Home Tools
Log in
Products Inhibitors Libraries Recombinant Proteins Kits Services Contact Us
Cart
Peptides Monoclonal Antibodies Dye Reagents PROTAC Virtual Screening TargetMol Kits Cell Counting Kit-8 (CCK-8) Inhibitor Cocktails Natural Products Phenols Alkaloids Flavonoids
Inhibitors Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK
Membrane transporter/Ion channel Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Compound Libraries Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD Drug-like Compound Libraries Fragment Libraries Custom Compound Library
Signaling Pathways Angiogenesis Apoptosis Autophagy Cell Cycle/Checkpoint Chromatin/Epigenetic Cytoskeletal Signaling
DNA Damage/DNA Repair Endocrinology/Hormones GPCR/G Protein Immunology/Inflammation JAK/STAT signaling MAPK Membrane transporter/Ion channel
Metabolism Microbiology/Virology Neuroscience NF-Κb oxidation-reduction PI3K/Akt/mTOR signaling Proteases/Proteasome
Stem Cells Tyrosine Kinase/Adaptors Ubiquitination PROTAC Others
Focused Bioactive Libraries General Bioactive Libraries Approved / Repurposing Disease Focused Target / Pathway Focused Characteristic Bioactive Libraries
Natural Product Libraries Natural Product Library for HTS Characteristic Natural Product Libraries Natural Product Derivatives Libraries Natural Product Library for CADD
Drug-like Compound Libraries Compound Libraries for HTS/HCS
Fragment Libraries General Fragment Libraries Characteristic Fragment Libraries Custom Compound Library
TargetMol
Cytokines and Growth Factors •   Cytokines •   Growth Factors Receptor Proteins •   Fc Receptors •   Cytokines and Growth Factor Receptors
CD Proteins •   T Cell CD Proteins •   B Cell CD Proteins Immune Checkpoint Proteins •   Co-inhibitory Immune Checkpoint Proteins •   Co-stimulatory Immune Checkpoint Proteins
CAR-T Therapy Target Proteins •   Hematologic Malignancies Target Proteins •   Solid Tumors Target Proteins Enzymes •   Oxidoreductases,EC 1 •   Transferases,EC 2
Viral Proteins •   Coronavirus (CoV) Proteins •   Influenza Proteins Fluorescent Proteins Others

Search Result

Search Results for " neuropeptide y receptor "

Targets

Neuropeptide Y Receptor Neuropeptide Y Receptor

55

Compounds

2

Recombinant Proteins

Cat No. Product Name Synonyms Targets
TP2206 [Leu31,Pro34]-Neuropeptide Y (porcine) Neuropeptide Y Receptor
High affinity neuropeptide Y Y1 receptor agonist
T23094 NTNCB hydrochloride Others , Neuropeptide Y Receptor
NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.
TQ0286 MK-0557 Neuropeptide Y Receptor
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
T8963 CYM2503 Neuropeptide Y Receptor
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orthosteric galanin binding site of the receptor (as measured by ...
T10539 BIBO3304 TFA Neuropeptide Y Receptor
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 receptor).
T17222 Velneperit S2367 Neuropeptide Y Receptor
Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
T5587 CGP71683 hydrochloride CGP71683A Neuropeptide Y Receptor
CGP71683 hydrochloride (CGP71683A) is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes.
TP1380 Galanin (1-16), mouse, porcine, rat Neuropeptide Y Receptor
Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.
T1997 JNJ-31020028 JNJ 31020028 Neuropeptide Y Receptor
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold selectivity for Y2 versus human Y1/Y4/Y5 receptors.
T74350 Neuropeptide Y Y1 receptor antagonist 1
Neuropeptide Y Y1 receptor antagonist 1 (compound 39), a fluorescent probe, serves as a powerful antagonist against the neuropeptide Y Y1 receptor (Y1R), exhibiting a Kᵢ value of 0.19 nM [1]. It should be stored in condi...
T5455 HT-2157 SNAP37889,SNAP-37889 Neuropeptide Y Receptor
HT-2157 (SNAP-37889) is a selective, high-affinity competitive antagonist of the galanin-3 receptor (Gal3), demonstrating effective inhibition of this target.
TP1059 Peptide YY (PYY) (3-36), human Peptide YY (3-36) Neuropeptide Y Receptor
Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.
T8456 GALNON Neuropeptide Y Receptor
Galnon is a galanin receptor agonist, improves intrinsic cortical bone tissue properties
T12895 SHA 68 Neuropeptide Y Receptor
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respectively).
T23087 NPY 5RA972 Neuropeptide Y Receptor
neuropeptide Y Y5 receptor antagonist
TP1984L [D-Trp34]-Neuropeptide Y Acetate [D-Trp34]-Neuropeptide Y Acetate (153549-84-9 Free base) Neuropeptide Y Receptor
[D-Trp34]-Neuropeptide Y Acetate is a potent and selective agonist of neuropeptide Y (NPY) Y5 receptor. [D-Trp34]-Neuropeptide acetate Y is a significantly less potent agonist at the NPY Y1, Y2, Y4, and y6 receptors. [D-...
T21611L BWX 46 Acetate BWX 46 Acetate(172997-92-1 Free base) Neuropeptide Y Receptor
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.
T23349 SF 11 Others
SF 11 is a potent and brain penetrant neuropeptide Y Y2 receptor antagonist with IC50 of 199 nM. Antidepressant-like activity
TP1137L Pancreatic Polypeptide (human) acetate Neuropeptide Y Receptor
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.
T15679 L 152804 Neuropeptide Y Receptor
L 152804 is a specific antagonist of the neuropeptide Y Y5 receptor and modulates food intake and energy expenditure thus causing weight loss in diet-induced obese mice.
T26801 BIBP3226 BIBP 3226,BIBP-3226
BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.
T36447 Neuropeptide Y 13-36 (porcine)
Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.
T27345 FMS586 FMS-586,FMS 586
FMS586 is a selective antagonist of neuropeptide Y Y5 receptor with oral activity.
T23287 S 25585 Others
S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.
T22935 LU AA33810 Others
LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.
T36445 Neuropeptide Y (3-36) (human, rat)
Neuropeptide Y (3-36) (human, rat) is a metabolite of neuropeptide Y (NPY) generated by dipeptidyl peptidase-4 (DPP4). Known as a selective Y2 receptor agonist, Neuropeptide Y (3-36) (human, rat) effectively reduces the ...
TP1081 Neuropeptide Y (13-36), amide, human Neuropeptide Y (13-36), human
Neuropeptide Y (13-36), amide, human is a neuropeptide Y receptor agonist.
T26008 PYX 2 PYX2,PYX-2
PYX 2 is used as a neuropeptide Y receptor antagonist.
T76355 Neuropeptide Y (3-36) (porcine)
Neuropeptide Y (3-36) (porcine) acts as an agonist for the Y2 subtype of the neuropeptide Y (NPY) receptor, effectively stimulating feeding behavior in rats. This compound exhibits high selectivity for the Y2 receptor co...
T10921 CYM 9484 Others
CYM 9484 is a selective and potent neuropeptide Y (NPY) Y2 receptor antagonist with IC50 value of 19 nM.
T10540 BIBP3226 TFA Others
BIBP3226 TFA is an effective and selective antagonist of neuropeptide Y Y1 (NPY Y1) and neuropeptide FF (NPFF) receptor (Kis: 1.1, 79, and 108 nM for rNPY Y1, hNPFF2, and rNPFF).
T14572 BIIE-0246 AR-H 053591 Others
BIIE-0246 is a potent and highly selective non-peptide neuropeptide Y (NPY) Y2 receptor antagonist. With an IC50 of 15 nM.
T10514 FR252384 Others
FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).
T37528 TBPC
Positive allosteric modulator of neuropeptide Y receptor 4 (Y4R). Potentiates Y4R response to pancreatic polypeptide (PP), neuropeptide Y (NPY) and peptide YY (PYY) (EC50 values are 0.03, 0.4 and 0.5 nM respectively). Sh...
T22608 BMS 193885 BMS193885 Neuropeptide Y Receptor
BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.
TP1985 [Leu31,Pro34]-Neuropeptide Y(human,rat) [Leu31,Pro34]-Neuropeptide Y (human, rat)
High affinity neuropeptide Y Y1 receptor agonist (Ki = 0.39 nM). Also shows affinity for Y4 and Y5 receptors.
T75912 [Leu31,Pro34]-Neuropeptide Y(human,rat) TFA
[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA acts as a specific agonist for the neuropeptide Y Y1 receptor, while also activating receptors Y4 and Y5. This compound is known to elevate blood pressure in anesthetized rats ...
T75911 [D-Trp34]-Neuropeptide Y TFA
[D-Trp34]-Neuropeptide Y TFA acts as a potent and selective agonist for the neuropeptide Y (NPY) Y5 receptor, demonstrating significantly lower potency at the NPY Y1, Y2, Y4, and Y6 receptors. It has been observed to sig...
T69621 BIIE-0246 HCl
BIIE-0246 is a potent, selective and competitive non-peptide antagonist for the neuropeptide Y Y2 receptor. BIIE-0246 displays > 650-fold selectivity over Y1, Y4 and Y5 receptors.
T76357 Neuropeptide Y (18-36) (porcine)
Neuropeptide Y (18-36) (porcine) acts as a competitive antagonist of the neuropeptide Y (NPY) cardiac receptor, effectively blocking the attachment of I-NPY to cardiac ventricular membranes. Its action is concentration-d...
T41188 BIBP 3226 trifluoroacetate
BIBP 3226 trifluoroacetate is a mixed non-peptide neuropeptide Y Y1(NPY Y1) and neuropeptide FF (NPFF) receptor antagonist (Kivalues are 1.1, 79, 108, > 1000, > 1000 and >1000 for rNPY Y1, hNPFF2, rNPFF, rNPY Y2, rNPY Y4...
T36481 BIIE 0246 hydrochloride
Potent, selective and competitive nonpeptide antagonist for the neuropeptide Y Y2 receptor (IC50 = 15 nM). Displays > 650-fold selectivity for NPY Y2 over Y1, Y4 and Y5 receptors. Active in vivo.
T12623 (R)-JNJ-31020028 Others
(R)-JNJ-31020028 is a high affinity, selective brain penetrant antagonist of neuropeptide Y Y2 receptor(pIC50 values of 8.07, 8.22 and 8.21 for human, rat, and mouse Y2 receptor, respectively).
T75730 [D-Arg25]-Neuropeptide Y (human)
[D-Arg25]-Neuropeptide Y (human) ([D-Arg25] NPY), a Y1 receptor selective agonist, plays a role in Alzheimer's disease (AD) and safeguards rat cortical neurons from β-Amyloid toxicity [1].
TP2022 GR231118 GR 231118
Potent neuropeptide Y (NPY) Y1 receptor antagonist (pA2 = 10 and 10.5 at rY1 and hY1, receptors respectively). Also a potent and selective NPY Y4 receptor agonist (pEC50 values are 6.0, 8.6 and 6.1 for rY2, hY4 and rY5 r...
T74459 Y1R probe-1
Compound 39, also known as Y1R probe-1, is a high-affinity fluorescent probe targeting the Neuropeptide Y Y1 Receptor, with potential applications in cancer research [1].
T76423 Neuropeptide AF (cattle)
Neuropeptide AF (cattle), an amidated octadecapeptide and RFamide neuropeptide, serves as a ligand for Mas-related gene receptor A4 (MrgprA4) (Mas-related G-protein-coupled Receptor (MRGPR)) with an EC50 of approximately...
T75910 GR231118 TFA
GR231118 TFA, a neuropeptide Y C-terminus analogue, acts as a potent, competitive, and relatively selective antagonist at the human neuropeptide YY receptor, exhibiting a pKi of 10.4. It serves as a strong agonist at the...
T15620 JNJ-5207787 Others
JNJ-5207787 is a penetrates the blood-brain barrier neuropeptide Y Y2 receptor (Y2) antagonist. It is >100-fold selective versus human Y1, Y4, and Y5 receptors. JNJ-5207787 suppresses the binding of peptide YY with pIC50...
TP1963 [cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide
Potent, selective peptide agonist for the neuropeptide Y Y5 receptor (IC50 values for inhibition of NPY binding to human Y5, Y1, Y2 and Y4 receptors are 0.24, 530, > 500, and 51 nM respectively, Ki at Y5 = 0.1 - 0.15 nM)...

Compounds

[Leu31,Pro34]-Neuropeptide Y (porcine)
TP2206
Synonym:
Target: Neuropeptide Y Receptor
NTNCB hydrochloride
T23094
Synonym:
Target: Others, Neuropeptide Y Receptor
MK-0557
TQ0286
Synonym:
Target: Neuropeptide Y Receptor
CYM2503
T8963
Synonym:
Target: Neuropeptide Y Receptor
BIBO3304 TFA
T10539
Synonym:
Target: Neuropeptide Y Receptor
Velneperit
T17222
Synonym: S2367
Target: Neuropeptide Y Receptor
CGP71683 hydrochloride
T5587
Synonym: CGP71683A
Target: Neuropeptide Y Receptor
Galanin (1-16), mouse, porcine, rat
TP1380
Synonym:
Target: Neuropeptide Y Receptor
JNJ-31020028
T1997
Synonym: JNJ 31020028
Target: Neuropeptide Y Receptor
Neuropeptide Y Y1 receptor antagonist 1
T74350
Synonym:
Target:
HT-2157
T5455
Synonym: SNAP37889,SNAP-37889
Target: Neuropeptide Y Receptor
Peptide YY (PYY) (3-36), human
TP1059
Synonym: Peptide YY (3-36)
Target: Neuropeptide Y Receptor
GALNON
T8456
Synonym:
Target: Neuropeptide Y Receptor
SHA 68
T12895
Synonym:
Target: Neuropeptide Y Receptor
NPY 5RA972
T23087
Synonym:
Target: Neuropeptide Y Receptor
[D-Trp34]-Neuropeptide Y Acetate
TP1984L
Synonym: [D-Trp34]-Neuropeptide Y Acetate (153549-84-9 Free base)
Target: Neuropeptide Y Receptor
BWX 46 Acetate
T21611L
Synonym: BWX 46 Acetate(172997-92-1 Free base)
Target: Neuropeptide Y Receptor
SF 11
T23349
Synonym:
Target: Others
Pancreatic Polypeptide (human) acetate
TP1137L
Synonym:
Target: Neuropeptide Y Receptor
L 152804
T15679
Synonym:
Target: Neuropeptide Y Receptor
BIBP3226
T26801
Synonym: BIBP 3226,BIBP-3226
Target:
Neuropeptide Y 13-36 (porcine)
T36447
Synonym:
Target:
FMS586
T27345
Synonym: FMS-586,FMS 586
Target:
S 25585
T23287
Synonym:
Target: Others
LU AA33810
T22935
Synonym:
Target: Others
Neuropeptide Y (3-36) (human, rat)
T36445
Synonym:
Target:
Neuropeptide Y (13-36), amide, human
TP1081
Synonym: Neuropeptide Y (13-36), human
Target:
PYX 2
T26008
Synonym: PYX2,PYX-2
Target:
Neuropeptide Y (3-36) (porcine)
T76355
Synonym:
Target:
CYM 9484
T10921
Synonym:
Target: Others
BIBP3226 TFA
T10540
Synonym:
Target: Others
BIIE-0246
T14572
Synonym: AR-H 053591
Target: Others
FR252384
T10514
Synonym:
Target: Others
tBPC
T37528
Synonym:
Target:
BMS 193885
T22608
Synonym: BMS193885
Target: Neuropeptide Y Receptor
[Leu31,Pro34]-Neuropeptide Y(human,rat)
TP1985
Synonym: [Leu31,Pro34]-Neuropeptide Y (human, rat)
Target:
[Leu31,Pro34]-Neuropeptide Y(human,rat) TFA
T75912
Synonym:
Target:
[D-Trp34]-Neuropeptide Y TFA
T75911
Synonym:
Target:
BIIE-0246 HCl
T69621
Synonym:
Target:
Neuropeptide Y (18-36) (porcine)
T76357
Synonym:
Target:
BIBP 3226 trifluoroacetate
T41188
Synonym:
Target:
BIIE 0246 hydrochloride
T36481
Synonym:
Target:
(R)-JNJ-31020028
T12623
Synonym:
Target: Others
[D-Arg25]-Neuropeptide Y (human)
T75730
Synonym:
Target:
GR231118
TP2022
Synonym: GR 231118
Target:
Y1R probe-1
T74459
Synonym:
Target:
Neuropeptide AF (cattle)
T76423
Synonym:
Target:
GR231118 TFA
T75910
Synonym:
Target:
JNJ-5207787
T15620
Synonym:
Target: Others
[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
TP1963
Synonym: cpp1-7-npy19-23-ala31-aib32-gln34-hpancreatic-polypeptide,[cPP1-7,NPY19-23,Ala31,Aib32,Gln34] - hPancreatic Polypeptide
Target:
1 2

Recombinant Proteins

Species：
Human (1)
Mouse (1)
Expression System：
E. coli (1)
in vitro E. coli expression system (1)
Tag：
N-terminal 10xHis-tagged (2)
Cat No. Product Name Species Expression System
TMPH-02809 NPY2R Protein, Mouse, Recombinant (His) Mouse E. coli
Receptor for neuropeptide Y and peptide YY.
TMPH-01767 NPY2R Protein, Human, Recombinant (His) Human in vitro E. coli expression system
Receptor for neuropeptide Y and peptide YY. The rank order of affinity of this receptor for pancreatic polypeptides is PYY > NPY > PYY (3-36) > NPY (2-36) > [Ile-31, Gln-34] PP > [Leu-31, Pro-34] NPY > PP, [Pro-34] PYY a...
CORPORATE
About Us Careers Privacy Notice Events & News Terms & Conditions
SUPPORT
Contact Us Worldwide Distributors Quality Control Technical Support
RESOURCE
Product Catalog Product Citations Signaling Pathways Solution Calculators
FOLLOW OUR
Social Network
Newsletter Subscription
Subscribe to receive our lastest product updates and special offers!
Corporate
Support
Resource
Products are chemical reagents for research use only and are not intended for human use. We do not sell to patients.
TargetMol
Copyright © 2015-2024 TargetMol Chemicals Inc. All rights reserved.