T28257 |
OPC-51803
|
192514-54-8
|
98%
|
|
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.
|
T7434 |
Argipressin
|
113-79-1
|
98%
|
|
Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
|
T4996 |
Atosiban
|
90779-69-4
|
98%
|
|
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
|
TP2082L |
D[Cha4]-AVP acetate(500170-27-4 free base)
|
TP2082L
|
98%
|
|
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
|
TP1192L |
Conopressin S acetate(111317-90-9 free base)
|
TP1192L
|
98%
|
|
Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
|
T13920L |
Terlipressin Acetate
|
1884420-36-3
|
98%
|
|
Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
|
T2568 |
Felypressin
|
56-59-7
|
98%
|
|
Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
|
T14494 |
Balovaptan
|
1228088-30-9
|
98%
|
|
Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
|
T7303 |
LIXIVAPTAN
|
168079-32-1
|
98%
|
|
Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
|
T6288 |
Mozavaptan
|
137975-06-5
|
98%
|
|
Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
|
T5148 |
Atosiban acetate
|
914453-95-5
|
98%
|
|
Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
|
TP1927L1 |
D[Leu4,Lys8]-VP acetate
|
TP1927L1
|
98%
|
|
d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respe...
|
T28153 |
Nelivaptan
|
439687-69-1
|
98%
|
|
Nelivaptan is a vasopressin V1b receptor antagonist.
|
T5019 |
Desmopressin
|
16679-58-6
|
98%
|
|
Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
|
T2568L |
Felypressin acetate
|
914453-97-7
|
98%
|
|
Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
|
T2326 |
Tolvaptan
|
150683-30-0
|
98%
|
|
Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
|
T15682 |
L-371,257
|
162042-44-6
|
98%
|
|
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
|
T5144 |
Desmopressin acetate (16679-58-6 free base)
|
62288-83-9
|
98%
|
|
Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
|
T6453 |
Conivaptan hydrochloride
|
168626-94-6
|
98%
|
|
Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
|
T4141 |
RG7713
|
920022-47-5
|
98%
|
|
RO5028442 has been used in trials studying Autistic Disorder.
|