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GPCR/G Protein Neuropeptide Y Receptor

Neuropeptide Y Receptor

Cat No. product name
T8963 CYM2503 CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orth...
TP1930L1 Spexin acetate(1370290-58-6 free base) Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galan...
TP1937L1 RFRP-1 (human) acetate(311309-25-8 free base) RFRP-1 (human) acetate is a potent endogenous NPFF receptor agonist (EC50 values are 0.0011 and 29 nM for NPFF2 and NPFF1, respectively). Attenuates contractile...
TP1992L M40 acetate(143896-17-7 free base) M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) b...
TP1074L Neuropeptide FF acetate(99566-27-5 free base) NPFF acetate is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).
T8559 GALNON TFA(475115-35-6(free base)) Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).
T17222 Velneperit Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
T10539 BIBO3304 TFA BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recep...
T12895 SHA 68 SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respective...
TP1704 Galanin Receptor Ligand M35 TFA(142846-71-7 free base) Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).
TQ0286 MK-0557 MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
T5455 HT-2157 HT-2157 is a selective, high-affinity, competitive antagonists of galanin-3 receptor (Gal3).
T5587 CGP71683 hydrochloride CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 n...
T1997 JNJ31020028 JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold...
CYM2503
T8963CAS 1308833-36-4
CYM2503 is a positive allosteric modulator (PAM) of the GAL2 receptor that potentiates galanin-induced IP1 production in vitro. It has no affinity for the orth...
Spexin acetate(1370290-58-6 free base)
TP1930L1CAS TP1930L1
Spexin acetate is a potent galanin receptor 2/3 (GAL2/GAL3) agonist (EC50 values are 45.7 and 112.2 nM, respectively). Exhibits no significant activity at galan...
RFRP-1 (human) acetate(311309-25-8 free base)
TP1937L1CAS TP1937L1
RFRP-1 (human) acetate is a potent endogenous NPFF receptor agonist (EC50 values are 0.0011 and 29 nM for NPFF2 and NPFF1, respectively). Attenuates contractile...
M40 acetate(143896-17-7 free base)
TP1992LCAS TP1992L
M40 acetate is a potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) b...
Neuropeptide FF acetate(99566-27-5 free base)
TP1074LCAS TP1074L
NPFF acetate is an octapeptide belonging to the RF amide family. NPFF interacts with G-protein-coupled receptors NPFF (1) and NPFF (2).
GALNON TFA(475115-35-6(free base))
T8559CAS T8559
Galnon is a novel non-peptide galanin receptor agonist (GAL1 and GAL2 with Ki of 11.7 and 34.1 μM respectively).
Velneperit
T17222CAS 342577-38-2
Velneperit is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.
BIBO3304 TFA
T10539CAS 191868-14-1
BIBO3304 TFA is an effective, orally active, and selective neuropeptide Y (NPY) Y1 receptor antagonist (IC50:0.38 and 0.72 nM for the human and the rat Y1 recep...
SHA 68
T12895CAS 847553-89-3
SHA 68 is a potent and selective non-peptide antagonist of neuropeptide S receptor (NPSR)(NPSR Asn107 and NPSR Ile107 with IC50s of 22.0 and 23.8 nM, respective...
Galanin Receptor Ligand M35 TFA(142846-71-7 free base)
TP1704CAS TP1704
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).
MK-0557
TQ0286CAS 328232-95-7
MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).
HT-2157
T5455CAS 303149-14-6
HT-2157 is a selective, high-affinity, competitive antagonists of galanin-3 receptor (Gal3).
CGP71683 hydrochloride
T5587CAS 192322-50-2
CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 n...
JNJ31020028
T1997CAS 1094873-14-9
JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity(pIC50=8.07, human; pIC50=8.22, rat); it exhibits >100-fold...