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Serine/threonin kinase

Serine threonine kinase belongs to protein kinase, which can phosphorylate the OH group of serine or threonine residues. Serine threonine kinases contain Rho kinase, Aurora kinase, AMP kinase, RAF kinase, Polo like kinase, PIM kinase, ATM kinase and other kinases. The cAMP/cGMP, Ca2+/calmodulin and diacylglycerol and multiple chenmical signals can regulate the activity of serine threonine kinases.
Signaling Pathways | Target | TargetMol
Cat. No. Product name CAS No. Purity Chemical Structure
T16931 SRPKIN-1 2089226-94-6 98%
SRPKIN-1
SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
T8957 CRT0066101 956121-30-5 98%
CRT0066101
CRT0066101 is an inhibitor of PKD.
T3060 Fasudil hydrochloride 105628-07-7 99.98%
Fasudil hydrochloride
Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.
T8362 Benzamidine hydrochloride 1670-14-0 99.97%
Benzamidine hydrochloride
Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 μM, r...
T8535 GAK inhibitor 49 319492-82-5 99.93%
GAK inhibitor 49
GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
T8957L CRT0066101 dihydrochloride(956121-30-5 free base) 2308510-39-4 99.92%
CRT0066101 dihydrochloride(956121-30-5 free base)
CRT0066101 dihydrochloride is an inhibitor of PKD.
T1808 Kb-NB77-78 1350622-33-1 99.89%
kb-NB77-78
kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor).
TQ0104 CRT0066101 dihydrochloride 1883545-60-5 99.85%
CRT0066101 dihydrochloride
CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
T1606 Fasudil 103745-39-7 99.84%
Fasudil
Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
T2458 CID755673 521937-07-5 99.84%
CID755673
CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CA...
T9276 SBC-115337 423148-46-3 99.81%
SBC-115337
SBC-115337 is a PCSK9 inhibitor.
T4524 SBC-110736 1629166-02-4 99.76%
SBC-110736
SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor
T6283 Wortmannin 19545-26-7 99.76%
Wortmannin
Wortmannin (SL-2052) is a PI3K inhibitor (IC50=3 nM) that is covalent and irreversible. Wortmannin is also an inhibitor of PlK1 and PlK3 (IC50=5.8/48 nM) that bl...
T4291 (+)-Isocorydine hydrochloride 13552-72-2 99.72%
(+)-Isocorydine hydrochloride
(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.
T4058 R-IMPP 2133832-83-2 99.7%
R-IMPP
R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells by increasing LDL-R levels, without altering levels of secreted ...
T2391 Camostat mesylate 59721-29-8 99.69%
Camostat mesylate
Camostat mesylate (FOY-S980) is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.
T15781 LP-935509 1454555-29-3 99.64%
LP-935509
LP-935509 is highly brain-penetrant and reverses fully established pain behavior following the SNL procedure. LP-935509 is also an effective inhibitor of BIKE (I...
T3050 ML-7 hydrochloride 110448-33-4 99.61%
ML-7 hydrochloride
ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM); also...
TP1890L1 MLCK inhibitor peptide 18 acetate TP1890L1 99.57%
MLCK inhibitor peptide 18 acetate
MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinas...
T7444 6-(Dimethylamino)purine 938-55-6 99.49%
6-(Dimethylamino)purine
6-(Dimethylamino)purine (N,N-Dimethyladenine) is a serine threonine protein kinase and CDK inhibitor
SRPKIN-1
T16931
SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
CRT0066101
T8957
CRT0066101 is an inhibitor of PKD.
Fasudil hydrochloride
T3060
Fasudil hydrochloride (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK with Ki of 0.33 μM, 1.0 μM, 9.3 μM and 55 μM, respectively.
Benzamidine hydrochloride
T8362
Benzamidine hydrochloride (Benzamidine HCl) is a reversible inhibitor of serine proteases, including trypsin, plasmin, and thrombin (Ki of 35, 350, and 220 μM, r...
GAK inhibitor 49
T8535
GAK inhibitor 49 is a highly selective and ATP-competitive cyclin G associated kinase (GAK) inhibitor (IC50: 56 nM; Ki: 0.54 nM ).
CRT0066101 dihydrochloride(956121-30-5 free base)
T8957L
CRT0066101 dihydrochloride is an inhibitor of PKD.
kb-NB77-78
T1808
kb-NB77-78 is an analog of CID797718, which is a by-product of the synthesis of the parental compound, CID755673(PKD1 inhibitor).
CRT0066101 dihydrochloride
TQ0104
CRT0066101 dihydrochloride is an effective and selective PKD inhibitor (IC50s: 1, 2.5 and 2 nM for PKD1, 2, and 3).
Fasudil
T1606
Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
CID755673
T2458
CID755673 is an effective and specific cell-active inhibitor for PKD (IC50: 182 nM); exhibits selective PKD1 inhibition when compared with PLK1, AKT, CAMKIIα, CA...
SBC-115337
T9276
SBC-115337 is a PCSK9 inhibitor.
SBC-110736
T4524
SBC-110736 is a proprotein convertase subtilisin kexin type 9 (PCSK9) inhibitor
Wortmannin
T6283
Wortmannin (SL-2052) is a PI3K inhibitor (IC50=3 nM) that is covalent and irreversible. Wortmannin is also an inhibitor of PlK1 and PlK3 (IC50=5.8/48 nM) that bl...
(+)-Isocorydine hydrochloride
T4291
(+)-Isocorydine hydrochloride (Isocorydine HCl) is a eukaryote protein kinases Inhibitor.
R-IMPP
T4058
R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells by increasing LDL-R levels, without altering levels of secreted ...
Camostat mesylate
T2391
Camostat mesylate (FOY-S980) is a trypsin-like protease inhibitor and inhibits airway epithelial sodium channel (ENaC) function.
LP-935509
T15781
LP-935509 is highly brain-penetrant and reverses fully established pain behavior following the SNL procedure. LP-935509 is also an effective inhibitor of BIKE (I...
ML-7 hydrochloride
T3050
ML-7 hydrochloride (ML-7 HCl) is a cell-permeable, reversible, effective, ATP-competitive, and specific inhibitor of myosin light chain kinase (Ki: 300 nM); also...
MLCK inhibitor peptide 18 acetate
TP1890L1
MLCK inhibitor peptide 18 acetate is a selective competitive inhibitor of myosin light chain kinase (IC50 = 50 nM). Displays 4000-fold selectivity over CaM kinas...
6-(Dimethylamino)purine
T7444
6-(Dimethylamino)purine (N,N-Dimethyladenine) is a serine threonine protein kinase and CDK inhibitor
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TargetMol