronine sulfate is the main metabolite of thyroid hormone t...
Glutaurine aceate
T25455L
Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid. Glutaurine aceate, as a hormone, is isolated from par...
L-Thyroxine sodium salt pentahydrate
T15699
L-Thyroxine sodium salt pentahydrate is a synthetic hormone for the research of hypothyroidism. DIO enzymes convert biologically active thyroid hormone (Triiodot...
KAT681
T15644
KAT681 is a liver selective thyromimetic.
Taltirelin
T7590
Taltirelin is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic Ca2+ conc...
Propylthiouracil
T1309
Propylthiouracil is a thyroid peroxidase inhibitor and also a 5' -deiodinase inhibitor.
Taltirelin acetate
T13072
Taltirelin acetate is a superagonist at thyrotropin-releasing hormone receptor (TRH-R)(IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in cytosolic ...
3,5-Diiodothyropropionic acid
T13492
3,5-Diiodothyropropionic acid is a thyroid hormone analog. It induces α-myosin heavy chain mRNA expression, binds to thyroid hormone receptor (Ka: 2.40/M and 4.0...
Liothyronine
T1653
Liothyronine is an active form of thyroid hormone, binding to β1 thyroid hormone receptor (TRβ1), and activates its activity.
Carbimazole
T0952
Carbimazole is an Imidazolium thyroid antagonist, which is rapidly transformed into MMI in vivo and can be converted into methidazole in vitro, and can be used i...
Tiratricol
T1604
Tiratricol is a metabolite of T3 and T4 thyroid hormones; promoted for hyperlipidemia, localized lipodystrophy, and obesity. Tiratricol has been used in trials s...
Resmetirom
T3595
MGL-3196 is a highly selective thyroid hormone receptor β (THR-β) agonist.
Sobetirome
T5313
Sobetirome is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).
L-Thyroxine
T0864
Levothyroxine is the major hormone derived from the thyroid gland. Thyroxine is synthesized via the iodination of tyrosines (MONOIODOTYROSINE) and the coupling o...
AH-3960
T23673
AH-3960 is an thyroid hormone receptor-1 (PTHR1) agonist.
Eprotirome
T5360
Eprotirome, a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.
Liothyronine sodium
T1669
Liothyronine Sodium is the sodium salt form of liothyronine, a synthetic form of the levorotatory isomer of the naturally occurring thyroid hormone triiodothyron...
REVERSE T3
T7578
reverse T3 inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate
T9691L
(D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate is a highly potent antagonist of parathyroid hormone (PTH) The Ki value is 69 nM in bovine renal cortical membr...
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