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Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.
Cat. No. Product name CAS No. Purity Chemical Structure
T28257 OPC-51803 192514-54-8 98%
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.
T7434 Argipressin 113-79-1 98%
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
T4996 Atosiban 90779-69-4 98%
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
TP2082L D[Cha4]-AVP acetate(500170-27-4 free base) TP2082L 98%
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
TP1192L Conopressin S acetate(111317-90-9 free base) TP1192L 98%
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
T13920L Terlipressin Acetate 1884420-36-3 98%
Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
T2568 Felypressin 56-59-7 98%
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
T14494 Balovaptan 1228088-30-9 98%
Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
T7303 LIXIVAPTAN 168079-32-1 98%
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
T6288 Mozavaptan 137975-06-5 98%
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T5148 Atosiban acetate 914453-95-5 98%
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
TP1927L1 D[Leu4,Lys8]-VP acetate TP1927L1 98%
d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respe...
T28153 Nelivaptan 439687-69-1 98%
Nelivaptan is a vasopressin V1b receptor antagonist.
T5019 Desmopressin 16679-58-6 98%
Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
T2568L Felypressin acetate 914453-97-7 98%
Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
T2326 Tolvaptan 150683-30-0 98%
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
T15682 L-371,257 162042-44-6 98%
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
T5144 Desmopressin acetate (16679-58-6 free base) 62288-83-9 98%
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
T6453 Conivaptan hydrochloride 168626-94-6 98%
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
T4141 RG7713 920022-47-5 98%
RO5028442 has been used in trials studying Autistic Disorder.
OPC-51803
T28257
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.
Argipressin
T7434
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
Atosiban
T4996
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
d[Cha4]-AVP acetate(500170-27-4 free base)
TP2082L
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
Conopressin S acetate(111317-90-9 free base)
TP1192L
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
Terlipressin Acetate
T13920L
Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
Felypressin
T2568
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
Balovaptan
T14494
Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
LIXIVAPTAN
T7303
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
Mozavaptan
T6288
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
Atosiban acetate
T5148
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
d[Leu4,Lys8]-VP acetate
TP1927L1
d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respe...
Nelivaptan
T28153
Nelivaptan is a vasopressin V1b receptor antagonist.
Desmopressin
T5019
Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
Felypressin acetate
T2568L
Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
Tolvaptan
T2326
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
L-371,257
T15682
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
Desmopressin acetate (16679-58-6 free base)
T5144
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
Conivaptan hydrochloride
T6453
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
RG7713
T4141
RO5028442 has been used in trials studying Autistic Disorder.
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