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Results for "

muscle relaxant

" in TargetMol Product Catalog
  • Inhibitors & Agonists
    110
    TargetMol | Inhibitors_Agonists
  • Natural Products
    8
    TargetMol | Natural_Products
  • Isotope Products
    3
    TargetMol | Isotope_Products
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    1
    TargetMol | Inhibitors_Agonists
CS-722 Free base
T10893749179-13-3In house
CS-722 Free base is a synthetic central muscle relaxant exhibiting muscle relaxant effects and inhibition of spinal reflexes. In hippocampal cultures, CS-722 Free base may suppress spontaneous inhibitory and excitatory post-synaptic currents by inhibiting sodium and calcium currents.
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6-8 weeks
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Silperisone HCl
RGH5002, SILA336, RGH-5002, Silperisone hydrochloride, SILA-336
T28778140944-30-5In house
Silperisone HCl (RGH-5002) blocks sodium and calcium channels in cells, decreases excitability and contractility of muscle cells, reduces peripheral tone, and acts as a muscle relaxant and peripheral vasodilator. Silperisone HCl is used to treat recurrent painful myoclonus due to spinal cord injury, abnormal hypertonia due to cerebrovascular disease, dystonia symptoms, cone tension syndrome, multiple sclerosis myospasm and myelitis. silperisone is a sodium channel protein type 2 alpha channel blocker. silperisone is an organosilicon similar to tolperisone, an organosilicon compound with centrally acting muscle relaxant properties.
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6-8weeks
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Inaperisone
T6808799323-21-4In house
Inaperisone is a novel centrally acting muscle relaxant that inhibits the voiding reflex. Inaperisone may inhibit the voiding reflex by acting indirectly on GABAB receptors in the brainstem.
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Lanperisone HCl
NK 433
T71356116287-13-9In house
Lanperisone HCl (NK 433) is a novel orally available centrally acting muscle relaxant with anticancer activity and inhibits mono- and polysynaptic reflex potentials.Lanperisone HCl acts by inducing non-apoptotic cell death in the cell cycle and translational independence.
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6-8 weeks
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Mephenesin
Cresoxydiol, Memphenesin, Mephedan, Decontractyl
T001559-47-2
Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.
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Dantrolene sodium
Dantrolene sodium salt
T007714663-23-1
Dantrolene sodium (Dantrolene sodium salt) is a skeletal muscle relaxant and can interfere with excitation-contraction coupling in the muscle fiber. It is used for the treatment of spasticity and other neuromuscular abnormalities. Its mechanism of action is may not central, but dantrolene is usually grouped with the central muscle relaxants.
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Rocuronium bromide
ORG 9426, ORG 9426 (Bromide)
T0156119302-91-9
Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker. During surgery or mechanical ventilation, it is used to facilitate endotracheal intubation and to provide skeletal muscle relaxation.
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Pancuronium dibromide
Pancuronium bromide, Pavulon
T016615500-66-0
Pancuronium dibromide (Pavulon), a competitive AChR antagonist (IC50 = 5.5 nM), acts as a skeletal muscle relaxant. Pancuronium dibromide(Pancuronium bromide) blocking neuromuscular transmission is achieved by competing with acetylcholine for receptor sites on the motor end-plate.
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Cyclandelate
BS 572, 3,5,5-Trimethylcyclohexyl mandelate
T0504456-59-7
Cyclandelate (BS 572), a direct-acting smooth muscle relaxant, is used to dilate blood vessels.
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Tolperisone hydrochloride
Tolperisone HCl, Muscalm, Midocalm
T05113644-61-9
Tolperisone hydrochloride (Muscalm), a centrally acting muscle relaxant, is used in the therapy of pathologically increased tone of the cross-striated muscle resulted by neurological diseases (damage of the encephalomyelitis, myelopathy, multiple sclerosis, pyramidal tract) and of spastic paralysis and other encephalopathies manifested with muscular dystonia.
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Homoveratronitrile
T056393-17-4
Homoveratronitrile is an impurity of Verapamil. It is also an intermediate in the preparation of the muscle relaxant Papverine.
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Carbenoxolone disodium
Biogastrone, Duogastrone, Bioral
T09927421-40-1
Carbenoxolone disodium (Duogastrone) salt is an agent derived from licorice root. It is used for the treatment of digestive tract ulcers, especially in the stomach. Antidiuretic side effects are frequent, but otherwise, the drug is low in toxicity.
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Methocarbamol
Robaxin, Metocarbamol, Lumirelax, AHR 85
T1409532-03-6
Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established. It is used as an adjunct in the symptomatic treatment of musculoskeletal conditions associated with painful muscle spasm.
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Cisatracurium besylate
51W89
T145996946-42-8
Cisatracurium besylate (51W89) is a nondepolarizing skeletal muscle relaxant intended for intravenous administration.
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Fesoterodine fumarate
Toviaz, SPM 907
T1475286930-03-8
Fesoterodine fumarate (Toviaz) is the fumarate salt form of fesoterodine, a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties. Fesoterodine is rapidly hydrolyzed in vivo into its active metabolite 5-hydroxymethyl tolterodine, which binds and inhibits muscarinic receptors on the bladder detrusor muscle, thereby preventing bladder contractions or spasms caused by acetylcholine.
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Vecuronium bromide
ORG NC 45
T159450700-72-6
Vecuronium bromide (ORG NC 45) is a synthetic, intermediate-acting, mono-quaternary steroid that functions as a non-depolarizing neuromuscular blocking agent with muscle relaxant properties.
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Metaxalone
Zorane, Skelaxin, NSC170959, Methaxalonum, AHR438
T16101665-48-1
Metaxalone (Methaxalonum) (marketed by King Pharmaceuticals under the brand name Skelaxin ) is a muscle relaxant used to relax muscles and relieve pain caused by strains, sprains, and other musculoskeletal conditions.
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Chlorzoxazone
Paraflex, Chlorzoxazon
T165095-25-0
Chlorzoxazone (Chlorzoxazon) is a Muscle Relaxant. The physiologic effect of chlorzoxazone is by means of Centrally-mediated Muscle Relaxation.
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Dantrolene sodium hemiheptahydrate
Dantrolene sodium hydrate, Dantrolene sodium salt, Dantrium, Sodium dantrolene
T405424868-20-0
Dantrolene depresses excitation-contraction coupling in skeletal muscle by binding to the ryanodine receptor 1 and decreasing intracellular calcium concentration. Ryanodine receptors mediate the release of calcium from the sarcoplasmic reticulum, an essential step in muscle contraction. Dantrolene sodium hemiheptahydrate (Sodium dantrolene) is the sodium salt form of dantrolene, a hydantoin derivative, and direct-acting skeletal muscle relaxant.
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Quinine dihydrochloride
Quinine bimuriate
T433360-93-5
Quinine dihydrochloride (Quinine bimuriate) is a primary alkaloid of various species of Cinchona (Rubiaceae). It is also an antimalarial and muscle relaxant (skeletal).
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Eperisone hydrochloride
T500556839-43-1
Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.
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Phenprobamate
Proformiphen, MH 532, 3-Phenylpropyl carbamate
T64851673-31-4
Phenprobamate (MH 532) is a relaxant that acts on central skeletal muscle and has anticonvulsant and psychostimulant effects.
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7-10 days
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Dantrolene
T84527261-97-4
Dantrolene is a postsynaptic muscle relaxant by inhibiting Ca2+ ions release from sarcoplasmic reticulum stores by antagonizing ryanodine receptors.
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Zoxazolamine
NSC 24995, Contrazole
T092261-80-3
Zoxazolamine (NSC-24995) is a uricosuric and muscle relaxant. Zoxazolamine acts centrally as a muscle relaxant, but the mechanism of its action is not understood.
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