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Results for "
tgr1202 tosylate
" in TargetMol Product Catalog- Inhibitors & Agonists1
umbralisib tosylate
TGR-1202 tosylate ; RP5264 tosylate, TGR-1202 tosylate, RP5264 tosylate
T724651532533-72-4
Umbralisib Tosylate (TGR-1202) is a potent, selectively dual inhibitor targeting PI3Kδ and casein kinase-1-ε (CK1ε), demonstrating oral activity. With EC50 values of 22.2 nM and 6.0 μM for PI3Kδ and CK1ε respectively, it shows unique immunomodulatory effects on T cells in chronic lymphocytic leukemia (CLL). This compound is utilized in the research of hematological malignancies.
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