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Search Result

Search Results for " vanilloid receptor "

Targets

TRP/TRPV Channel

47

Compounds

2

Natural Products

Cat No. Product Name Synonyms Targets
T9247 Vanilloid receptor antagonist 1 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile TRP/TRPV Channel
Vanilloid receptor antagonist 1 (4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile) is a potent vanilloid receptor TRPV1 antagonist.
T6977 SB-366791 SB366791 TRP/TRPV Channel
SB-366791 is a new and selective cinnamide TRPV1 antagonist.
T6848 GSK1016790A GSK101 Calcium Channel , TRP/TRPV Channel
GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial cells.
T12306 OMDM-5 Cannabinoid Receptor , Endogenous Metabolite , TRP/TRPV Channel
OMDM-5 is a selective anandamide cellular uptake (ACU)inhibitor(Ki of 4.8 μM).
T83701 TRPV1-Tat TFA Transient Receptor Potential Vanilloid 1-Tat,736-745-Tat
TRPV1-Tat, a peptide antagonist targeting transient receptor potential vanilloid 1 (TRPV1), is composed of amino acids 736-745 derived from TRPV1's A-kinase anchor protein (AKAP)-binding domain, combined with the HIV Tat...
T12302 OMDM-1 (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide Endogenous Metabolite
OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor with a Ki of 2.4 μM.
T23106 Olvanil N-Vanillyloleamide,N-Vannilyloleoylamide TRP/TRPV Channel
Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.
T29522 ABT 102 ABT102,CHEMBL398338,ABT-102 TRP/TRPV Channel
ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
T23322 SB 452533 TRP/TRPV Channel
SB 452533 is an antagonist of the vanilloid receptor 1(pKb: 7.8).
T14087 ABT-239 TRP/TRPV Channel
ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists. It also acts as a transient receptor potential vanilloid type 1 (TRPV1) antagonist.
T13214L TRPV4 agonist-1 free base OUN67600 TRP/TRPV Channel
TRPV4 agonist-1 free base (OUN67600) is an agonist of transient receptor potential vanilloid 4 (TRPV4;EC50 of 60 nM, in the hTRPV4 Ca2+ assay).
T7189 AMG9810 TRP/TRPV Channel
AMG 9810 is a competitive antagonist of capsaicin activation of the vanilloid receptor 1 (TRPV1) (IC50s = 24.5 and 85.6 nM for human and rat TRPV1, respectively).
T37097 SET 2 TRP/TRPV Channel
SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 of 0.46 μM. SET 2 shows selectivity over TRPV1, TRPV3 and TRPV4.
T22360 MDR-652 TRP/TRPV Channel
MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for hTRPV1 and rTRPV1 respectively and EC50s for hTRPV1 and rTRPV1 ...
T23178 PPAHV Others
vanilloid TRPV1 (VR1) receptor agonist
T22527 6'-Iodoresiniferatoxin Others
TRPV1 (VR1) vanilloid receptor partial agonist
T23723 AMG8163 AMG 8163,AMG-8163
AMG8163 is an antagonist of vanilloid receptor TRPV1.
T24237 JYL-79 JYL79,JYL 79
JYL-79 is an agonist of the vanilloid receptor.
T23721 AMG7905 AMG-7905,AMG 7905
AMG7905 is a modulator of transient receptor potential vanilloid type 1.
T26663 AS1928370
AS1928370 is an antagonist of transient receptor potential vanilloid 1 (TRPV1).
T10176 TRPV antagonist 1 Others
TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 < 250 nM).
T16426 Asivatrep PAC-14028 Others
Asivatrep is an effective and selective transient receptor potential vanilloid type I antagonist.
T26386 4alpha-PDD 4α-Phorbol 12,13-didecanoate
4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.
T68256 JNJ-38893777
JNJ-38893777 is a potent and selective transient receptor potential vanilloid 1 (TRPV1) channel antagonist.
T69785 GSK3527497
GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).
T37086 PDDHV
PDDHV is a resiniferatoxin-type phorboid vanilloid with capsaicin-like selectivity for the cloned rat transient receptor potential cation channel subfamily V member 1 (TRPV1), formerly known as vanilloid receptor 1. It i...
T15439 GSK3395879 TRP/TRPV Channel
GSK3395879 is a selective and orally bioavailable antagonist of transient receptor potential vanilloid-4 (TRPV4) (IC50: 1 nM for hTRPV4).
TP1934 L-R4W2
Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC50 ~ 0.1 μM); blocks Ca2+ currents in dorsal root ganglion neurons. Analgesic in vivo.
T37668 CAY10448 CAY10448
Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Capsaicin signals are transduced by a heat-activated ion channel, the vanilloid receptor 1 (VR1), or...
T39293 Tivanisiran SYL1001,Tivanisiran
Tivanisiran (SYL1001) is a siRNA developed specifically to inhibit the expression of transient receptor potential vanilloid 1 (TRPV1) to explore its implications in dry eye disease research.
T71563 10-oxo-12(Z)-Octadecenoic Acid
10-oxo-12(Z)-Octadecenoic acid is a metabolite of linoleic acid and an activator of transient receptor potential vanilloid 1 (TRPV1) and selectively increases calcium levels in HEK293 cells expressing TRPV1.
T41091 JTS-653
JTS-653 is a potent and selective in vitro and in vivo antagonist of transient receptor potential vanilloid 1 (TRPV1). It effectively attenuates chronic pain resistant to non-steroidal anti-inflammatory drugs.
T15434 GSK2798745 TRP/TRPV Channel
GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: 1.8 and 1.6 nM for hTRPV4 and rTRPV4). It is used in research for the treatment of pulmonary edema associated wi...
T76369 CEDAEVFKDSMVPGEK
CEDAEVFKDSMVPGEK, the peptide sequence corresponding to the rat vanilloid receptor subtype 1 (VR1), facilitates the detection and mapping of VR1 distribution [1].
T69784 GSK3527497 HCl
GSK3527497 is a potent and selective inhibitor of Transient Receptor Potential Vanilloid‑4 (TRPV4) with IC50 = 12 nM) for the treatment of heart failure and respiratory diseases. GSK3527497 is a preclinical candidate sui...
T37092 20-HEPE
20-HEPE is a metabolite of eicosapentaenoic acid that is formed via ω-oxidation of EPA by cytochrome P450 (CYP) ω-oxidases, including human CYP4F3B. It activates peroxisome proliferator-activated receptor α (PPARα) in CO...
T75830 L-R4W2 TFA
L-R4W2 TFA acts as a potent antagonist of vanilloid receptor 1 (VR1, TRPV1), demonstrating significant inhibitory activity with an IC50 value of 0.1 μM. This compound potentially offers powerful analgesic properties [1] ...
T35921 N-Oleoyl Valine
N-Oleoyl valine is an endogenous N-acyl amine that acts as an antagonist at the transient receptor potential vanilloid type 3 (TRPV3) receptor, which is involved in thermoregulation. N-Oleoyl valine is increased in mice ...
T37321 RN-9893 (hydrochloride)
RN-9893 is an antagonist of transient receptor potential vanilloid 4 (TRPV4; IC50s = 0.42 and 0.66 μM, respectively, for the human and rat receptors).1 It is selective for TRPV4 over TRPV1, TRPV3, and TRPM8 (IC50s = 10, ...
T71295 SOR-C13
SOR-C13 is an inhibitor of transient receptor potential cation channel vanilloid family member 6 (TRPV6, CaT1 or CATL) with potential antineoplastic activity. TRPV6 calcium channel inhibitor SOR-C13 binds to TRPV6 and pr...
T62543 JNc-440
JNc-440 is a potent anti-hypertensive agent. jNc-440 enhances the interaction between the transient receptor potential vanilloid subtype 4 (TRPV4) and calcium-activated potassium channel 3 (KCa2.3) in endothelial cells. ...
T36064 N-Oleoyl Glutamine
N-Oleoyl glutamine is an endogenous N-acyl amine.1,2It is both formed and degraded by peptidase M20 domain-containing 1 (PM20D1), a factor secreted by thermogenic adipose cells. N-Oleoyl glutamine (50 μM) induces mitocho...
T37732 AMG 21629
Potent and selective TRPV1 antagonist. Blocks Ca2+ uptake by CHO cells expressing TRPV1 receptors and acid-induced Ca2+ uptake, respectively). Exhibits >4000-fold selectivity for TRPV1 over other TRP channels. Blocks cap...
T35918 N-Arachidonoyl Taurine
N-Arachidonoyl taurine is an arachidonoyl amino acid. It is oxygenated by 12(S)- and 15(S)-lipoxygenase and is converted to 12-HETE-taurine (12-HETE-T) in murine resident peritoneal macrophages. N-Arachidonoyl taurine is...
T21750 A 784168
A-784168, a potent and orally active inhibitor of vanilloid receptor type 1 (TRPV1), acts on a ligand-gated nonselective cation channel pivotal in integrating pain stimuli including endogenous lipids, capsaicin, heat, an...
T38028 (R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
N-Acyl ethanolamines (NAEs) have diverse biological actions that are strongly affected by the associated acyl group. Docosahexaenoyl ethanolamide (DHEA) has potential signaling roles in cancer, inflammation, and neurolog...
T83728 Tat-AKAP79 (326-336) TFA Tat-A-kinase Anchor Protein 79 (326-336)
Tat-AKAP79 (326-336) is a peptide that links the HIV-1 Tat protein transduction domain with an 11-amino acid sequence from A-kinase anchor protein 79 (AKAP79). This compound effectively inhibits the activation-induced se...

Compounds

Vanilloid receptor antagonist 1
T9247
Synonym: 4-(7-Hydroxy-2-isopropyl-4-oxoquinazolin-3(4H)-yl)benzonitrile
Target: TRP/TRPV Channel
SB-366791
T6977
Synonym: SB366791
Target: TRP/TRPV Channel
GSK1016790A
T6848
Synonym: GSK101
Target: Calcium Channel, TRP/TRPV Channel
OMDM-5
T12306
Synonym:
Target: Cannabinoid Receptor, Endogenous Metabolite, TRP/TRPV Channel
TRPV1-Tat TFA
T83701
Synonym: Transient Receptor Potential Vanilloid 1-Tat,736-745-Tat
Target:
OMDM-1
T12302
Synonym: (Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide
Target: Endogenous Metabolite
Olvanil
T23106
Synonym: N-Vanillyloleamide,N-Vannilyloleoylamide
Target: TRP/TRPV Channel
ABT 102
T29522
Synonym: ABT102,CHEMBL398338,ABT-102
Target: TRP/TRPV Channel
SB 452533
T23322
Synonym:
Target: TRP/TRPV Channel
ABT-239
T14087
Synonym:
Target: TRP/TRPV Channel
TRPV4 agonist-1 free base
T13214L
Synonym: OUN67600
Target: TRP/TRPV Channel
AMG9810
T7189
Synonym:
Target: TRP/TRPV Channel
SET 2
T37097
Synonym:
Target: TRP/TRPV Channel
MDR-652
T22360
Synonym:
Target: TRP/TRPV Channel
PPAHV
T23178
Synonym:
Target: Others
6'-Iodoresiniferatoxin
T22527
Synonym:
Target: Others
AMG8163
T23723
Synonym: AMG 8163,AMG-8163
Target:
JYL-79
T24237
Synonym: JYL79,JYL 79
Target:
AMG7905
T23721
Synonym: AMG-7905,AMG 7905
Target:
AS1928370
T26663
Synonym:
Target:
TRPV antagonist 1
T10176
Synonym:
Target: Others
Asivatrep
T16426
Synonym: PAC-14028
Target: Others
4alpha-PDD
T26386
Synonym: 4α-Phorbol 12,13-didecanoate
Target:
JNJ-38893777
T68256
Synonym:
Target:
GSK3527497
T69785
Synonym:
Target:
PDDHV
T37086
Synonym:
Target:
GSK3395879
T15439
Synonym:
Target: TRP/TRPV Channel
L-R4W2
TP1934
Synonym:
Target:
CAY10448
T37668
Synonym: CAY10448
Target:
Tivanisiran
T39293
Synonym: SYL1001,Tivanisiran
Target:
10-oxo-12(Z)-Octadecenoic Acid
T71563
Synonym:
Target:
JTS-653
T41091
Synonym:
Target:
GSK2798745
T15434
Synonym:
Target: TRP/TRPV Channel
CEDAEVFKDSMVPGEK
T76369
Synonym:
Target:
GSK3527497 HCl
T69784
Synonym:
Target:
20-HEPE
T37092
Synonym:
Target:
L-R4W2 TFA
T75830
Synonym:
Target:
N-Oleoyl Valine
T35921
Synonym:
Target:
RN-9893 (hydrochloride)
T37321
Synonym:
Target:
SOR-C13
T71295
Synonym:
Target:
JNc-440
T62543
Synonym:
Target:
N-Oleoyl Glutamine
T36064
Synonym:
Target:
AMG 21629
T37732
Synonym:
Target:
N-Arachidonoyl Taurine
T35918
Synonym:
Target:
A 784168
T21750
Synonym:
Target:
(R)-(+)-Docosahexaenyl-1'-Hydroxy-2'-Propylamide
T38028
Synonym:
Target:
Tat-AKAP79 (326-336) TFA
T83728
Synonym: Tat-A-kinase Anchor Protein 79 (326-336)
Target:
Cat No. Product Name Synonyms Targets
TN1377 α-Spinasterol alpha-Spinasterol COX , Antibacterial , TRP/TRPV Channel
α-Spinasterol is a transient receptor potential vanilloid 1 (TRPV1) antagonist, has anti-inflammatory, antidepressant, antioxidant and antinociceptive effects. α-Spinasterol inhibits COX-1 andCOX-2 activities with IC50 v...
T2163 Dihydrocapsaicin CCRIS1589,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide Others , TRP/TRPV Channel
Dihydrocapsaicin (CCRIS1589) is isolated from Capsicum fruit. Capsaicin is the primary active component of the heat and pain-eliciting lipid soluble fraction of the Capsicum pepper. Like capsaicin, dihydrocapsaicin is an...

Natural Products

α-Spinasterol
TN1377
Synonym: alpha-Spinasterol
Target: COX, Antibacterial, TRP/TRPV Channel
Dihydrocapsaicin
T2163
Synonym: CCRIS1589,6,7-Dihydrocapsaicin,8-Methyl-N-vanillylnonanamide
Target: Others, TRP/TRPV Channel
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