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Search Result

Search Results for " oxytocin receptor "

Targets

Oxytocin Receptor Oxytocin Receptor

38

Compounds

2

Natural Products

6

Recombinant Proteins

Cat No. Product Name Synonyms Targets
T11857 LIT-001 Oxytocin Receptor
LIT-001 improves social interaction in a mouse model of autism.It is the first nonpeptide oxytocin receptor agonist with EC50 of 55 nM and Ki of 226 nM.
T5148 Atosiban acetate RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164 Oxytocin Receptor , Vasopressin Receptor
Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban acetate (RW22164) inhibits...
T12331 OT-R antagonist 2 Oxytocin receptor antagonist 2 Others
OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .
T12331L OT-R antagonist 1 Oxytocin receptor antagonist 1 Others
OT-R antagonist 1 inhibits oxytocin-evoked intracellular Ca2+ mobilization (IC50 = 8 nM). OT-R antagonist 1 is a new effective and selective nonpeptide low molecular weight OT-R antagonist.
T4996 Atosiban RWJ22164,RW22164 Oxytocin Receptor , Vasopressin Receptor
Atosiban (RW22164) is an inhibitor of the hormones oxytocin and vasopressin. It is used as an intravenous medication as a labour repressant (tocolytic) to halt premature labor. Atosiban inhibits the oxytocin-mediated rel...
T7601L Carbetocin acetate Carbetocin acetate(37025-55-1 free base) Oxytocin Receptor
Carbetocin acetate is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.
T7601 Carbetocin Oxytocin Receptor
Carbetocin is an obstetric drug used to control postpartum hemorrhage and bleeding after giving birth.
T21534L Oxytocin C-terminal tripeptide Acetate Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base) Others
Oxytocin C-terminal tripeptide Acetate is the C-terminal tripeptide of Oxytocin.Oxytocin is a mammalian neuropituitary hormone, a ligand for the oxytocin receptor.
T3347 PF3274167 PF 3274167,Cligosiban,PF-3274167 OX Receptor
PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.
T28855 SSR126768A SSR-126768A,SSR 126768A Oxytocin Receptor
SSR126768A is a novel and selective, orally active and potent oxytocin (OT) receptor antagonist with inhibitory effects on uterine contractions for the prevention of preterm labor.
T15682 L-371,257 Oxytocin Receptor , Vasopressin Receptor
L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.
TP2082L D[Cha4]-AVP acetate(500170-27-4 free base) Vasopressin Receptor
d[Cha4]-AVP acetate is a potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secre...
T23528 WAY-267464 Others
oxytocin receptor (OTR) agonist
T23441 TC OT 39 Others
oxytocin receptor partial agonist
T11502 Epelsiban GSK 557296 Others
Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).
T69504 Barusiban
Barusiban is an oxytocin receptor antagonist.
T25902 Ota-vasotocin OVTA
Ota-vasotocin is a ligand utilized in quantitative receptor autoradiography for oxytocin receptors.
T31647 Epelsiban besylate GSK-557296B,GSK557296B
Epelsiban Besylate is an oral drug that is a highly selective anamol oxytocin receptor antagonist.
T24292 L 366948 L366,948,L-366948,L-366,948,L 366,948,L366948
L 366948 is an antagonist of the oxytocin receptor.
T79172 PF-06655075 Oxytocin Receptor
PF-06655075 is a novel, non-brain-penetrant oxytocin receptor agonist that demonstrates enhanced selectivity for the oxytocin receptor and substantially improved pharmacokinetic stability. This compound serves as a tool ...
T11794 L-368,899 hydrochloride Others
L-368,899 hydrochloride, used as a tocolytic agent, is a potent, selective, orally bioavailable, non-peptide oxytocin receptor antagonist, with IC50s of 8.9 nM and 26 nM for rat uterus and human uterus oxytocin receptor,...
T12904 SHR1653 Others
SHR1653 is a highly potent, selective and brain penetrated antagonist of oxytocin receptor (OTR)(IC50 of 15 nM for hOTR).
T26602 ALS-I-41
ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.
T28018 Merotocin FE202767,FE 202767,FE-202767
Merotocin is a potent and highly selective peptidic agonist of the oxytocin receptor.
T80140 (Val3,Pro8)-Oxytocin Oxytocin Receptor
(Val3,Pro8)-Oxytocin functions primarily as a Gq-dependent pathway agonist and exhibits secondary activity as a reduced efficacy agonist for β-arrestin recruitment and receptor-mediated endocytosis at the oxytocin recept...
T76265 (Thr4,Gly7)-Oxytocin
(Thr4,Gly7)-Oxytocin, an analogue of Oxytocin and a specific OT receptor agonist, not only activates TRPV1 channels to excite subicular neurons but also reduces the activity of potassium (K+) channels. [1] [2].
T80136 Val9-Oxytocin Vasopressin Receptor
Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.
T80126 (d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin Oxytocin Receptor
(d(CH2)51,Tyr(Me)2, Orn8)-Oxytocin (OVT) is an antagonist of the oxytocin receptor that finds application in the study of neurological diseases [1].
T24370 L-368899 free base L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899
L-368899 is a non-peptide and orally active antagonist of oxytocin receptor (IC50: 8.9 nM). It displays 40-fold selectivity over vasopressin V1a and V2 receptors (IC50: 370 and 570 nM respectively).
T81501 PF-06655075 TFA Oxytocin Receptor
PF-06655075 (TFA) is the trifluoroacetic acid (TFA) salt of PF-06655075, a novel, non-brain-penetrant oxytocin receptor agonist that exhibits enhanced selectivity for the oxytocin receptor and improved pharmacokinetic st...
T76590 (d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
(D(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin, serving as an oxytocin receptor antagonist, effectively nullifies the augmentation of inhibitory postsynaptic currents in CA1 pyramidal neurons by oxytocin [1].
T70570 Erlosiban
Erlosiban, also known as OBE001, is a novel, orally active nonpeptide oxytocin receptor antagonist under development for the treatment of preterm labor and improvement in embryo implantation and pregnancy rate in assiste...
TP1927 D[Leu4,Lys8]-VP
Selective vasopressin V1B receptor agonist (Ki values are 0.16, 64, 100 and 3800 nM for V1B, oxytocin, V2 and V1A receptors respectively). Displays weak antidiuretic, vasopressor and in vitro oxytocic activities.
TP2082 D[Cha4]-AVP
Potent and selective human vasopressin V1B receptor agonist (Ki values are 1.2, 151, 240 and 750 nM for V1B, V1A, Oxytocin and V2 receptors respectively). Stimulates ACTH and corticosterone secretion and exhibits negligi...
TP2136 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Selective vasopressin V1A receptor antagonist. Inhibits vasopressin and oxytocin-induced increases in intracellular calcium concentrations in vitro (IC50 values are 5 and 30 nM respectively). Exhibits potent and prolonge...
T11856 LIT-001 free base Others
LIT-001 free base improves social interaction in a mouse model of autism. LIT-001 free base is the first nonpeptide oxytocin receptor (OT-R) agonist (EC50=55 nM; Ki=226 nM).
T79173 PF-06478939 Oxytocin Receptor
PF-06478939 is a peptide that functions as an agonist at the oxytocin (OT) receptor and vasopressin receptor without crossing the blood-brain barrier. It exhibits EC50 values of 0.01 nM at the OT receptor and 0.078 nM at...
T75933 D[Cha4]-AVP TFA
d[Cha4]-AVP TFA is a potent and selective agonist for the vasopressin (AVP) V1b receptor, displaying a high affinity with a K i of 1.2 nM. It exhibits greater selectivity for the V1b receptor over the V1a receptor, V2 re...

Compounds

LIT-001
T11857
Synonym:
Target: Oxytocin Receptor
Atosiban acetate
T5148
Synonym: RW22164,Atosiban acetate (90779-69-4 free base),RWJ22164
Target: Oxytocin Receptor, Vasopressin Receptor
OT-R antagonist 2
T12331
Synonym: Oxytocin receptor antagonist 2
Target: Others
OT-R antagonist 1
T12331L
Synonym: Oxytocin receptor antagonist 1
Target: Others
Atosiban
T4996
Synonym: RWJ22164,RW22164
Target: Oxytocin Receptor, Vasopressin Receptor
Carbetocin acetate
T7601L
Synonym: Carbetocin acetate(37025-55-1 free base)
Target: Oxytocin Receptor
Carbetocin
T7601
Synonym:
Target: Oxytocin Receptor
Oxytocin C-terminal tripeptide Acetate
T21534L
Synonym: Oxytocin C-terminal tripeptide Acetate(2002-44-0 Free base)
Target: Others
PF3274167
T3347
Synonym: PF 3274167,Cligosiban,PF-3274167
Target: OX Receptor
SSR126768A
T28855
Synonym: SSR-126768A,SSR 126768A
Target: Oxytocin Receptor
L-371,257
T15682
Synonym:
Target: Oxytocin Receptor, Vasopressin Receptor
d[Cha4]-AVP acetate(500170-27-4 free base)
TP2082L
Synonym:
Target: Vasopressin Receptor
WAY-267464
T23528
Synonym:
Target: Others
TC OT 39
T23441
Synonym:
Target: Others
Epelsiban
T11502
Synonym: GSK 557296
Target: Others
Barusiban
T69504
Synonym:
Target:
Ota-vasotocin
T25902
Synonym: OVTA
Target:
Epelsiban besylate
T31647
Synonym: GSK-557296B,GSK557296B
Target:
L 366948
T24292
Synonym: L366,948,L-366948,L-366,948,L 366,948,L366948
Target:
PF-06655075
T79172
Synonym:
Target: Oxytocin Receptor
L-368,899 hydrochloride
T11794
Synonym:
Target: Others
SHR1653
T12904
Synonym:
Target: Others
ALS-I-41
T26602
Synonym:
Target:
Merotocin
T28018
Synonym: FE202767,FE 202767,FE-202767
Target:
(Val3,Pro8)-Oxytocin
T80140
Synonym:
Target: Oxytocin Receptor
(Thr4,Gly7)-Oxytocin
T76265
Synonym:
Target:
Val9-Oxytocin
T80136
Synonym:
Target: Vasopressin Receptor
(d(CH2)51,Tyr(Me)2,Orn8)-Oxytocin
T80126
Synonym:
Target: Oxytocin Receptor
L-368899 free base
T24370
Synonym: L 368899,L 368,899,L368,899,L-368899,L368899,L-368,899
Target:
PF-06655075 TFA
T81501
Synonym:
Target: Oxytocin Receptor
(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
T76590
Synonym:
Target:
Erlosiban
T70570
Synonym:
Target:
d[Leu4,Lys8]-VP
TP1927
Synonym:
Target:
d[Cha4]-AVP
TP2082
Synonym:
Target:
(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
TP2136
Synonym:
Target:
LIT-001 free base
T11856
Synonym:
Target: Others
PF-06478939
T79173
Synonym:
Target: Oxytocin Receptor
d[Cha4]-AVP TFA
T75933
Synonym:
Target:
Cat No. Product Name Synonyms Targets
T5145 Oxytocin acetate Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base) Oxytocin Receptor
Oxytocin acetate (α-Hypophamine acetate) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor.
T5026 Oxytocin α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon) Oxytocin Receptor
Oxytocin (Oxytocin (Syntocinon)) is a mammalian neurohypophysial hormone, a ligand of oxytocin receptor.

Natural Products

Oxytocin acetate
T5145
Synonym: Oxytocic hormone acetate,α-Hypophamine acetate,Oxytocin acetate (50-56-6 free base)
Target: Oxytocin Receptor
Oxytocin
T5026
Synonym: α-Hypophamine,Oxytocic hormone,Oxytocin (Syntocinon)
Target: Oxytocin Receptor

Recombinant Proteins

Species：
Human (4)
Bovine (2)
Expression System：
E. coli (3)
Yeast (2)
HEK293 (1)
Tag：
N-terminal 6xHis-tagged (3)
N-terminal 10xHis-SUMO-tagged and C-terminal Myc-tagged (1)
N-terminal 6xHis-Myc-tagged (1)
N-terminal 6xHis-SUMO-tagged (1)
Cat No. Product Name Species Expression System
TMPH-01820 OXT Protein, Human, Recombinant (His) Human Yeast
Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR).
TMPH-01821 OXT Protein, Human, Recombinant (His & Myc & SUMO) Human E. coli
Neurophysin 1 specifically binds oxytocin.; Oxytocin causes contraction of the smooth muscle of the uterus and of the mammary gland. Acts by binding to oxytocin receptor (OXTR).
TMPH-00279 Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (His) Bovine Yeast
Paracrine hormone primarily responsible for maternal recognition of pregnancy. Interacts with endometrial receptors, probably type I interferon receptors, and blocks estrogen receptor expression, preventing the estrogen-...
TMPH-00278 Interferon tau-1/IFNT1 Protein, Bovine, Recombinant (E. coli, His) Bovine E. coli
Paracrine hormone primarily responsible for maternal recognition of pregnancy. Interacts with endometrial receptors, probably type I interferon receptors, and blocks estrogen receptor expression, preventing the estrogen-...
TMPH-01794 NR2F6 Protein, Human, Recombinant (His & Myc) Human HEK293
Transcription factor predominantly involved in transcriptional repression. Binds to promoter/enhancer response elements that contain the imperfect 5'-AGGTCA-3' direct or inverted repeats with various spacings which are a...
TMPH-01795 NR2F6 Protein, Human, Recombinant (His & SUMO) Human E. coli
Transcription factor predominantly involved in transcriptional repression. Binds to promoter/enhancer response elements that contain the imperfect 5'-AGGTCA-3' direct or inverted repeats with various spacings which are a...
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