T8957 |
CRT0066101
|
956121-30-5
|
98%
|
|
CRT0066101 is an inhibitor of PKD.
|
T16931 |
SRPKIN-1
|
2089226-94-6
|
98%
|
|
SRPKIN-1 is a covalent and irreversible inhibitor of SRPK1/2 (IC50s: 35.6 and 98 nM, respectively).
|
T24152 |
HTH-01-091
|
2000209-42-5
|
98%
|
|
HTH-01-091 is a potent and selective maternal embryonic leucine zipper kinase (MELK) inhibitor (IC50: 10.5 nM).HTH-01-091 inhibits PIM1/2/3, RIPK2, DYRK3, smMLCK...
|
T1606 |
Fasudil
|
103745-39-7
|
98%
|
|
Fasudil is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.
|
T5456 |
WNK-IN-11
|
2123489-30-3
|
98%
|
|
WNK-IN-11 is an allosteric With-No-Lysine (WNK) kinase inhibitor,WNK1(IC50 : 4 nM)
|
T4058 |
R-IMPP
|
2133832-83-2
|
98%
|
|
R-IMPP is an inhibitor of PCSK9 translation. R-IMPP stimulates uptake of LDL-C in hepatoma cells by increasing LDL-R levels, without altering levels of secreted ...
|
T11666 |
IPR-803
|
892243-35-5
|
98%
|
|
IPR-803 is an effective inhibitor of the uPAR·uPA protein-protein interaction (PPI) with anti-tumor activity. IPR-803 binds directly to uPAR with a Ki of 0.2 μM....
|
T10547 |
BioE-1115
|
1268863-35-9
|
98%
|
|
BioE-1115 is a selective and potent inhibitor of serine-threonine protein kinase (PASK, IC50 = 4 nM). BioE-1115 is a potent inhibitor of CK2α (IC50 = 10 μM).
|
T7017 |
WNK463
|
2012607-27-9
|
98%
|
|
WNK463 is a pan-WNK-kinase inhibitor. It effectively inhibits the in vitro kinase activity of all four WNK family members (WNK1/2/3/4).
|
T19763 |
Cetraxate hydrochloride
|
27724-96-5
|
98%
|
|
Cetraxate HCl is an oral gastrointestinal medication. It has a cytoprotective effect.
|
T9256 |
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine
|
1071135-06-2
|
98%
|
|
N-Cyclohexyl-4-[1-(1-piperazinyl)-2,6-naphthyridin-3-yl]-2-pyridinamine is a novel 2,6-naphthyridine identified by high throughput screen (HTS) as a dual protein...
|
T77501 |
TAO Kinase inhibitor 2
|
850467-77-5
|
98%
|
|
TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
|
T13257 |
Upamostat
|
590368-25-5
|
98%
|
|
Upamostat is an inhibitor of a serine protease and is a urokinase plasminogen activator (uPA) inhibitor.
|
T72025 |
PCSK9-IN-10
|
368434-98-4
|
98%
|
|
PCSK9-IN-10 is a potent and orally active PCSK9 inhibitor with an IC 50 value of 6.4 µM. PCSK9-IN-10 increases the expression of LDLR protein and decreases the e...
|
T27525 |
HA-1004
|
91742-10-8
|
98%
|
|
HA-1004 is a inhibitor of PKG, PKA, PKC and MLC.
|
T8676 |
FOY 251
|
71079-09-9
|
98%
|
|
FOY 251 is a proteinase inhibitor, and is an anti-proteolytic active metabolite camostate.
|
T10572L |
BMT-124110 Formate
|
T10572L
|
98%
|
|
BMT-124110 Formate is a selective AAK1 inhibitor (IC50: 0.9 nM) with anti-injury sensory activity.BMT-124110 Formate inhibits the BMP-2-inducible protein kinase ...
|
T2153 |
1-NM-PP1
|
221244-14-0
|
98%
|
|
1 nM-PP1 is a cell-permeable PP1 analog that acts as a potent and selective inhibitor of mutant kinases over their wild-type progenitors.
|
T1858 |
CID-797718
|
370586-05-3
|
98%
|
|
CID797718 is a protein kinase D1 (PKD1) inhibitor.
|
T5194 |
SPHINX31
|
1818389-84-2
|
98%
|
|
SPHINX31 is a potent inhibitor of serine/arginine-rich protein kinase 1 (SRPK1; IC50: 5.9 nM).
|