Vasopressin Receptor

The actions of vasopressin are mediated by stimulation of tissue-specific G protein-coupled receptors (GPCRs) called vasopressin receptors that are classified into the V1 (V1A), V2, and V3 (V1B) receptor subtypes. These three subtypes differ in localization, function and signal transduction mechanisms.

Cat. No.	Product name	CAS No.	Purity
T7434	Argipressin	113-79-1	98%
T7434	Argipressin is a peptide hormone with vasoconstrictive and antidiuretic activities that binds to the vascular arginine vasopressin receptor, V1, with Kd values o...
T4996	Atosiban	90779-69-4	98%
T4996	Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...
TP1927L1	D[Leu4,Lys8]-VP acetate	TP1927L1	98%
TP1927L1	d[Leu4,Lys8]-VP acetate is a selective vasopressin V1b receptor agonist. The Kis for rat, human and mouse V1b receptors are 0.16 nM, 0.52 nM and 0.1.38 nM, respe...
T5144	Desmopressin acetate (16679-58-6 free base)	62288-83-9	100%
T5144	Desmopressin is the synthetic analog of the antidiuretic hormone arginine vasopressin. Vasopressin Receptor The antidiuretic properties of desmopressin have led ...
T15682	L-371,257	162042-44-6	100%
T15682	L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
T2568L	Felypressin acetate	914453-97-7	97.06%
T2568L	Felypressin acetate is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS. Felypressin acetate can be used in dental procedures.
T5019	Desmopressin	16679-58-6	97.45%
T5019	Desmopressin(DDAVP) is the synthetic analogue of the antidiuretic hormone arginine vasopressin.Vasopressin Receptor The antidiuretic properties of desmopressin h...
T4355	Fuscoside	131631-89-5	97.98%
T4355	OPC 21268 is a non-peptide Arginine vasopressin(AVP) Receptor V antagonist.
T28153	Nelivaptan	439687-69-1	98.35%
T28153	Nelivaptan is a vasopressin V1b receptor antagonist.
T6288	Mozavaptan	137975-06-5	99.26%
T6288	Mozavaptan is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.
T7303	LIXIVAPTAN	168079-32-1	99.33%
T7303	Lixivaptan is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)
T14494	Balovaptan	1228088-30-9	99.34%
T14494	Balovaptan is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) ...
T2568	Felypressin	56-59-7	99.65%
T2568	Felypressin is a synthetic analog of LYPRESSIN with a PHENYLALANINE substitution at residue 2. Felypressin is a vasoconstrictor with reduced antidiuretic activit...
T13920L	Terlipressin Acetate	1884420-36-3	99.69%
T13920L	Terlipressin, a highly selective vasopressin V1 receptor agonist, on oxygen and glucose deprivation/re-oxygenation (OGD/R)-induced damage in intestinal epithelia...
T4141	RG7713	920022-47-5	99.75%
T4141	RO5028442 has been used in trials studying Autistic Disorder.
T2326	Tolvaptan	150683-30-0	99.75%
T2326	Tolvaptan is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.
TP1192L	Conopressin S acetate(111317-90-9 free base)	TP1192L	99.79%
TP1192L	Conopressin S acetate is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b receptor (AVPR1B), with a Ki of 8.3 nM.
T6453	Conivaptan hydrochloride	168626-94-6	99.86%
T6453	Conivaptan HCl is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and euvolemic.
TP2082L	D[Cha4]-AVP acetate(500170-27-4 free base)	TP2082L	99.86%
TP2082L	d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 recept...
T5148	Atosiban acetate	914453-95-5	99.92%
T5148	Atosiban is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature l...